5A6K
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![BU of 5a6k by Molmil](/molmil-images/mine/5a6k) | GH20C, Beta-hexosaminidase from Streptococcus pneumoniae in complex with Gal-NGT | Descriptor: | (2S,3aR,5R,6R,7R,7aR)-5-(hydroxymethyl)-2-methyl-2,3a,5,6,7,7a-hexahydro-1H-pyrano[3,2-d][1,3]thiazole-6,7-diol, GH20C | Authors: | Cid, M, Robb, C.S, Higgins, M.A, Boraston, A.B. | Deposit date: | 2015-06-26 | Release date: | 2015-09-23 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | A Second Beta-Hexosaminidase Encoded in the Streptococcus Pneumoniae Genome Provides an Expanded Biochemical Ability to Degrade Host Glycans J.Biol.Chem., 290, 2015
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5AWN
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![BU of 5awn by Molmil](/molmil-images/mine/5awn) | |
5AMU
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![BU of 5amu by Molmil](/molmil-images/mine/5amu) | IglE I39A,Y40A,V44A | Descriptor: | IGLE | Authors: | Robb, C.S, Nano, F.E, Boraston, A.B. | Deposit date: | 2015-09-01 | Release date: | 2016-10-05 | Last modified: | 2024-01-10 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | The Structure, Dimerisation and Impact on Intramacrophage Replication of Igle in Francisella Novicida To be Published
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5A55
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![BU of 5a55 by Molmil](/molmil-images/mine/5a55) | The native structure of GH101 from Streptococcus pneumoniae TIGR4 | Descriptor: | 1,2-ETHANEDIOL, CALCIUM ION, ENDO-ALPHA-N-ACETYLGALACTOSAMINIDASE, ... | Authors: | Gregg, K.J, Suits, M.D.L, Deng, L, Vocadlo, D.J, Boraston, A.B. | Deposit date: | 2015-06-16 | Release date: | 2015-09-02 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Structural Analysis of a Family 101 Glycoside Hydrolase in Complex with Carbohydrates Reveals Insights Into its Mechanism. J.Biol.Chem., 290, 2015
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5A5A
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![BU of 5a5a by Molmil](/molmil-images/mine/5a5a) | The structure of GH101 E796Q mutant from Streptococcus pneumoniae TIGR4 in complex with PNP-T-antigen | Descriptor: | 1,2-ETHANEDIOL, CALCIUM ION, CITRIC ACID, ... | Authors: | Gregg, K.J, Suits, M.D.L, Deng, L, Vocadlo, D.J, Boraston, A.B. | Deposit date: | 2015-06-16 | Release date: | 2015-09-02 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (1.75 Å) | Cite: | Structural Analysis of a Family 101 Glycoside Hydrolase in Complex with Carbohydrates Reveals Insights Into its Mechanism. J.Biol.Chem., 290, 2015
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3DT3
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![BU of 3dt3 by Molmil](/molmil-images/mine/3dt3) | Human Estrogen receptor alpha LBD with GW368 | Descriptor: | 5-(4-hydroxyphenoxy)-6-(3-hydroxyphenyl)-7-methylnaphthalen-2-ol, Estrogen receptor | Authors: | Williams, S.P, Miller, A.B. | Deposit date: | 2008-07-14 | Release date: | 2008-09-09 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Synthesis of 3-alkyl naphthalenes as novel estrogen receptor ligands. Bioorg.Med.Chem.Lett., 18, 2008
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5AN1
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![BU of 5an1 by Molmil](/molmil-images/mine/5an1) | |
5AMT
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![BU of 5amt by Molmil](/molmil-images/mine/5amt) | Intracellular growth locus protein E | Descriptor: | 1,2-ETHANEDIOL, BROMIDE ION, IGLE | Authors: | Robb, C.S, Nano, F.E, Boraston, A.B. | Deposit date: | 2015-09-01 | Release date: | 2016-10-05 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (1.62 Å) | Cite: | Cloning, Expression, Purification, Crystallization and Preliminary X-Ray Diffraction Analysis of Intracellular Growth Locus E (Igle) Protein from Francisella Tularensis Subsp. Novicida. Acta Crystallogr.,Sect.F, 66, 2010
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3B88
