8ER7
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![BU of 8er7 by Molmil](/molmil-images/mine/8er7) | FKBP12-FRB in Complex with Compound 12 | Descriptor: | (3S,5R,6R,7E,9R,10R,12R,14S,15E,17E,19E,21S,23S,26R,27R,30R,34aS)-9,27-dihydroxy-3-{(2R)-1-[(1S,3R,4R)-4-hydroxy-3-methoxycyclohexyl]propan-2-yl}-5,10,21-trimethoxy-6,8,12,14,20,26-hexamethyl-5,6,9,10,12,13,14,21,22,23,24,25,26,27,32,33,34,34a-octadecahydro-3H-23,27-epoxypyrido[2,1-c][1,4]oxazacyclohentriacontine-1,11,28,29(4H,31H)-tetrone, CHLORIDE ION, Peptidyl-prolyl cis-trans isomerase FKBP1A, ... | Authors: | Tomlinson, A.C.A, Yano, J.K. | Deposit date: | 2022-10-11 | Release date: | 2022-12-28 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (3.07 Å) | Cite: | Discovery of RMC-5552, a Selective Bi-Steric Inhibitor of mTORC1, for the Treatment of mTORC1-Activated Tumors. J.Med.Chem., 66, 2023
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7Y8C
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![BU of 7y8c by Molmil](/molmil-images/mine/7y8c) | Crystal structure of CotA laccase complexed with syringaldehyde | Descriptor: | 3,5-dimethoxy-4-oxidanyl-benzaldehyde, COPPER (II) ION, Spore coat protein A, ... | Authors: | Liu, Z.C, Xie, T, Wang, G.G. | Deposit date: | 2022-06-23 | Release date: | 2023-06-28 | Last modified: | 2023-12-20 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Molecular insights into substrate promiscuity of CotA laccase catalyzing lignin-phenol derivatives. Int.J.Biol.Macromol., 256, 2023
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7Y8B
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![BU of 7y8b by Molmil](/molmil-images/mine/7y8b) | Crystal structure of CotA laccase complexed with syringic acid | Descriptor: | 3,5-dimethoxy-4-oxidanyl-benzoic acid, COPPER (II) ION, Spore coat protein A, ... | Authors: | Liu, Z.C, Xie, T, Wang, G.G. | Deposit date: | 2022-06-23 | Release date: | 2023-06-28 | Last modified: | 2023-12-20 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Molecular insights into substrate promiscuity of CotA laccase catalyzing lignin-phenol derivatives. Int.J.Biol.Macromol., 256, 2023
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7Y5N
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![BU of 7y5n by Molmil](/molmil-images/mine/7y5n) | Structure of 1:1 PAPP-A.ProMBP complex(half map) | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Bone marrow proteoglycan, ... | Authors: | Zhong, Q.H, Chu, H.L, Wang, G.P, Zhang, C, Wei, Y, Qiao, J, Hang, J. | Deposit date: | 2022-06-17 | Release date: | 2023-01-11 | Method: | ELECTRON MICROSCOPY (3.45 Å) | Cite: | Structural insights into the covalent regulation of PAPP-A activity by proMBP and STC2. Cell Discov, 8, 2022
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7Y5Q
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![BU of 7y5q by Molmil](/molmil-images/mine/7y5q) | Structure of 1:1 PAPP-A.STC2 complex(half map) | Descriptor: | Maltose/maltodextrin-binding periplasmic protein,Pappalysin-1, Stanniocalcin-2, ZINC ION | Authors: | Zhong, Q.H, Chu, H.L, Wang, G.P, Zhang, C, Wei, Y, Qiao, J, Hang, J. | Deposit date: | 2022-06-17 | Release date: | 2023-01-11 | Method: | ELECTRON MICROSCOPY (3.8 Å) | Cite: | Structural insights into the covalent regulation of PAPP-A activity by proMBP and STC2. Cell Discov, 8, 2022
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5QKC
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![BU of 5qkc by Molmil](/molmil-images/mine/5qkc) | |
5QKS
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![BU of 5qks by Molmil](/molmil-images/mine/5qks) | |
5QL9
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![BU of 5ql9 by Molmil](/molmil-images/mine/5ql9) | |
5QLS
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![BU of 5qls by Molmil](/molmil-images/mine/5qls) | |
5QM7
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![BU of 5qm7 by Molmil](/molmil-images/mine/5qm7) | |
5QKI
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![BU of 5qki by Molmil](/molmil-images/mine/5qki) | |
5QKT
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![BU of 5qkt by Molmil](/molmil-images/mine/5qkt) | |
5QLE
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![BU of 5qle by Molmil](/molmil-images/mine/5qle) | |
5QLR
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![BU of 5qlr by Molmil](/molmil-images/mine/5qlr) | |
5QM3
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![BU of 5qm3 by Molmil](/molmil-images/mine/5qm3) | |
5QMH
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![BU of 5qmh by Molmil](/molmil-images/mine/5qmh) | |
5QMY
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![BU of 5qmy by Molmil](/molmil-images/mine/5qmy) | |
5QKM
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![BU of 5qkm by Molmil](/molmil-images/mine/5qkm) | |
5QL1
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![BU of 5ql1 by Molmil](/molmil-images/mine/5ql1) | |
5QLK
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![BU of 5qlk by Molmil](/molmil-images/mine/5qlk) | |
5QLZ
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![BU of 5qlz by Molmil](/molmil-images/mine/5qlz) | |
5QKK
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![BU of 5qkk by Molmil](/molmil-images/mine/5qkk) | |
5QKZ
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![BU of 5qkz by Molmil](/molmil-images/mine/5qkz) | |
5QLD
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![BU of 5qld by Molmil](/molmil-images/mine/5qld) | |
5QLT
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![BU of 5qlt by Molmil](/molmil-images/mine/5qlt) | |