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3QN7
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BU of 3qn7 by Molmil
Potent and selective bicyclic peptide inhibitor (UK18) of human urokinase-type plasminogen activator(uPA)
分子名称: 1,3,5-tris(bromomethyl)benzene, Bicyclic peptide inhibitor, Urokinase-type plasminogen activator
著者Angelini, A, Cendron, L, Touati, J, Winter, G, Zanotti, G, Heinis, C.
登録日2011-02-08
公開日2012-02-15
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Bicyclic peptide inhibitor reveals large contact interface with a protease target
Acs Chem.Biol., 7, 2012
4GLY
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BU of 4gly by Molmil
Human urokinase-type plasminogen activator uPA in complex with the two-disulfide bridge peptide UK504
分子名称: BICYCLIC PEPTIDE INHIBITOR UK504, CHLORIDE ION, GLYCEROL, ...
著者Buth, S.A, Leiman, P.G, Chen, S, Heinis, C.
登録日2012-08-15
公開日2013-05-15
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.518 Å)
主引用文献Bicyclic Peptide Ligands Pulled out of Cysteine-Rich Peptide Libraries.
J.Am.Chem.Soc., 135, 2013

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件を2024-09-11に公開中

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