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3WOK
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BU of 3wok by Molmil
Crystal structure of the DAP BII (Space)
分子名称: GLYCEROL, ZINC ION, dipeptidyl aminopeptidase BII
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
3WOJ
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BU of 3woj by Molmil
Crystal structure of the DAP BII
分子名称: GLYCEROL, ZINC ION, dipeptidyl aminopeptidase BII
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
4Y04
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BU of 4y04 by Molmil
Crystal structure of dipeptidyl peptidase 11 (DPP11) from Porphyromonas gingivalis (Space)
分子名称: GLYCEROL, POTASSIUM ION, Peptidase S46
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Inaka, K, Tanaka, H, Yamada, M, Ohta, K, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2015-02-05
公開日2015-07-15
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.66 Å)
主引用文献Structural and mutational analyses of dipeptidyl peptidase 11 from Porphyromonas gingivalis reveal the molecular basis for strict substrate specificity.
Sci Rep, 5, 2015
4XZY
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BU of 4xzy by Molmil
Crystal structure of dipeptidyl peptidase 11 (DPP11) from Porphyromonas gingivalis
分子名称: GLYCEROL, Peptidase S46
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2015-02-05
公開日2015-07-15
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural and mutational analyses of dipeptidyl peptidase 11 from Porphyromonas gingivalis reveal the molecular basis for strict substrate specificity.
Sci Rep, 5, 2015
4Y01
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BU of 4y01 by Molmil
Crystal structure of dipeptidyl peptidase 11 (DPP11) from Porphyromonas gingivalis
分子名称: GLYCEROL, Peptidase S46
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2015-02-05
公開日2015-07-15
最終更新日2020-02-05
実験手法X-RAY DIFFRACTION (2.46 Å)
主引用文献Structural and mutational analyses of dipeptidyl peptidase 11 from Porphyromonas gingivalis reveal the molecular basis for strict substrate specificity.
Sci Rep, 5, 2015
4Y02
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BU of 4y02 by Molmil
Crystal structure of dipeptidyl peptidase 11 (DPP11) from Porphyromonas gingivalis (Ground)
分子名称: GLYCEROL, POTASSIUM ION, Peptidase S46
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2015-02-05
公開日2015-07-15
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Structural and mutational analyses of dipeptidyl peptidase 11 from Porphyromonas gingivalis reveal the molecular basis for strict substrate specificity.
Sci Rep, 5, 2015
4Y06
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BU of 4y06 by Molmil
Crystal structure of the DAP BII (G675R) dipeptide complex
分子名称: Dipeptidyl aminopeptidase BII, GLUTAMIC ACID, GLYCEROL, ...
著者Sakamoto, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2015-02-05
公開日2015-07-15
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Structural and mutational analyses of dipeptidyl peptidase 11 from Porphyromonas gingivalis reveal the molecular basis for strict substrate specificity.
Sci Rep, 5, 2015
6JTB
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BU of 6jtb by Molmil
Crystal structure of dipeptidyl peptidase 11 (DPP11) with citrate from Porphyromonas gingivalis (Space)
分子名称: Asp/Glu-specific dipeptidyl-peptidase, CITRIC ACID, DI(HYDROXYETHYL)ETHER, ...
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Roppongi, S, Kushibiki, C, Nakamura, A, Ogasawara, W, Tanaka, N.
登録日2019-04-10
公開日2019-10-02
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Fragment-based discovery of the first nonpeptidyl inhibitor of an S46 family peptidase.
Sci Rep, 9, 2019
6JTC
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BU of 6jtc by Molmil
Crystal structure of dipeptidyl peptidase 11 (DPP11) with SH-5 from Porphyromonas gingivalis (Space)
分子名称: 2-(2-azanylethylamino)-5-nitro-benzoic acid, Asp/Glu-specific dipeptidyl-peptidase, GLYCEROL
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Roppongi, S, Kushibiki, C, Nakamura, A, Ogasawara, W, Tanaka, N.
登録日2019-04-10
公開日2019-10-02
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.39 Å)
主引用文献Fragment-based discovery of the first nonpeptidyl inhibitor of an S46 family peptidase.
Sci Rep, 9, 2019
1WOJ
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BU of 1woj by Molmil
Crystal structure of human phosphodiesterase
分子名称: 2',3'-cyclic-nucleotide 3'-phosphodiesterase, PHOSPHATE ION
著者Sakamoto, Y, Tanaka, N, Ichimiya, T, Kurihara, T, Nakamura, K.T.
登録日2004-08-19
公開日2005-03-15
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of the catalytic fragment of human brain 2',3'-cyclic-nucleotide 3'-phosphodiesterase
J.Mol.Biol., 346, 2005
3WOR
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BU of 3wor by Molmil
Crystal structure of the DAP BII octapeptide complex
分子名称: Angiotensin II, GLYCEROL, ZINC ION, ...
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
3WOP
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BU of 3wop by Molmil
Crystal structure of the DAP BII hexapeptide complex II
分子名称: Angiotensin IV, GLYCEROL, ZINC ION, ...
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
3WOQ
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BU of 3woq by Molmil
Crystal structure of the DAP BII hexapeptide complex III
分子名称: Angiotensin IV, GLYCEROL, ZINC ION, ...
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
3WON
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BU of 3won by Molmil
Crystal structure of the DAP BII dipeptide complex III
分子名称: GLYCEROL, TYROSINE, VALINE, ...
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
3WOL
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BU of 3wol by Molmil
Crystal structure of the DAP BII dipeptide complex I
分子名称: GLYCEROL, TYROSINE, VALINE, ...
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
3WOM
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BU of 3wom by Molmil
Crystal structure of the DAP BII dipeptide complex II
分子名称: GLYCEROL, TYROSINE, VALINE, ...
