Search by PDB author

Human FGF in complex with a covalent inhibitor
分子名称:	Fibroblast growth factor receptor 1, GLYCEROL, SULFATE ION, ...
著者	Debreczeni, J, Breed, J, Mukherjee, H, Aquila, B, Kaiser, C, Tentarelli, S, Whitty, A, Grimster, N.
登録日	2017-05-26
公開日	2018-02-07
実験手法	X-RAY DIFFRACTION (2.01 Å)
主引用文献	A study of the reactivity of S(VI)-F containing warheads with nucleophilic amino-acid side chains under physiological conditions. Org. Biomol. Chem., 15, 2017

Human FGF in complex with a covalent inhibitor
分子名称:	Fibroblast growth factor receptor 1, SULFATE ION, [(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoate
著者	Debreczeni, J, Breed, J, Mukherjee, H, Aquila, B, Kaiser, C, Tentarelli, S, Whitty, A, Grimster, N.
登録日	2017-05-26
公開日	2018-02-07
実験手法	X-RAY DIFFRACTION (1.91 Å)
主引用文献	A study of the reactivity of S(VI)-F containing warheads with nucleophilic amino-acid side chains under physiological conditions. Org. Biomol. Chem., 15, 2017

BCL-XL in a complex with a covalent small molecule inhibitor
分子名称:	4-(4-fluorophenyl)-3-fluorosulfonyl-benzoic acid, BROMIDE ION, Bcl-2-like protein 1
著者	Hargreaves, D.
登録日	2019-05-09
公開日	2019-10-02
最終更新日	2019-11-20
実験手法	X-RAY DIFFRACTION (2.4 Å)
主引用文献	Discovery and optimization of covalent Bcl-xL antagonists. Bioorg.Med.Chem.Lett., 29, 2019