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![BU of 3b88 by Molmil](/molmil-images/mine/3b88) | Complex of T57A Substituted Drosophila LUSH Protein with Ethanol | Descriptor: | 2-{2-[2-2-(METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, ACETATE ION, General odorant-binding protein lush | Authors: | Jones, D.N.M, Thode, A.B. | Deposit date: | 2007-10-31 | Release date: | 2008-02-05 | Last modified: | 2021-10-20 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | The role of multiple hydrogen-bonding groups in specific alcohol binding sites in proteins: insights from structural studies of LUSH. J.Mol.Biol., 376, 2008
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3BLV
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![BU of 3blv by Molmil](/molmil-images/mine/3blv) | Yeast Isocitrate Dehydrogenase with Citrate Bound in the Regulatory Subunits | Descriptor: | CITRATE ANION, Isocitrate dehydrogenase [NAD] subunit 1, Isocitrate dehydrogenase [NAD] subunit 2 | Authors: | Taylor, A.B, Hu, G, Hart, P.J, McAlister-Henn, L. | Deposit date: | 2007-12-11 | Release date: | 2008-02-05 | Last modified: | 2023-11-15 | Method: | X-RAY DIFFRACTION (3.2 Å) | Cite: | Allosteric Motions in Structures of Yeast NAD+-specific Isocitrate Dehydrogenase. J.Biol.Chem., 283, 2008
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1UB5
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![BU of 1ub5 by Molmil](/molmil-images/mine/1ub5) | Crystal structure of Antibody 19G2 with hapten at 100K | Descriptor: | 4-(4-STYRYL-PHENYLCARBAMOYL)-BUTYRIC ACID, antibody 19G2, alpha chain, ... | Authors: | Beuscher, A.B, Wirsching, P, Lerner, R.A, Janda, K, Stevens, R.C. | Deposit date: | 2003-03-30 | Release date: | 2004-04-20 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Structure and Dynamics of Blue Fluorescent Antibody 19G2 at Blue and Violet Fluorescent Temperatures To be published
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1TTK
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![BU of 1ttk by Molmil](/molmil-images/mine/1ttk) | NMR solution structure of omega-conotoxin MVIIA, a N-type calcium channel blocker | Descriptor: | Omega-conotoxin MVIIa | Authors: | Adams, D.J, Smith, A.B, Schroeder, C.I, Yasuda, T, Lewis, R.J. | Deposit date: | 2004-06-22 | Release date: | 2004-07-06 | Last modified: | 2022-03-02 | Method: | SOLUTION NMR | Cite: | omega-conotoxin CVID inhibits a pharmacologically distinct voltage-sensitive calcium channel associated with transmitter release from preganglionic nerve terminals J.Biol.Chem., 278, 2003
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1TT3
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![BU of 1tt3 by Molmil](/molmil-images/mine/1tt3) | NMR soulution structure of omega-conotoxin [K10]MVIIA | Descriptor: | Omega-conotoxin MVIIa | Authors: | Adams, D.J, Smith, A.B, Schroeder, C.I, Yasuda, T, Lewis, R.J. | Deposit date: | 2004-06-21 | Release date: | 2004-07-06 | Last modified: | 2021-11-10 | Method: | SOLUTION NMR | Cite: | omega-conotoxin CVID inhibits a pharmacologically distinct voltage-sensitive calcium channel associated with transmitter release from preganglionic nerve terminals J.Biol.Chem., 278, 2003
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1U8E
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![BU of 1u8e by Molmil](/molmil-images/mine/1u8e) | HUMAN DIPEPTIDYL PEPTIDASE IV/CD26 MUTANT Y547F | Descriptor: | 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | Authors: | Bjelke, J.R, Christensen, J, Branner, S, Wagtmann, N, Olsen, C, Kanstrup, A.B, Rasmussen, H.B. | Deposit date: | 2004-08-05 | Release date: | 2004-08-17 | Last modified: | 2021-10-20 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Tyrosine 547 constitutes an essential part of the catalytic mechanism of dipeptidyl peptidase IV J.Biol.Chem., 279, 2004
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1TU6
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![BU of 1tu6 by Molmil](/molmil-images/mine/1tu6) | Cathepsin K complexed with a ketoamide inhibitor | Descriptor: | Cathepsin K, SULFATE ION, [1-(4-FLUOROBENZYL)CYCLOBUTYL]METHYL (1S)-1-[OXO(1H-PYRAZOL-5-YLAMINO)ACETYL]PENTYLCARBAMATE | Authors: | Barrett, D.G, Catalano, J.G, Deaton, D.N, Hassell, A.M, Long, S.T, Miller, A.B, Miller, L.R, Shewchuk, L.M, Wells-Knecht, K.J, Wright, L.L. | Deposit date: | 2004-06-24 | Release date: | 2004-09-21 | Last modified: | 2023-08-23 | Method: | X-RAY DIFFRACTION (1.75 Å) | Cite: | Potent and selective P2-P3 ketoamide inhibitors of cathepsin K with improved pharmacokinetic properties via favorable P1', P1, and/or P3 substitutions BIOORG.MED.CHEM.LETT., 14, 2004
