1ZWU
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![BU of 1zwu by Molmil](/molmil-images/mine/1zwu) | 30 NMR structures of AcAMP2-like peptide with non natural beta-(2-naphthyl)-alanine residue. | Descriptor: | AMARANTHUS CAUDATUS ANTIMICROBIAL PEPTIDE 2 (ACMP2) | Authors: | Chavez, M.I, Andreu, C, Vidal, P, Freire, F, Aboitiz, N, Groves, P, Asensio, J.L, Asensio, G, Muraki, M, Canada, F.J, Jimenez-Barbero, J. | Deposit date: | 2005-06-06 | Release date: | 2005-12-06 | Last modified: | 2021-10-20 | Method: | SOLUTION NMR | Cite: | On the Importance of Carbohydrate-Aromatic Interactions for the Molecular Recognition of Oligosaccharides by Proteins: NMR Studies of the Structure and Binding Affinity of AcAMP2-like Peptides with Non-Natural Naphthyl and Fluoroaromatic Residues. Chemistry, 11, 2005
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3D5F
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![BU of 3d5f by Molmil](/molmil-images/mine/3d5f) | Crystal Structure of PPAR-delta complex | Descriptor: | Peroxisome proliferator-activated receptor delta, {4-[3-(4-acetyl-3-hydroxy-2-propylphenoxy)propoxy]phenoxy}acetic acid | Authors: | Amano, Y. | Deposit date: | 2008-05-16 | Release date: | 2008-06-03 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | PPAR-Delta Activation Contributes to Neuroprotectio Against Thapsigargin-Induced SH-SY5Y Cell Death to be published
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3VND
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![BU of 3vnd by Molmil](/molmil-images/mine/3vnd) | Crystal structure of tryptophan synthase alpha-subunit from the psychrophile Shewanella frigidimarina K14-2 | Descriptor: | 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, SULFATE ION, Tryptophan synthase alpha chain | Authors: | Mitsuya, D, Tanaka, S, Matsumura, H, Takano, K, Urano, N, Ishida, M. | Deposit date: | 2012-01-12 | Release date: | 2013-01-16 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Strategy for cold adaptation of the tryptophan synthase alpha subunit from the psychrophile Shewanella frigidimarina K14-2: crystal structure and physicochemical properties J.Biochem., 155, 2014
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2Z6C
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![BU of 2z6c by Molmil](/molmil-images/mine/2z6c) | |
2Z6D
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![BU of 2z6d by Molmil](/molmil-images/mine/2z6d) | |
2Z8Z
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![BU of 2z8z by Molmil](/molmil-images/mine/2z8z) | Crystal structure of a platinum-bound S445C mutant of Pseudomonas sp. MIS38 lipase | Descriptor: | CALCIUM ION, Lipase, PLATINUM (II) ION, ... | Authors: | Angkawidjaja, C, You, D.J, Matsumura, H, Koga, Y, Takano, K, Kanaya, S. | Deposit date: | 2007-09-13 | Release date: | 2007-10-30 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Crystal structure of a family I.3 lipase from Pseudomonas sp. MIS38 in a closed conformation FEBS Lett., 581, 2007
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3W5E
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![BU of 3w5e by Molmil](/molmil-images/mine/3w5e) | Crystal structure of phosphodiesterase 4B in complex with compound 31e | Descriptor: | CALCIUM ION, N-tert-butyl-2-{4-[(5,5-dioxido-2-phenyl-7,8-dihydro-6H-thiopyrano[3,2-d]pyrimidin-4-yl)amino]phenyl}acetamide, ZINC ION, ... | Authors: | Takahashi, M, Hanzawa, H. | Deposit date: | 2013-01-28 | Release date: | 2013-05-29 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Identification of the fused bicyclic 4-amino-2-phenylpyrimidine derivatives as novel and potent PDE4 inhibitors Bioorg.Med.Chem.Lett., 23, 2013
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3AA9
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![BU of 3aa9 by Molmil](/molmil-images/mine/3aa9) | Crystal Structure Analysis of the Mutant CutA1 (E61V) from E. coli | Descriptor: | Divalent-cation tolerance protein cutA | Authors: | Matsuura, Y, Tanaka, T, Bagautdinov, B, Kunishima, N, Yutani, K. | Deposit date: | 2009-11-12 | Release date: | 2010-08-11 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Remarkable improvement in the heat stability of CutA1 from Escherichia coli by rational protein design J.Biochem., 148, 2010
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3WIG
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![BU of 3wig by Molmil](/molmil-images/mine/3wig) | Human MEK1 kinase in complex with CH5126766 and MgAMP-PNP | Descriptor: | CHLORIDE ION, Dual specificity mitogen-activated protein kinase kinase 1, MAGNESIUM ION, ... | Authors: | Lukacs, C.M, Janson, C, Schuck, V. | Deposit date: | 2013-09-12 | Release date: | 2014-06-04 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Disruption of CRAF-Mediated MEK Activation Is Required for Effective MEK Inhibition in KRAS Mutant Tumors Cancer Cell, 25, 2014
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3WD9
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![BU of 3wd9 by Molmil](/molmil-images/mine/3wd9) | Crystal structure of phosphodiesterase 4B in complex with compound 10f | Descriptor: | 4-[(4-{2-[(2,2-dimethylpropyl)amino]-2-oxoethyl}phenyl)amino]-2-phenylpyrimidine-5-carboxamide, CALCIUM ION, ZINC ION, ... | Authors: | Takahashi, M, Hanzawa, H. | Deposit date: | 2013-06-11 | Release date: | 2013-10-23 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Synthesis and biological evaluation of 5-carbamoyl-2-phenylpyrimidine derivatives as novel and potent PDE4 inhibitors Bioorg.Med.Chem., 21, 2013
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3AA8
