4DG6
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![BU of 4dg6 by Molmil](/molmil-images/mine/4dg6) | Crystal structure of domains 1 and 2 of LRP6 | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Low-density lipoprotein receptor-related protein 6, PHOSPHATE ION | Authors: | Ceska, T.A, Doyle, C, Slocombe, P. | Deposit date: | 2012-01-25 | Release date: | 2012-06-13 | Last modified: | 2020-07-29 | Method: | X-RAY DIFFRACTION (2.9 Å) | Cite: | Characterization of the interaction of sclerostin with the LRP family of Wnt co-receptors To be Published
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3S7M
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![BU of 3s7m by Molmil](/molmil-images/mine/3s7m) | |
3S7L
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![BU of 3s7l by Molmil](/molmil-images/mine/3s7l) | |
6YI5
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![BU of 6yi5 by Molmil](/molmil-images/mine/6yi5) | In-situ structure of the trimeric HEF from influenza C by flexible fitting into a cryo-ET map. | Descriptor: | Hemagglutinin-esterase-fusion glycoprotein, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose | Authors: | Halldorsson, S, Rosenthal, P.B. | Deposit date: | 2020-03-31 | Release date: | 2021-03-24 | Last modified: | 2021-03-31 | Method: | ELECTRON MICROSCOPY (9.1 Å) | Cite: | In situ structure and organization of the influenza C virus surface glycoprotein. Nat Commun, 12, 2021
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6VBC
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6VBM
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![BU of 6vbm by Molmil](/molmil-images/mine/6vbm) | Crystal structure of a S310A mutant of PBP2 from Neisseria gonorrhoeae | Descriptor: | PHOSPHATE ION, Probable peptidoglycan D,D-transpeptidase PenA | Authors: | Singh, A, Davies, C. | Deposit date: | 2019-12-19 | Release date: | 2020-04-15 | Last modified: | 2023-10-11 | Method: | X-RAY DIFFRACTION (1.71 Å) | Cite: | Mutations in Neisseria gonorrhoeae penicillin-binding protein 2 associated with extended-spectrum cephalosporin resistance create an energetic barrier against acylation via restriction of protein dynamics J.Biol.Chem., 2020
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6VBD
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![BU of 6vbd by Molmil](/molmil-images/mine/6vbd) | |
6VBL
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![BU of 6vbl by Molmil](/molmil-images/mine/6vbl) | |
6HKG
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![BU of 6hkg by Molmil](/molmil-images/mine/6hkg) | Structure of FISW84 Fab Fragment | Descriptor: | FISW84 Fab Fragment Heavy Chain, FISW84 Fab Fragment Light Chain, SULFATE ION | Authors: | Benton, D.J, Rosenthal, P.B. | Deposit date: | 2018-09-06 | Release date: | 2018-09-26 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.87 Å) | Cite: | Influenza hemagglutinin membrane anchor. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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6HJN
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![BU of 6hjn by Molmil](/molmil-images/mine/6hjn) | Structure of Influenza Hemagglutinin ectodomain (A/duck/Alberta/35/76) | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, Hemagglutinin, ... | Authors: | Benton, D.J, Rosenthal, P.B. | Deposit date: | 2018-09-04 | Release date: | 2018-09-26 | Last modified: | 2020-07-29 | Method: | ELECTRON MICROSCOPY (3.3 Å) | Cite: | Influenza hemagglutinin membrane anchor. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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6HJQ
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![BU of 6hjq by Molmil](/molmil-images/mine/6hjq) | |
6HJP
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![BU of 6hjp by Molmil](/molmil-images/mine/6hjp) | |
6HJR
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![BU of 6hjr by Molmil](/molmil-images/mine/6hjr) | |
3OOZ
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![BU of 3ooz by Molmil](/molmil-images/mine/3ooz) | Bace1 in complex with the aminohydantoin Compound 102 | Descriptor: | (5R)-2-amino-5-[4-(difluoromethoxy)phenyl]-5-[4-fluoro-3-(5-fluoropent-1-yn-1-yl)phenyl]-3-methyl-3,5-dihydro-4H-imidazol-4-one, Beta-secretase 1 | Authors: | Olland, A.M. | Deposit date: | 2010-08-31 | Release date: | 2011-08-31 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Design and Synthesis of Aminohydantoins as Potent and Selective Human beta-Secretase (BACE1) Inhibitors with Enhanced Brain Permeability Bioorg.Med.Chem.Lett., 20, 2010
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2QU3
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![BU of 2qu3 by Molmil](/molmil-images/mine/2qu3) | BACE1 with Compound 2 | Descriptor: | Beta-secretase 1, N-[amino(imino)methyl]-2-[2-(2-chlorophenyl)-4-(4-propoxyphenyl)-3-thienyl]acetamide | Authors: | Chopra, R. | Deposit date: | 2007-08-03 | Release date: | 2008-08-05 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Thiophene substituted acylguanidines as BACE1 inhibitors. Bioorg.Med.Chem.Lett., 17, 2007
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3SLS
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![BU of 3sls by Molmil](/molmil-images/mine/3sls) | Crystal Structure of human MEK-1 kinase in complex with UCB1353770 and AMPPNP | Descriptor: | 2-[(2-fluoro-4-iodophenyl)amino]-5,5-dimethyl-8-oxo-N-[(3R)-piperidin-3-yl]-5,6,7,8-tetrahydro-4H-thieno[2,3-c]azepine-3-carboxamide, Dual specificity mitogen-activated protein kinase kinase 1, MAGNESIUM ION, ... | Authors: | Meier, C, Ceska, T.A. | Deposit date: | 2011-06-25 | Release date: | 2012-02-29 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Engineering human MEK-1 for structural studies: A case study of combinatorial domain hunting. J.Struct.Biol., 177, 2012
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5V30
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![BU of 5v30 by Molmil](/molmil-images/mine/5v30) | Crystal structure of the sensor domain of the transcriptional regulator HcpR from Porphyromonas Gingivalis | Descriptor: | GLYCEROL, SULFATE ION, Transcriptional regulator | Authors: | Musayev, F.N, Belvin, B.R, Escalante, C.R, Turner, J, Lewis, J.P. | Deposit date: | 2017-03-06 | Release date: | 2018-06-13 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (3.15 Å) | Cite: | Nitrosative stress sensing in Porphyromonas gingivalis: structure of and heme binding by the transcriptional regulator HcpR. Acta Crystallogr D Struct Biol, 75, 2019
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