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6Y1Z
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BU of 6y1z by Molmil
Mouse serotonin 5HT3 receptor in complex with palonosetron
Descriptor: (3~{a}~{S})-2-[(3~{S})-1-azabicyclo[2.2.2]octan-3-yl]-3~{a},4,5,6-tetrahydro-3~{H}-benzo[de]isoquinolin-1-one, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Zarkadas, E, Perot, J, Nury, H.
Deposit date:2020-02-14
Release date:2020-03-04
Last modified:2022-09-14
Method:ELECTRON MICROSCOPY (2.82 Å)
Cite:The Binding of Palonosetron and Other Antiemetic Drugs to the Serotonin 5-HT3 Receptor.
Structure, 28, 2020
6HIQ
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BU of 6hiq by Molmil
Mouse serotonin 5-HT3 receptor, serotonin-bound, I2 conformation
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5-hydroxytryptamine receptor 3A, ...
Authors:Polovinkin, L, Neumann, E, Schoehn, G, Nury, H.
Deposit date:2018-08-30
Release date:2018-11-07
Last modified:2022-09-14
Method:ELECTRON MICROSCOPY (3.2 Å)
Cite:Conformational transitions of the serotonin 5-HT3receptor.
Nature, 563, 2018
6HIN
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BU of 6hin by Molmil
Mouse serotonin 5-HT3 receptor, serotonin-bound, F conformation
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5-hydroxytryptamine receptor 3A, ...
Authors:Polovinkin, L, Neumann, E, Schoehn, G, Nury, H.
Deposit date:2018-08-30
Release date:2018-11-07
Last modified:2022-09-14
Method:ELECTRON MICROSCOPY (4.1 Å)
Cite:Conformational transitions of the serotonin 5-HT3receptor.
Nature, 563, 2018
6HIO
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BU of 6hio by Molmil
Mouse serotonin 5-HT3 receptor, serotonin-bound, I1 conformation
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5-hydroxytryptamine receptor 3A, ...
Authors:Polovinkin, L, Neumann, E, Schoehn, G, Nury, H.
Deposit date:2018-08-30
Release date:2018-11-07
Last modified:2022-09-14
Method:ELECTRON MICROSCOPY (4.2 Å)
Cite:Conformational transitions of the serotonin 5-HT3receptor.
Nature, 563, 2018
6HIS
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BU of 6his by Molmil
Mouse serotonin 5-HT3 receptor, tropisetron-bound, T conformation
Descriptor: (3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-INDOLE-3-CARBOXYLATE, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5-hydroxytryptamine receptor 3A, ...
Authors:Polovinkin, L, Neumann, E, Schoehn, G, Nury, H.
Deposit date:2018-08-30
Release date:2018-11-07
Last modified:2022-09-14
Method:ELECTRON MICROSCOPY (4.5 Å)
Cite:Conformational transitions of the serotonin 5-HT3receptor.
Nature, 563, 2018

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