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8F4Q
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BU of 8f4q by Molmil
rat branched chain ketoacid dehydrogenase kinase in complex with inhibtors
分子名称: 3-chloro-5-fluorothieno[3,2-b]thiophene-2-carboxylic acid, ADENOSINE-5'-DIPHOSPHATE, SULFATE ION, ...
著者Liu, S.
登録日2022-11-11
公開日2023-12-13
実験手法X-RAY DIFFRACTION (2.151 Å)
主引用文献Discovery of branched-chain ketoacid dehydrogenase kinase (BDK) inhibitors acting as stabilizers or destabilizers
To Be Published
8F5F
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BU of 8f5f by Molmil
human branched chain ketoacid dehydrogenase kinase in complex with inhibitors
分子名称: (2P)-2-[(4P)-4-{6-[(1-ethylcyclopropyl)methoxy]pyridin-3-yl}-1,3-thiazol-2-yl]benzoic acid, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Liu, S, Roth Flach, R, Bollinger, E, Filipski, K.
登録日2022-11-14
公開日2023-07-05
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (3.149 Å)
主引用文献Small molecule branched-chain ketoacid dehydrogenase kinase (BDK) inhibitors with opposing effects on BDK protein levels.
Nat Commun, 14, 2023
8F5J
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BU of 8f5j by Molmil
human branched chain ketoacid dehydrogenase kinase in complex with inhibitors
分子名称: 3-chloro-5-fluorothieno[3,2-b]thiophene-2-carboxylic acid, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Liu, S, Roth Flach, R, Bollinger, E, Filipski, K.
登録日2022-11-14
公開日2023-07-05
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.545 Å)
主引用文献Small molecule branched-chain ketoacid dehydrogenase kinase (BDK) inhibitors with opposing effects on BDK protein levels.
Nat Commun, 14, 2023
8F5S
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BU of 8f5s by Molmil
human branched chain ketoacid dehydrogenase kinase in complex with inhibitors
分子名称: (2M)-2-[2-(4-methylphenyl)-1,3-thiazol-4-yl]benzoic acid, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Liu, S, Roth Flach, R, Bollinger, E, Filipski, K.
登録日2022-11-15
公開日2023-07-05
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.793 Å)
主引用文献Small molecule branched-chain ketoacid dehydrogenase kinase (BDK) inhibitors with opposing effects on BDK protein levels.
Nat Commun, 14, 2023

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件を2024-07-24に公開中

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