8CKH
| Crystal structure of IspE from Klebsiella pneumoniae | Descriptor: | 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER | Authors: | Hamid, R. | Deposit date: | 2023-02-15 | Release date: | 2024-02-28 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Crystal structure of IspE from Klebsiella pneumoniae To Be Published
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8A29
| Apo 1-deoxy-D-xylulose 5-phosphate synthase from Pseudomonas aeruginosa | Descriptor: | 1-deoxy-D-xylulose-5-phosphate synthase, CALCIUM ION, CHLORIDE ION, ... | Authors: | Hamid, R, Adam, S, Lacour, A, Monjas, L, Hirsch, A. | Deposit date: | 2022-06-02 | Release date: | 2023-06-14 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | 1-deoxy-D-xylulose-5-phosphate synthase from Pseudomonas aeruginosa and Klebsiella pneumoniae reveals conformational changes upon cofactor binding. J.Biol.Chem., 299, 2023
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8A4D
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8A45
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8A5K
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8QCO
| E.coli IspE in complex with a ligand (3) | Descriptor: | 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, ADENOSINE-5'-DIPHOSPHATE, ~{N}-[3-(4-azanyl-2-oxidanylidene-1~{H}-pyrimidin-5-yl)prop-2-ynyl]cyclopentanesulfonamide | Authors: | Hamid, R. | Deposit date: | 2023-08-28 | Release date: | 2024-09-11 | Method: | X-RAY DIFFRACTION (1.55 Å) | Cite: | E.coli IspE in complex with a ligand (3) To Be Published
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8QC7
| New monoclinic EcIspE | Descriptor: | 4-DIPHOSPHOCYTIDYL-2-C-METHYL-D-ERYTHRITOL, 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, ADENOSINE-5'-DIPHOSPHATE, ... | Authors: | Hamid, R. | Deposit date: | 2023-08-25 | Release date: | 2024-09-11 | Method: | X-RAY DIFFRACTION (2.03 Å) | Cite: | New monoclinic EcIspE To Be Published
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8QCN
| E.coli IspE in complex with a ligand (2) | Descriptor: | 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, ADENOSINE-5'-DIPHOSPHATE, ~{N}-[3-(4-azanyl-2-oxidanylidene-1~{H}-pyrimidin-5-yl)prop-2-ynyl]cyclopropanesulfonamide | Authors: | Hamid, R. | Deposit date: | 2023-08-27 | Release date: | 2024-09-11 | Method: | X-RAY DIFFRACTION (1.86 Å) | Cite: | E.coli IspE in complex with a ligand (2) To Be Published
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8QCC
| E.coli IspE in complex with a ligand (1) | Descriptor: | 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... | Authors: | Hamid, R. | Deposit date: | 2023-08-25 | Release date: | 2024-09-11 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | E.coli IspE in complex with a ligand (1) To Be Published
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8BZX
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3SFK
| Crystal structure of Plasmodium falciparum dihydroorotate dehydrogenase bound with Inhibitor DSM267 | Descriptor: | 2-(1,1-difluoroethyl)-5-methyl-N-[4-(trifluoromethyl)phenyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine, Dihydroorotate dehydrogenase (quinone), mitochondrial, ... | Authors: | Deng, X, Phillips, M. | Deposit date: | 2011-06-13 | Release date: | 2011-07-06 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.95 Å) | Cite: | Structure-Guided Lead Optimization of Triazolopyrimidine-Ring Substituents Identifies Potent Plasmodium falciparum Dihydroorotate Dehydrogenase Inhibitors with Clinical Candidate Potential. J.Med.Chem., 54, 2011
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