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STREPTAVIDIN, PH 5.6, BOUND TO PEPTIDE FCHPQNT
Descriptor:	FCHPQNT, STREPTAVIDIN
Authors:	Katz, B.A.
Deposit date:	1995-03-10
Release date:	1996-04-03
Last modified:	2024-02-14
Method:	X-RAY DIFFRACTION (1.76 Å)
Cite:	Binding to protein targets of peptidic leads discovered by phage display: crystal structures of streptavidin-bound linear and cyclic peptide ligands containing the HPQ sequence Biochemistry, 34, 1995

1STS

STREPTAVIDIN DIMERIZED BY DISULFIDE-BONDED PEPTIDE FCHPQNT-NH2 DIMER
Descriptor:	FCHPQNT-NH2, STREPTAVIDIN
Authors:	Katz, B.A, Cass, R.T, Liu, B, Arze, R, Collins, N.
Deposit date:	1995-09-12
Release date:	1996-03-08
Last modified:	2024-06-05
Method:	X-RAY DIFFRACTION (1.95 Å)
Cite:	Topochemical catalysis achieved by structure-based ligand design. J.Biol.Chem., 270, 1995

1C5Y

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor:	CITRATE ANION, PROTEIN (UROKINASE-TYPE PLASMINOGEN ACTIVATOR), THIENO[2,3-B]PYRIDINE-2-CARBOXAMIDINE
Authors:	Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L.
Deposit date:	1999-12-22
Release date:	2000-12-22
Last modified:	2024-04-03
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000

1C5L

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor:	CALCIUM ION, Hirudin, SODIUM ION, ...
Authors:	Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L.
Deposit date:	1999-12-22
Release date:	2000-12-22
Last modified:	2023-11-15
Method:	X-RAY DIFFRACTION (1.47 Å)
Cite:	Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000

1C5M

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor:	PROTEIN (COAGULATION FACTOR X)
Authors:	Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L.
Deposit date:	1999-12-22
Release date:	2000-12-22
Last modified:	2023-08-09
Method:	X-RAY DIFFRACTION (1.95 Å)
Cite:	Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000

1C5N

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor:	4-IODOBENZO[B]THIOPHENE-2-CARBOXAMIDINE, CALCIUM ION, Hirudin, ...
Authors:	Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L.
Deposit date:	1999-12-22
Release date:	2000-12-22
Last modified:	2023-11-15
Method:	X-RAY DIFFRACTION (1.5 Å)
Cite:	Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000

1C5O

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor:	BENZAMIDINE, Hirudin, SODIUM ION, ...
Authors:	Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L.
Deposit date:	1999-12-22
Release date:	2000-12-22
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.9 Å)
Cite:	Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000

1C5W

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor:	4-IODOBENZO[B]THIOPHENE-2-CARBOXAMIDINE, CITRATE ANION, PROTEIN (UROKINASE-TYPE PLASMINOGEN ACTIVATOR)
Authors:	Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L.
Deposit date:	1999-12-22
Release date:	2000-12-22
Last modified:	2024-04-03
Method:	X-RAY DIFFRACTION (1.94 Å)
Cite:	Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000

1C5X

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor:	4-IODOBENZO[B]THIOPHENE-2-CARBOXAMIDINE, CITRATE ANION, PROTEIN (UROKINASE-TYPE PLASMINOGEN ACTIVATOR)
Authors:	Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L.
Deposit date:	1999-12-22
Release date:	2000-12-22
Last modified:	2024-04-03
Method:	X-RAY DIFFRACTION (1.75 Å)
Cite:	Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000

1C5Z

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor:	BENZAMIDINE, CITRATE ANION, PROTEIN (UROKINASE-TYPE PLASMINOGEN ACTIVATOR)
Authors:	Katz, B.A, Mackman, R, Luong, C, Radika, K, Martelli, A, Sprengeler, P.A, Wang, J, Chan, H, Wong, L.
Deposit date:	1999-12-22
Release date:	2000-12-22
Last modified:	2024-04-03
Method:	X-RAY DIFFRACTION (1.85 Å)
Cite:	Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem.Biol., 7, 2000

1C1O

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	CALCIUM ION, MAGNESIUM ION, SULFATE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.4 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1V

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-BENZIMIDAZOLYL)METHANE, Hirudin-2, SODIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-11-15
Method:	X-RAY DIFFRACTION (1.98 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2I

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE, CALCIUM ION, CHLORIDE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.47 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2D

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE, CALCIUM ION, MAGNESIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1P

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	(5-AMIDINO-2-BENZIMIDAZOLYL)(2-BENZIMIDAZOLYL)METHANE, CALCIUM ION, DIMETHYL SULFOXIDE, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.37 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1U

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	(5-AMIDINO-2-BENZIMIDAZOLYL)(2-BENZIMIDAZOLYL)METHANE, ACETYL HIRUDIN, ALPHA THROMBIN, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-11-15
Method:	X-RAY DIFFRACTION (1.75 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2F

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE HYDRATE, CALCIUM ION, DIMETHYL SULFOXIDE, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.7 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1S

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-BENZIMIDAZOLYL)METHANE, CALCIUM ION, PHOSPHATE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.63 Å)
Cite:	Recruiting Zn2+ to mediate potent, specific inhibition of serine proteases. J.Mol.Biol., 292, 1999

1C1R

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	(5-AMIDINO-2-BENZIMIDAZOLYL)(2-BENZIMIDAZOLYL)METHANE, CALCIUM ION, DIMETHYL SULFOXIDE, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.37 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2K

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	5-AMIDINO-BENZIMIDAZOLE, CALCIUM ION, CHLORIDE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2M

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	CALCIUM ION, MAGNESIUM ION, SULFATE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.4 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2G

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE HYDRATE, CALCIUM ION, DIMETHYL SULFOXIDE, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C2E

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE, CALCIUM ION, MAGNESIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-22
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1N

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BENZAMIDINE, CALCIUM ION, SULFATE ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-12-27
Method:	X-RAY DIFFRACTION (1.4 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

1C1W

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor:	BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANE KETONE HYDRATE, Hirudin-2, SODIUM ION, ...
Authors:	Katz, B.A, Luong, C.
Deposit date:	1999-07-21
Release date:	2000-07-26
Last modified:	2023-11-15
Method:	X-RAY DIFFRACTION (1.9 Å)
Cite:	Design of potent selective zinc-mediated serine protease inhibitors. Nature, 391, 1998

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Total results:	198
Displayed results:	25
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