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3AUL
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BU of 3aul by Molmil
Crystal structure of wild-type Lys48-linked diubiquitin in an open conformation
分子名称: Polyubiquitin-C
著者Hirano, T, Olivier, S, Yagi, M, Takemoto, E, Hiromoto, T, Satoh, T, Mizushima, T, Kato, K.
登録日2011-02-09
公開日2011-09-07
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.39 Å)
主引用文献Conformational dynamics of wild-type Lys48-linked diubiquitin in solution
J.Biol.Chem., 286, 2011
6TCU
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BU of 6tcu by Molmil
Glycogen synthase kinase-3 beta (GSK3b) in complex with ligand 1
分子名称: 5-[2,3-bis(fluoranyl)phenyl]-~{N}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{H}-indazole-3-carboxamide, ACETATE ION, Glycogen synthase kinase-3 beta
著者Lammens, A, Krapp, S, Buonfiglio, R, Ombrato, R.
登録日2019-11-06
公開日2020-09-16
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Optimization of Indazole-Based GSK-3 Inhibitors with Mitigated hERG Issue andIn VivoActivity in a Mood Disorder Model.
Acs Med.Chem.Lett., 11, 2020

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件を2024-07-24に公開中

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