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![BU of 3aa8 by Molmil](/molmil-images/mine/3aa8) | Crystal Structure Analysis of the Mutant CutA1 (S11V/E61V) from E. coli | Descriptor: | Divalent-cation tolerance protein cutA | Authors: | Matsuura, Y, Tanaka, T, Bagautdinov, B, Kunishima, N, Yutani, K. | Deposit date: | 2009-11-12 | Release date: | 2010-08-11 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Remarkable improvement in the heat stability of CutA1 from Escherichia coli by rational protein design J.Biochem., 148, 2010
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2Z8X
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![BU of 2z8x by Molmil](/molmil-images/mine/2z8x) | Crystal structure of extracellular lipase from Pseudomonas sp. MIS38 | Descriptor: | CALCIUM ION, Lipase, ZINC ION | Authors: | Angkawidjaja, C, You, D.J, Matsumura, H, Koga, Y, Takano, K, Kanaya, S. | Deposit date: | 2007-09-11 | Release date: | 2007-10-30 | Last modified: | 2024-03-13 | Method: | X-RAY DIFFRACTION (1.48 Å) | Cite: | Crystal structure of a family I.3 lipase from Pseudomonas sp. MIS38 in a closed conformation FEBS Lett., 581, 2007
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2ZOM
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![BU of 2zom by Molmil](/molmil-images/mine/2zom) | Crystal structure of CutA1 from Oryza sativa | Descriptor: | GLYCEROL, Protein CutA, chloroplast, ... | Authors: | Kezuka, Y, Bagautdinov, B, Katoh, S, Ohtake, Y, Yutani, K, Nonaka, T, Katoh, E. | Deposit date: | 2008-05-23 | Release date: | 2009-05-26 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (3.02 Å) | Cite: | Crystal structure of CutA1 from Oryza sativa To be Published
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3AH6
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![BU of 3ah6 by Molmil](/molmil-images/mine/3ah6) | Remarkable improvement of the heat stability of CutA1 from E.coli by rational protein designing | Descriptor: | Divalent-cation tolerance protein cutA | Authors: | Matsuura, Y, Tanaka, T, Bagautdinov, B, Kunishima, N, Yutani, K. | Deposit date: | 2010-04-15 | Release date: | 2010-08-11 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Remarkable improvement in the heat stability of CutA1 from Escherichia coli by rational protein design J.Biochem., 148, 2010
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3BPP
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![BU of 3bpp by Molmil](/molmil-images/mine/3bpp) | |
3BK6
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![BU of 3bk6 by Molmil](/molmil-images/mine/3bk6) | |
3VI0
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![BU of 3vi0 by Molmil](/molmil-images/mine/3vi0) | |
3VW9
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![BU of 3vw9 by Molmil](/molmil-images/mine/3vw9) | Human Glyoxalase I with an N-hydroxypyridone inhibitor | Descriptor: | 1-hydroxy-6-[1-(3-methoxypropyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]-4-phenylpyridin-2(1H)-one, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Lactoylglutathione lyase, ... | Authors: | Fukami, T.A, Irie, M, Matsuura, T. | Deposit date: | 2012-08-10 | Release date: | 2012-12-12 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.47 Å) | Cite: | Design and evaluation of azaindole-substituted N-hydroxypyridones as glyoxalase I inhibitors Bioorg.Med.Chem.Lett., 22, 2012
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3VVK
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3W0T
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![BU of 3w0t by Molmil](/molmil-images/mine/3w0t) | Human Glyoxalase I with an N-hydroxypyridone derivative inhibitor | Descriptor: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Lactoylglutathione lyase, N-[3-(1-hydroxy-6-oxo-4-phenyl-1,6-dihydropyridin-2-yl)phenyl]methanesulfonamide, ... | Authors: | Fukami, T.A, Irie, M, Matsuura, T. | Deposit date: | 2012-11-02 | Release date: | 2013-11-06 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.351 Å) | Cite: | N-Hydroxypyridone-based glyoxalase I inhibitors mimicking binding interactions of the substrate To be Published
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3VHZ
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3W0U
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![BU of 3w0u by Molmil](/molmil-images/mine/3w0u) | human Glyoxalase I with an N-hydroxypyridone inhibitor | Descriptor: | Lactoylglutathione lyase, N-[3-(1-Hydroxy-6-oxo-4-phenyl-1,6-dihydro-pyridin-2-yl)-5-methanesulfonylamino-phenyl]-methanesulfonamide, ZINC ION | Authors: | Fukami, T.A, Irie, M, Matsuura, T. | Deposit date: | 2012-11-02 | Release date: | 2013-11-06 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | N-Hydroxypyridone-based glyoxalase I inhibitors mimicking binding interactions of the substrate to be published
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2ZOI
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![BU of 2zoi by Molmil](/molmil-images/mine/2zoi) | |
3A1R
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![BU of 3a1r by Molmil](/molmil-images/mine/3a1r) | |
3A22
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![BU of 3a22 by Molmil](/molmil-images/mine/3a22) | Crystal Structure of beta-L-Arabinopyranosidase complexed with L-arabinose | Descriptor: | 2-(2-{2-[2-(2-METHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHANOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, ... | Authors: | Fujimoto, Z, Ichinose, H, Kaneko, S. | Deposit date: | 2009-04-27 | Release date: | 2009-07-14 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | A beta-l-Arabinopyranosidase from Streptomyces avermitilis is a novel member of glycoside hydrolase family 27. J.Biol.Chem., 284, 2009
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