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1UB6
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![BU of 1ub6 by Molmil](/molmil-images/mine/1ub6) | Crystal structure of Antibody 19G2 with sera ligand | Descriptor: | antibody 19G2, alpha chain, beta chain | Authors: | Beuscher, A.B, Wirsching, P, Lerner, R.A, Janda, K, Stevens, R.C. | Deposit date: | 2003-03-30 | Release date: | 2004-04-20 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (2.12 Å) | Cite: | Structure and Dynamics of Blue Fluorescent Antibody 19G2 at Blue and Violet Fluorescent Temperatures To be published
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4OTB
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![BU of 4otb by Molmil](/molmil-images/mine/4otb) | |
4OQM
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![BU of 4oqm by Molmil](/molmil-images/mine/4oqm) | Crystal structure of thymidine kinase from herpes simplex virus type 1 in complex with F-ARA-EdU | Descriptor: | 1-(2-deoxy-2-fluoro-beta-D-arabinofuranosyl)-5-ethynylpyrimidine-2,4(1H,3H)-dione, SULFATE ION, Thymidine kinase | Authors: | Pernot, L, Neef, A.B, Westermaier, Y, Perozzo, R, Luedtke, N, Scapozza, L. | Deposit date: | 2014-02-10 | Release date: | 2014-08-13 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Crystal structure of thymidine kinase from herpes simplex virus type 1 in complex with F-ARA-EdU To be Published
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4OTA
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![BU of 4ota by Molmil](/molmil-images/mine/4ota) | |
1UY4
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![BU of 1uy4 by Molmil](/molmil-images/mine/1uy4) | |
1UY3
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4OQL
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![BU of 4oql by Molmil](/molmil-images/mine/4oql) | Crystal structure of thymidine kinase from herpes simplex virus type 1 in complex with dF-EdU | Descriptor: | 2'-deoxy-5-ethynyl-2',2'-difluorouridine, SULFATE ION, Thymidine kinase | Authors: | Pernot, L, Neef, A.B, Westermaier, Y, Perozzo, R, Luedtke, N, Scapozza, L. | Deposit date: | 2014-02-10 | Release date: | 2014-08-13 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Crystal structure of thymidine kinase from herpes simplex virus type 1 in complex with dF-EdU To be Published
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4OQN
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![BU of 4oqn by Molmil](/molmil-images/mine/4oqn) | Crystal structure of thymidine kinase from herpes simplex virus type 1 in complex with EdU | Descriptor: | 2'-deoxy-5-ethynyluridine, SULFATE ION, Thymidine kinase | Authors: | Pernot, L, Neef, A.B, Westermaier, Y, Perozzo, R, Luedtke, N.W, Scapozza, L. | Deposit date: | 2014-02-10 | Release date: | 2014-08-13 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Crystal structure of thymidine kinase from herpes simplex virus type 1 in complex with EdU To be Published
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4OQX
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![BU of 4oqx by Molmil](/molmil-images/mine/4oqx) | Crystal structure of thymidine kinase from herpes simplex virus type 1 in complex with Me-ARA-EdU | Descriptor: | 1-(2-deoxy-2-methyl-beta-D-arabinofuranosyl)-5-ethynylpyrimidine-2,4(1H,3H)-dione, SULFATE ION, Thymidine kinase | Authors: | Pernot, L, Neef, A.B, Westermaier, Y, Perozzo, R, Luedtke, N, Scapozza, L. | Deposit date: | 2014-02-10 | Release date: | 2014-08-13 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Crystal structure of HSV1-TK complexed with Me-ARA-EdU To be Published
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1UY2
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![BU of 1uy2 by Molmil](/molmil-images/mine/1uy2) | |