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
3WOI
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BU of 3woi by Molmil
Crystal structure of the DAP BII (S657A)
分子名称: GLYCEROL, ZINC ION, dipeptidyl aminopeptidase BII
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
3WOO
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BU of 3woo by Molmil
Crystal structure of the DAP BII hexapeptide complex I
分子名称: Angiotensin II, GLYCEROL, ZINC ION, ...
著者Sakamoto, Y, Suzuki, Y, Iizuka, I, Tateoka, C, Roppongi, S, Fujimoto, M, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2013-12-29
公開日2014-09-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献S46 peptidases are the first exopeptidases to be members of clan PA
SCI REP, 4, 2014
7DKD
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BU of 7dkd by Molmil
Stenotrophomonas maltophilia DPP7 in complex with Asn-Tyr
分子名称: ASPARAGINE, Dipeptidyl-peptidase, GLYCEROL, ...
著者Sakamoto, Y, Nakamura, A, Suzuki, Y, Honma, N, Roppongi, S, Kushibiki, C, Yonezawa, N, Takahashi, M, Shida, Y, Gouda, H, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2020-11-23
公開日2021-11-03
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Structural basis for an exceptionally strong preference for asparagine residue at the S2 subsite of Stenotrophomonas maltophilia dipeptidyl peptidase 7.
Sci Rep, 11, 2021
7DKC
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BU of 7dkc by Molmil
Stenotrophomonas maltophilia DPP7 in complex with Tyr-Tyr
分子名称: Dipeptidyl-peptidase, GLYCEROL, TYROSINE
著者Sakamoto, Y, Nakamura, A, Suzuki, Y, Honma, N, Roppongi, S, Kushibiki, C, Yonezawa, N, Takahashi, M, Shida, Y, Gouda, H, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2020-11-23
公開日2021-11-03
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Structural basis for an exceptionally strong preference for asparagine residue at the S2 subsite of Stenotrophomonas maltophilia dipeptidyl peptidase 7.
Sci Rep, 11, 2021
7DKE
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BU of 7dke by Molmil
Stenotrophomonas maltophilia DPP7 in complex with Phe-Tyr
分子名称: Dipeptidyl-peptidase, GLYCEROL, PHENYLALANINE, ...
著者Sakamoto, Y, Nakamura, A, Suzuki, Y, Honma, N, Roppongi, S, Kushibiki, C, Yonezawa, N, Takahashi, M, Shida, Y, Gouda, H, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2020-11-23
公開日2021-11-03
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献Structural basis for an exceptionally strong preference for asparagine residue at the S2 subsite of Stenotrophomonas maltophilia dipeptidyl peptidase 7.
Sci Rep, 11, 2021
7DKB
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BU of 7dkb by Molmil
Stenotrophomonas maltophilia DPP7 in complex with Val-Tyr
分子名称: Dipeptidyl-peptidase, TYROSINE, VALINE
著者Sakamoto, Y, Nakamura, A, Suzuki, Y, Honma, N, Roppongi, S, Kushibiki, C, Yonezawa, N, Takahashi, M, Shida, Y, Gouda, H, Nonaka, T, Ogasawara, W, Tanaka, N.
登録日2020-11-23
公開日2021-11-03
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Structural basis for an exceptionally strong preference for asparagine residue at the S2 subsite of Stenotrophomonas maltophilia dipeptidyl peptidase 7.
Sci Rep, 11, 2021
8JNW
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BU of 8jnw by Molmil
PfDXR - Mn2+ - NADPH - MAMK89 quaternary complex
分子名称: 1-deoxy-D-xylulose 5-phosphate reductoisomerase, apicoplastic, CALCIUM ION, ...
著者Takada, S, Sakamoto, Y, Tanaka, N.
登録日2023-06-08
公開日2024-05-22
実験手法X-RAY DIFFRACTION (1.44 Å)
主引用文献Reverse N -Substituted Hydroxamic Acid Derivatives of Fosmidomycin Target a Previously Unknown Subpocket of 1-Deoxy-d-xylulose 5-Phosphate Reductoisomerase (DXR).
Acs Infect Dis., 10, 2024
8JNV
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BU of 8jnv by Molmil
PfDXR - Mn2+ - MAMK89 ternary complex
分子名称: 1-deoxy-D-xylulose 5-phosphate reductoisomerase, apicoplastic, CALCIUM ION, ...
著者Takada, S, Sakamoto, Y, Tanaka, N.
登録日2023-06-06
公開日2024-05-22
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Reverse N -Substituted Hydroxamic Acid Derivatives of Fosmidomycin Target a Previously Unknown Subpocket of 1-Deoxy-d-xylulose 5-Phosphate Reductoisomerase (DXR).
Acs Infect Dis., 10, 2024
5YP2
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BU of 5yp2 by Molmil
Crystal structure of dipeptidyl peptidase IV (DPP IV) with DPP4 inhibitor from Pseudoxanthomonas mexicana WO24
分子名称: (2S,5R)-1-[2-[[1-(hydroxymethyl)cyclopentyl]amino]ethanoyl]pyrrolidine-2,5-dicarbonitrile, Dipeptidyl aminopeptidase 4, GLYCEROL
著者Roppongi, S, Suzuki, Y, Tateoka, C, Fuimoto, M, Morisawa, S, Iizuka, I, Nakamura, A, Honma, N, Shida, Y, Ogasawara, W, Tanaka, N, Sakamoto, Y, Nonaka, T.
登録日2017-11-01
公開日2018-02-21
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.13 Å)
主引用文献Crystal structures of a bacterial dipeptidyl peptidase IV reveal a novel substrate recognition mechanism distinct from that of mammalian orthologues.
Sci Rep, 8, 2018

 

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