3A99
| Structure of PIM-1 kinase crystallized in the presence of P27KIP1 Carboxy-terminal peptide | 分子名称: | MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, Proto-oncogene serine/threonine-protein kinase pim-1 | 著者 | Morishita, D, Takami, M, Yoshikawa, S, Katayama, R, Sato, S, Kukimoto-Niino, M, Umehara, T, Shirouzu, M, Sekimizu, K, Yokoyama, S, Fujita, N. | 登録日 | 2009-10-22 | 公開日 | 2010-11-03 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Cell-permeable carboxyl-terminal p27(Kip1) peptide exhibits anti-tumor activity by inhibiting Pim-1 kinase J.Biol.Chem., 286, 2011
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2ZA0
| Crystal structure of mouse glyoxalase I complexed with methyl-gerfelin | 分子名称: | Glyoxalase I, ZINC ION, methyl 4-(2,3-dihydroxy-5-methylphenoxy)-2-hydroxy-6-methylbenzoate | 著者 | Okumura, H, Kawatani, M, Osada, H. | 登録日 | 2007-09-26 | 公開日 | 2008-08-12 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The identification of an osteoclastogenesis inhibitor through the inhibition of glyoxalase I Proc.Natl.Acad.Sci.Usa, 105, 2008
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7NZY
| Crystal structure of human Casein Kinase I delta in complex with CGS-15943 | 分子名称: | 9-chloranyl-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine, Casein kinase I isoform delta, MALONATE ION, ... | 著者 | Pichlo, C, Baumann, U. | 登録日 | 2021-03-24 | 公開日 | 2022-10-05 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Phenotypic Discovery of Triazolo[1,5- c ]quinazolines as a First-In-Class Bone Morphogenetic Protein Amplifier Chemotype. J.Med.Chem., 65, 2022
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2ZIB
| Crystal structure analysis of calcium-independent type II antifreeze protein | 分子名称: | SULFATE ION, Type II antifreeze protein | 著者 | Nishimiya, Y, Sato, R, Kondo, H, Noro, N, Sugimoto, H, Suzuki, M, Tsuda, S. | 登録日 | 2008-02-14 | 公開日 | 2008-08-19 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.34 Å) | 主引用文献 | Crystal structure and mutational analysis of Ca2+-independent type II antifreeze protein from longsnout poacher, Brachyopsis rostratus J.Mol.Biol., 382, 2008
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