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3A99
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BU of 3a99 by Molmil
Structure of PIM-1 kinase crystallized in the presence of P27KIP1 Carboxy-terminal peptide
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, Proto-oncogene serine/threonine-protein kinase pim-1
著者Morishita, D, Takami, M, Yoshikawa, S, Katayama, R, Sato, S, Kukimoto-Niino, M, Umehara, T, Shirouzu, M, Sekimizu, K, Yokoyama, S, Fujita, N.
登録日2009-10-22
公開日2010-11-03
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Cell-permeable carboxyl-terminal p27(Kip1) peptide exhibits anti-tumor activity by inhibiting Pim-1 kinase
J.Biol.Chem., 286, 2011
2ZA0
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BU of 2za0 by Molmil
Crystal structure of mouse glyoxalase I complexed with methyl-gerfelin
分子名称: Glyoxalase I, ZINC ION, methyl 4-(2,3-dihydroxy-5-methylphenoxy)-2-hydroxy-6-methylbenzoate
著者Okumura, H, Kawatani, M, Osada, H.
登録日2007-09-26
公開日2008-08-12
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The identification of an osteoclastogenesis inhibitor through the inhibition of glyoxalase I
Proc.Natl.Acad.Sci.Usa, 105, 2008
7NZY
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BU of 7nzy by Molmil
Crystal structure of human Casein Kinase I delta in complex with CGS-15943
分子名称: 9-chloranyl-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine, Casein kinase I isoform delta, MALONATE ION, ...
著者Pichlo, C, Baumann, U.
登録日2021-03-24
公開日2022-10-05
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Phenotypic Discovery of Triazolo[1,5- c ]quinazolines as a First-In-Class Bone Morphogenetic Protein Amplifier Chemotype.
J.Med.Chem., 65, 2022
2ZIB
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BU of 2zib by Molmil
Crystal structure analysis of calcium-independent type II antifreeze protein
分子名称: SULFATE ION, Type II antifreeze protein
著者Nishimiya, Y, Sato, R, Kondo, H, Noro, N, Sugimoto, H, Suzuki, M, Tsuda, S.
登録日2008-02-14
公開日2008-08-19
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.34 Å)
主引用文献Crystal structure and mutational analysis of Ca2+-independent type II antifreeze protein from longsnout poacher, Brachyopsis rostratus
J.Mol.Biol., 382, 2008

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件を2024-10-09に公開中

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