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8PQN
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BU of 8pqn by Molmil
NQO1 bound to RBS-10
Descriptor: FLAVIN-ADENINE DINUCLEOTIDE, NAD(P)H dehydrogenase [quinone] 1, ~{N}-[4-[(3-methylphenyl)carbonylamino]phenyl]-5-nitro-furan-2-carboxamide
Authors:Pous, J, Jose-Duran, F, Mayor-Ruiz, C, Riera, A.
Deposit date:2023-07-11
Release date:2024-01-10
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (3.8 Å)
Cite:Discovery and Mechanistic Elucidation of NQO1-Bioactivatable Small Molecules That Overcome Resistance to Degraders.
Angew.Chem.Int.Ed.Engl., 63, 2024

222926

数据于2024-07-24公开中

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