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5CL2
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BU of 5cl2 by Molmil
Crystal structure of Spo0M, sporulation control protein, from Bacillus subtilis.
分子名称: SODIUM ION, Sporulation-control protein spo0M
著者Sonoda, Y, Mizutani, K, Mikami, B.
登録日2015-07-16
公開日2015-12-16
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure of Spo0M, a sporulation-control protein from Bacillus subtilis.
Acta Crystallogr.,Sect.F, 71, 2015
4PM0
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BU of 4pm0 by Molmil
PDE7A catalytic domain in complex with 2-(Cyclopentylamino)thieno[3,2-d]pyrimidin-4(3H)-one derivative
分子名称: 2-(cyclopentylamino)-3-ethyl-7-ethynylthieno[3,2-d]pyrimidin-4(3H)-one, High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A, MAGNESIUM ION, ...
著者Kawai, K, Endo, Y, Asano, T, Amano, S, Sawada, K, Ueo, N, Takahashi, N, Sonoda, Y, Kamei, N, Nagata, N.
登録日2014-05-20
公開日2014-12-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Discovery of 2-(Cyclopentylamino)thieno[3,2-d]pyrimidin-4(3H)-one Derivatives as a New Series of Potent Phosphodiesterase 7 Inhibitors.
J.Med.Chem., 57, 2014
4Y2B
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BU of 4y2b by Molmil
Co-crystal structure of 3-ethyl-2-(isopropylamino)-7-(pyridin-3-yl)thieno[3,2-d]pyrimidin-4(3H)-one bound to PDE7A
分子名称: 3-ethyl-2-(propan-2-ylamino)-7-(pyridin-3-yl)thieno[3,2-d]pyrimidin-4(3H)-one, High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A, MAGNESIUM ION, ...
著者Endo, Y, Kawai, K, Asano, T, Amano, S, Asanuma, Y, Sawada, K, Onodera, Y, Ueo, N, Takahashi, N, Sonoda, Y, Kamei, N, Irie, T.
登録日2015-02-09
公開日2015-04-08
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献2-(Isopropylamino)thieno[3,2-d]pyrimidin-4(3H)-one derivatives as selective phosphodiesterase 7 inhibitors with potent in vivo efficacy
Bioorg.Med.Chem.Lett., 25, 2015
4YB9
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BU of 4yb9 by Molmil
Crystal structure of the Bovine Fructose transporter GLUT5 in an open inward-facing conformation
分子名称: Solute carrier family 2, facilitated glucose transporter member 5
著者Verdon, G, Kang, H.J, Iwata, S, Drew, D.
登録日2015-02-18
公開日2015-10-14
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structure and mechanism of the mammalian fructose transporter GLUT5.
Nature, 526, 2015
4YBQ
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BU of 4ybq by Molmil
Rat GLUT5 with Fv in the outward-open form
分子名称: Solute carrier family 2, facilitated glucose transporter member 5, antibody Fv fragment heavy chain, ...
著者Nomura, N, Shimamura, T, Iwata, S.
登録日2015-02-19
公開日2015-10-07
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (3.27 Å)
主引用文献Structure and mechanism of the mammalian fructose transporter GLUT5
Nature, 526, 2015

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件を2024-07-10に公開中

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