5ZWZ
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5ZWX
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7DCD
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7V4Q
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7V4R
| The crystal structure of KFDV NS3H bound with Pi | Descriptor: | NICKEL (II) ION, PHOSPHATE ION, Serine protease NS3 | Authors: | Zhang, C.Y, Jin, T.C. | Deposit date: | 2021-08-14 | Release date: | 2022-08-17 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Kyasanur Forest disease virus NS3 helicase: Insights into structure, activity, and inhibitors. Int.J.Biol.Macromol., 2023
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6BOJ
| Crystal Structure of the PDE4D Catalytic Domain and UCR2 Regulatory Helix with BPN5004 | Descriptor: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(4-{[2-(3-chlorophenyl)-6-ethylpyrimidin-4-yl]methyl}phenyl)acetamide, CHLORIDE ION, ... | Authors: | Fox III, D, Fairman, J.W, Gurney, M.E. | Deposit date: | 2017-11-20 | Release date: | 2018-08-22 | Last modified: | 2024-03-13 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Memory enhancing effects of BPN14770, an allosteric inhibitor of phosphodiesterase-4D, in wild-type and humanized mice. Neuropsychopharmacology, 43, 2018
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7Y7M
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7YRH
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7YRF
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7YV7
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7YV2
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7YMS
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7RX6
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7RX7
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7RX8
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5W93
| p130Cas complex with paxillin LD1 | Descriptor: | Breast cancer anti-estrogen resistance protein 1, Paxillin | Authors: | Miller, D.J, Zheng, J.J. | Deposit date: | 2017-06-22 | Release date: | 2017-09-06 | Last modified: | 2023-10-04 | Method: | X-RAY DIFFRACTION (2.001 Å) | Cite: | Structural and functional insights into the interaction between the Cas family scaffolding protein p130Cas and the focal adhesion-associated protein paxillin. J. Biol. Chem., 292, 2017
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4LGH
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4LGG
| Structure of 3MB-PP1 bound to analog-sensitive Src kinase | Descriptor: | 1-tert-butyl-3-(3-methylbenzyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine, Proto-oncogene tyrosine-protein kinase Src | Authors: | Lopez, M.S, Dar, A.C, Shokat, K.M. | Deposit date: | 2013-06-27 | Release date: | 2013-08-07 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (2.41 Å) | Cite: | Structure-guided inhibitor design expands the scope of analog-sensitive kinase technology. Acs Chem.Biol., 8, 2013
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8JJC
| Tubulin-Y62 | Descriptor: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 4-(6,7-dimethoxy-3,4-dihydro-1~{H}-isoquinolin-2-yl)-6-(3-methoxyphenyl)pyrimidin-2-amine, CALCIUM ION, ... | Authors: | Yang, J. | Deposit date: | 2023-05-30 | Release date: | 2024-03-27 | Method: | X-RAY DIFFRACTION (2.76 Å) | Cite: | Structure-based design and synthesis of BML284 derivatives: A novel class of colchicine-site noncovalent tubulin degradation agents. Eur.J.Med.Chem., 268, 2024
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8JJB
| Crystal structure of T2R-TTL-Y61 complex | Descriptor: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, CHLORIDE ION, ... | Authors: | Yang, J. | Deposit date: | 2023-05-30 | Release date: | 2024-03-27 | Method: | X-RAY DIFFRACTION (2.68 Å) | Cite: | Structure-based design and synthesis of BML284 derivatives: A novel class of colchicine-site noncovalent tubulin degradation agents. Eur.J.Med.Chem., 268, 2024
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7ESV
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7ESQ
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7ESP
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7ESO
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4Q65
| Structure of the E. coli Peptide Transporter YbgH | Descriptor: | Dipeptide permease D | Authors: | Zhang, C, Zhao, Y, Mao, G, Liu, M, Wang, X. | Deposit date: | 2014-04-21 | Release date: | 2014-08-13 | Last modified: | 2024-05-29 | Method: | X-RAY DIFFRACTION (3.4 Å) | Cite: | Crystal structure of the E. coli peptide transporter YbgH. Structure, 22, 2014
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