Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
8BW3
DownloadVisualize
BU of 8bw3 by Molmil
PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative
Descriptor: (2S)-N-(cyclopropylmethyl)-2-methyl-4-(1-methyl-1H-pyrrole-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Hassell-Hart, S, Bradshaw, W.J, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
Deposit date:2022-12-06
Release date:2022-12-21
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.3 Å)
Cite:PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative
To Be Published
8BW4
DownloadVisualize
BU of 8bw4 by Molmil
PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative
Descriptor: (2R)-4-(3-fluoranylthiophen-2-yl)carbonyl-N-(4-methoxyphenyl)-2-methyl-piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Hassell-Hart, S, Bradshaw, W.J, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
Deposit date:2022-12-06
Release date:2022-12-21
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative
To Be Published
8BW2
DownloadVisualize
BU of 8bw2 by Molmil
PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative
Descriptor: (2R)-N-(2-methoxyethyl)-2-methyl-4-thiophen-2-ylcarbonyl-piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Hassell-Hart, S, Bradshaw, W.J, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
Deposit date:2022-12-06
Release date:2022-12-21
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.35 Å)
Cite:PanDDA analysis -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative
To Be Published
7FUU
DownloadVisualize
BU of 7fuu by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z445977856
Descriptor: N-{[(2S)-oxolan-2-yl]methyl}-4-(thiophene-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.16 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVR
DownloadVisualize
BU of 7fvr by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z166737374
Descriptor: 4-(thiophene-2-carbonyl)-N-[(thiophen-2-yl)methyl]piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.19 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVM
DownloadVisualize
BU of 7fvm by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z1590917771
Descriptor: 4-(furan-2-carbonyl)-N-(1,2-oxazol-3-yl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.26 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FUV
DownloadVisualize
BU of 7fuv by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z183376720
Descriptor: N-cyclopropyl-4-(furan-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.19 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FUT
DownloadVisualize
BU of 7fut by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z44602357
Descriptor: 4-(furan-2-carbonyl)-N-propylpiperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.18 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FV0
DownloadVisualize
BU of 7fv0 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z44602337
Descriptor: 4-(furan-2-carbonyl)-N-phenylpiperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.21 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVC
DownloadVisualize
BU of 7fvc by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z495704106
Descriptor: N-(cyclopropylmethyl)-4-(3,4-dichlorobenzoyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.18 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FUW
DownloadVisualize
BU of 7fuw by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z961579360
Descriptor: (3S)-2-benzyl-N'-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline-3-carbohydrazide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.19 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVI
DownloadVisualize
BU of 7fvi by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z183306756
Descriptor: N-[(2H-1,3-benzodioxol-5-yl)methyl]-4-(furan-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.18 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FV1
DownloadVisualize
BU of 7fv1 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4912742920
Descriptor: PH-interacting protein, tert-butyl [3-({[4-(furan-2-carbonyl)piperazine-1-carbonyl]amino}methyl)phenyl]carbamate
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.19 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVL
DownloadVisualize
BU of 7fvl by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4140355932
Descriptor: N-{[(2S)-5,5-dimethyl-1,4-dioxan-2-yl]methyl}-4-(3-hydroxybenzoyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FV9
DownloadVisualize
BU of 7fv9 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z1004253138
Descriptor: 4-(5-methylfuran-2-carbonyl)-N-[(thiophen-2-yl)methyl]piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.17 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVQ
DownloadVisualize
BU of 7fvq by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z68576046
Descriptor: N-butyl-4-(thiophene-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVB
DownloadVisualize
BU of 7fvb by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z6617539657
Descriptor: N-(2-aminoethyl)-4-(furan-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.38 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVJ
DownloadVisualize
BU of 7fvj by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4913873236
Descriptor: (2S)-4-(furan-2-carbonyl)-2-methyl-N-(2,2,2-trifluoroethyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.19 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVP
DownloadVisualize
BU of 7fvp by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z1004277578
Descriptor: N-butyl-4-(5-methylfuran-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FV2
DownloadVisualize
BU of 7fv2 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z445899798
Descriptor: N-(2-methoxyethyl)-4-(thiophene-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FV6
DownloadVisualize
BU of 7fv6 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z1334218055
Descriptor: N-methyl-4-[5-(phenoxymethyl)furan-2-carbonyl]piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.19 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FV8
DownloadVisualize
BU of 7fv8 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z964297186
Descriptor: 4-(3-chlorobenzoyl)-N-[3-(6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)-3-oxopropyl]-1,4-diazepane-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FV3
DownloadVisualize
BU of 7fv3 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4912742924
Descriptor: (2R)-N-butyl-4-(furan-2-carbonyl)-2-methylpiperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FVA
DownloadVisualize
BU of 7fva by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4913872963
Descriptor: (2S)-N-(cyclopropylmethyl)-4-(furan-2-carbonyl)-2-methylpiperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.19 Å)
Cite:PanDDA analysis group deposition
To Be Published
7FV4
DownloadVisualize
BU of 7fv4 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z44602341
Descriptor: N-(2-fluorophenyl)-4-(furan-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
Deposit date:2023-03-09
Release date:2023-03-29
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published

221051

건을2024-06-12부터공개중

PDB statisticsPDBj update infoContact PDBjnumon