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7QYF
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Structure of the transaminase PluriZyme variant (TR2E2)
分子名称: Aminotransferase TR2
著者Roda, S, Fernandez-Lopez, L, Benedens, M, Bollinger, A, Thies, S, Schumacher, J, Coscolin, C, Kazemi, M, Santiago, G, Gertzen, C.G, Gonzalez-Alfonso, J, Plou, F.J, Jaeger, K.E, Smits, S.H, Ferrer, M, Guallar, V.
登録日2022-01-28
公開日2023-07-26
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献A Plurizyme with Transaminase and Hydrolase Activity Catalyzes Cascade Reactions.
Angew Chem Int Ed Engl, 61, 2022
7QX3
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Structure of the transaminase TR2E2 with EOS
分子名称: 2-azanylethyl hydrogen sulfate, Aminotransferase TR2
著者Roda, S, Fernandez-Lopez, L, Benedens, M, Bollinger, A, Thies, S, Schumacher, J, Coscolin, C, Kazemi, M, Santiago, G, Gertzen, C.G, Gonzalez-Alfonso, J, Plou, F.J, Jaeger, K.E, Smits, S.H, Ferrer, M, Guallar, V.
登録日2022-01-26
公開日2023-08-16
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献A Plurizyme with Transaminase and Hydrolase Activity Catalyzes Cascade Reactions.
Angew.Chem.Int.Ed.Engl., 61, 2022
7QX0
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Transaminase Structure of Plurienzyme (Tr2E2) in complex with PLP
分子名称: Aminotransferase TR2, PYRIDOXAL-5'-PHOSPHATE
著者Roda, S, Fernandez-Lopez, L, Benedens, M, Bollinger, A, Thies, S, Schumacher, J, Coscolin, C, Kazemi, M, Santiago, G, Gertzen, C.G, Gonzalez-Alfonso, J, Plou, F.J, Jaeger, K.E, Smits, S.H, Ferrer, M, Guallar, V.
登録日2022-01-26
公開日2023-08-16
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献A Plurizyme with Transaminase and Hydrolase Activity Catalyzes Cascade Reactions.
Angew Chem Int Ed Engl, 61, 2022
7QYG
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Structure of the transaminase TR2
分子名称: Aminotransferase TR2
著者Roda, S, Fernandez-Lopez, L, Benedens, M, Bollinger, A, Thies, S, Schumacher, J, Coscolin, C, Kazemi, M, Santiago, G, Gertzen, C.G, Gonzalez-Alfonso, J, Plou, F.J, Jaeger, K.E, Smits, S.H, Ferrer, M, Guallar, V.
登録日2022-01-28
公開日2023-08-16
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献A Plurizyme with Transaminase and Hydrolase Activity Catalyzes Cascade Reactions.
Angew Chem Int Ed Engl, 61, 2022
3I2V
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BU of 3i2v by Molmil
Crystal structure of human MOCS3 rhodanese-like domain
分子名称: Adenylyltransferase and sulfurtransferase MOCS3
著者Bacik, J.P, Walker, J.R, Lopez, L, Li, Y, Weigelt, J, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC)
登録日2009-06-29
公開日2009-07-21
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Crystal structure of the human MOCS3 rhodanese-like domain
To be Published
8CIQ
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BU of 8ciq by Molmil
JzTx-34 toxin peptide
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-10
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJP
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BU of 8cjp by Molmil
JzTx-34 toxin peptide H18A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJS
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JzTx-34 toxin peptide W31A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJQ
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JzTx-34 toxin peptide E20A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJR
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BU of 8cjr by Molmil
JzTx-34 toxin peptide W25A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
8CJT
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BU of 8cjt by Molmil
JzTx-34 toxin peptide W33A mutant
分子名称: Mu-theraphotoxin-Cg1a
著者Landon, C, Meudal, H.
登録日2023-02-13
公開日2023-07-26
実験手法SOLUTION NMR
主引用文献Structure-function relationship of new peptides activating human Na v 1.1.
Biomed Pharmacother, 165, 2023
7M7V
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BU of 7m7v by Molmil
Crystal Structure of Mtb Pks13 Thioesterase domain in complex with Compound 6
分子名称: 5-hydroxy-2-(4-hydroxyphenyl)-N-methyl-4-[(2-oxa-6-azaspiro[3.4]octan-6-yl)methyl]-1-benzofuran-3-carboxamide, Polyketide synthase Pks13
著者Aggarwal, A, Sacchettini, J.C.
登録日2021-03-29
公開日2022-02-16
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target.
J.Med.Chem., 65, 2022
6RB0
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BU of 6rb0 by Molmil
STRUCTURE OF ESTER-HYDROLASE EH1AB1 FROM THE METAGENOME OF LAKE ARREO COMPLEXED WITH A DERIVATIVE OF METHYL 4-NITROPHENYL HEXYLPHOSPHONATE
分子名称: EH1AB1, GLYCEROL, methyl hydrogen (R)-hexylphosphonate
著者Cea-Rama, I, Sanz-Aparicio, J.
