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CRYSTAL STRUCTURE OF CRUZAIN BOUND TO WRR-99
Descriptor:	CRUZAIN, N-[3-CARBOXY-2-HYDROXY-PROPIONYL]-D-HOMOPHENYLALANYL-AMINO-2-METHYLBUTANE
Authors:	Brinen, L.S, Gillmor, S.A, Fletterick, R.J.
Deposit date:	2000-04-26
Release date:	2003-06-10
Last modified:	2011-07-13
Method:	X-RAY DIFFRACTION (2 Å)
Cite:	Crystal Structure of Cruzain bound to WRR-99 To be Published

CRYSTAL STRUCTURE ANALYSIS OF CRUZAIN BOUND TO A VINYL SULFONE DERIVED INHIBITOR (I)
Descriptor:	3-[[N-[MORPHOLIN-N-YL]-CARBONYL]-PHENYLALANINYL-AMINO]-5- PHENYL-PENTANE-1-SULFONYLBENZENE, CRUZAIN
Authors:	Brinen, L.S, Hansell, E, Roush, W.R, McKerrow, J.H, Fletterick, R.J.
Deposit date:	2000-05-23
Release date:	2000-07-26
Last modified:	2011-07-13
Method:	X-RAY DIFFRACTION (2.15 Å)
Cite:	A target within the target: probing cruzain's P1' site to define structural determinants for the Chagas' disease protease. Structure Fold.Des., 8, 2000

High Resolution Crystal Structure Analysis Of Cruzain non-covalently Bound To A Hydroxymethyl Ketone Inhibitor (II)
Descriptor:	Cruzipain, [1-(3-HYDROXY-2-OXO-1-PHENETHYL-PROPYLCARBAMOYL)2-PHENYL-ETHYL]-CARBAMIC ACID PYRIDIN-4-YLMETHYL ESTER
Authors:	Brinen, L.S, Huang, L, Ellman, J.A.
Deposit date:	2002-08-07
Release date:	2002-12-18
Last modified:	2017-10-11
Method:	X-RAY DIFFRACTION (1.2 Å)
Cite:	Crystal Structures of Reversible Ketone-based Inhibitors of the Cysteine Protease Cruzain Bioorg.Med.Chem., 11, 2003

High Resolution Crystal Structure Analysis Of Cruzain non-covalently Bound To A Hydroxymethyl Ketone Inhibitor (I)
Descriptor:	CRUZIPAIN, [1-(1-BENZYL-3-HYDROXY-2-OXO-PROPYLCARBAMOYL)-2-PHENYL-ETHYL]-CARBAMIC ACID BENZYL ESTER
Authors:	Brinen, L.S, Huang, L, Ellman, J.A.
Deposit date:	2002-08-07
Release date:	2002-12-18
Last modified:	2017-10-11
Method:	X-RAY DIFFRACTION (1.2 Å)
Cite:	Crystal Structures of Reversible Ketone-based Inhibitors of the Cysteine Protease Cruzain Bioorg.Med.Chem., 11, 2003