Search by PDB author

Crystal structure of TrmD from Pseudomonas aeruginosa in complex with active-site inhibitor
分子名称:	N-{(3S)-1-[3-(pyridin-4-yl)-1H-pyrazol-5-yl]piperidin-3-yl}-1H-indole-2-carboxamide, S-ADENOSYLMETHIONINE, tRNA (guanine-N(1)-)-methyltransferase
著者	Zhong, W, Koay, A, Wong, Y.W, Sahili, A.E, Nah, Q, Kang, C, Poulsen, A, Chionh, Y.K, McBee, M, Matter, A, Hill, J, Lescar, J, Dedon, P.C.
登録日	2018-08-08
公開日	2019-08-14
最終更新日	2023-11-22
実験手法	X-RAY DIFFRACTION (2.75 Å)
主引用文献	Targeting the Bacterial Epitranscriptome for Antibiotic Development: Discovery of Novel tRNA-(N1G37) Methyltransferase (TrmD) Inhibitors. Acs Infect Dis., 5, 2019

Crystal structure of SmyD3 in complex with covalent inhibitor 4
分子名称:	Histone-lysine N-methyltransferase SMYD3, S-ADENOSYLMETHIONINE, ZINC ION, ...
著者	Baburajendran, N, Anna E, J.
登録日	2017-10-11
公開日	2018-10-17
最終更新日	2019-07-10
実験手法	X-RAY DIFFRACTION (2.135 Å)
主引用文献	Discovery of Irreversible Inhibitors Targeting Histone Methyltransferase, SMYD3. Acs Med.Chem.Lett., 10, 2019

Crystal structure of SmyD3 in complex with covalent inhibitor 5
分子名称:	Histone-lysine N-methyltransferase SMYD3, S-ADENOSYLMETHIONINE, ZINC ION, ...
著者	Baburajendran, N, Joy, J.
登録日	2018-10-10
公開日	2019-08-14
最終更新日	2024-03-27
実験手法	X-RAY DIFFRACTION (2.351 Å)
主引用文献	Discovery of Irreversible Inhibitors Targeting Histone Methyltransferase, SMYD3. Acs Med.Chem.Lett., 10, 2019