登録日2019-04-08
公開日2019-12-25
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Genetically engineered proteins with two active sites for enhanced biocatalysis and synergistic chemo- and biocatalysis
Nat Catal, 3, 2020
6RKY
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BU of 6rky by Molmil
STRUCTURE OF ESTER-HYDROLASE EH1AB1 FROM THE METAGENOME OF LAKE ARREO COMPLEXED WITH A DERIVATIVE OF BIPYRIDINE PHOSPHONATE
分子名称: DI(HYDROXYETHYL)ETHER, EH1AB1, GLYCEROL, ...
著者Cea-Rama, I, Sanz-Aparicio, J.
登録日2019-04-30
公開日2019-12-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.79 Å)
主引用文献Genetically engineered proteins with two active sites for enhanced biocatalysis and synergistic chemo- and biocatalysis
Nat Catal, 3, 2020
8PC7
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STRUCTURE OF ESTER-HYDROLASE EH3 FROM THE METAGENOME OF MARINE SEDIMENTS AT MILAZZO HARBOR (SICILY, ITALY) COMPLEXED WITH A DERIVATIVE OF BIPYRIDINE PHOSPHONATE
分子名称: DI(HYDROXYETHYL)ETHER, Esterase, GLYCEROL, ...
著者Cea-Rama, I, Sanz-Aparicio, J.
登録日2023-06-09
公開日2023-07-19
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Transforming an esterase into an enantioselective catecholase through bioconjugation of a versatile metal-chelating inhibitor.
Chem.Commun.(Camb.), 59, 2023
7QI8
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BU of 7qi8 by Molmil
CRYSTAL STRUCTURE OF LYSYL-TRNA SYNTHETASE FROM Mycobacterium tuberculosis COMPLEXED WITH L-LYSINE AND INHIBITOR
分子名称: 2-azanyl-6-[(1~{S},7~{S})-2,2-bis(fluoranyl)-7-oxidanyl-cycloheptyl]-4-methoxy-7~{H}-pyrrolo[3,4-d]pyrimidin-5-one, LYSINE, Lysine--tRNA ligase 1
著者Dawson, A, Robinson, D.A, Tamjar, J, Wyatt, P, Green, S.
登録日2021-12-14
公開日2022-10-19
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Lysyl-tRNA synthetase, a target for urgently needed M. tuberculosis drugs.
Nat Commun, 13, 2022
7QHN
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CRYSTAL STRUCTURE OF LYSYL-TRNA SYNTHETASE FROM Mycobacterium tuberculosis COMPLEXED WITH L-LYSINE and an inhibitor
分子名称: 6-azanyl-2-cyclohexyl-4-fluoranyl-1~{H}-pyrrolo[3,4-c]pyridin-3-one, LYSINE, Lysine--tRNA ligase 1
著者Dawson, A, Robinson, D.A, Tamjar, J, Wyatt, P, Green, S.
登録日2021-12-13
公開日2022-10-19
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.58 Å)
主引用文献Lysyl-tRNA synthetase, a target for urgently needed M. tuberculosis drugs.
Nat Commun, 13, 2022
7QH8
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CRYSTAL STRUCTURE OF LYSYL-TRNA SYNTHETASE FROM Mycobacterium tuberculosis COMPLEXED WITH L-LYSINE
分子名称: GLYCEROL, LYSINE, Lysine--tRNA ligase 1
著者Dawson, A, Robinson, D.A, Tamjar, J, Wyatt, P, Green, S.
登録日2021-12-10
公開日2022-10-19
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Lysyl-tRNA synthetase, a target for urgently needed M. tuberculosis drugs.
Nat Commun, 13, 2022
6I8F
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BU of 6i8f by Molmil
STRUCTURE OF ESTER-HYDROLASE EH1AB1 FROM THE METAGENOME OF LAKE ARREO
分子名称: DI(HYDROXYETHYL)ETHER, EH1AB1, GLYCEROL, ...
著者Cea-Rama, I, Sanz-Aparicio, J.
登録日2018-11-20
公開日2019-11-27
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献Genetically engineered proteins with two active sites for enhanced biocatalysis and synergistic chemo- and biocatalysis
Nat Catal, 3, 2020
7ALZ
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GqqA- a novel type of quorum quenching acylases
分子名称: PHENYLALANINE, Prephenate dehydratase
著者Werner, N, Betzel, C.
登録日2020-10-07
公開日2021-08-04
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献The Komagataeibacter europaeus GqqA is the prototype of a novel bifunctional N-Acyl-homoserine lactone acylase with prephenate dehydratase activity.
Sci Rep, 11, 2021
7AM0
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GqqA- a novel type of quorum quenching acylases
分子名称: PHENYLALANINE, Prephenate dehydratase
著者Werner, N, Betzel, C.
登録日2020-10-07
公開日2021-08-04
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The Komagataeibacter europaeus GqqA is the prototype of a novel bifunctional N-Acyl-homoserine lactone acylase with prephenate dehydratase activity.
Sci Rep, 11, 2021

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件を2024-07-17に公開中

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