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2N4V
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BU of 2n4v by Molmil
NMR structure of Fbp28 WW domain T456D mutant
分子名称: Transcription elongation regulator 1
著者Medina, J, Macias, M, Martin-Malpartida, P, Scheraga, H.A.
登録日2015-07-01
公開日2015-10-21
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Preventing fibril formation of a protein by selective mutation.
Proc.Natl.Acad.Sci.USA, 112, 2015
2N4S
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BU of 2n4s by Molmil
NMR structure of Fbp28 WW domain L453E mutant
分子名称: Transcription elongation regulator 1
著者Medina, J, Macias, M, Martin-Malpartida, P, Scheraga, H.A.
登録日2015-07-01
公開日2015-10-21
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Preventing fibril formation of a protein by selective mutation.
Proc.Natl.Acad.Sci.USA, 112, 2015
2N4W
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BU of 2n4w by Molmil
NMR structure of Fbp28 WW domain T456Y mutant
分子名称: Transcription elongation regulator 1
著者Medina, J, Macias, M, Martin-Malpartida, P, Scheraga, H.A.
登録日2015-07-01
公開日2015-10-21
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Preventing fibril formation of a protein by selective mutation.
Proc.Natl.Acad.Sci.USA, 112, 2015
2N4T
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BU of 2n4t by Molmil
NMR structure of Fbp28 WW domain L453W mutant
分子名称: Transcription elongation regulator 1
著者Medina, J, Macias, M, Martin-Malpartida, P, Scheraga, H.A.
登録日2015-07-01
公開日2015-10-21
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Preventing fibril formation of a protein by selective mutation.
Proc.Natl.Acad.Sci.USA, 112, 2015
2N4U
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BU of 2n4u by Molmil
NMR structure of Fbp28 WW domain E454Y mutant
分子名称: Transcription elongation regulator 1
著者Medina, J, Macias, M, Martin-Malpartida, P, Scheraga, H.A.
登録日2015-07-01
公開日2015-10-21
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Preventing fibril formation of a protein by selective mutation.
Proc.Natl.Acad.Sci.USA, 112, 2015
2N4R
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BU of 2n4r by Molmil
NMR structure of Fbp28 WW domain L453D mutant
分子名称: Transcription elongation regulator 1
著者Medina, J, Macias, M, Martin-Malpartida, P, Scheraga, H.A.
登録日2015-07-01
公開日2015-10-21
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Preventing fibril formation of a protein by selective mutation.
Proc.Natl.Acad.Sci.USA, 112, 2015
7SZQ
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BU of 7szq by Molmil
Human P300 complexed with an azaindazole inhibitor
分子名称: 1-[1-(4-chlorophenyl)cyclopentane-1-carbonyl]-N-1H-pyrazolo[4,3-b]pyridin-5-yl-D-prolinamide, Histone acetyltransferase p300
著者Shewchuk, L.M, Reid, R.A.
登録日2021-11-29
公開日2022-11-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
J.Med.Chem., 65, 2022
7SSK
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BU of 7ssk by Molmil
Human P300 complexed with a glycine-based inhibitor
分子名称: 1,2-ETHANEDIOL, ACETATE ION, Histone acetyltransferase p300, ...
著者Shewchuk, L.M, Reid, R.A.
登録日2021-11-11
公開日2022-11-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.36 Å)
主引用文献Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
J.Med.Chem., 65, 2022
7SS8
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BU of 7ss8 by Molmil
Human P300 complexed with a proline-based inhibitor
分子名称: 1,2-ETHANEDIOL, 1-[1-(4-chlorophenyl)cyclopentane-1-carbonyl]-N-{[3-(methylcarbamoyl)phenyl]methyl}-D-prolinamide, Histone acetyltransferase p300, ...
著者Shewchuk, L.M, Reid, R.A.
登録日2021-11-10
公開日2022-11-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
J.Med.Chem., 65, 2022

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件を2024-07-24に公開中

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