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7MDZ
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BU of 7mdz by Molmil
80S rabbit ribosome stalled with benzamide-CHX
分子名称: 18S rRNA, 28S rRNA, 40S ribosomal protein S21, ...
著者Koga, Y, Hoang, E.M, Park, Y, Keszei, A.F.A, Murray, J, Shao, S, Liau, B.B.
登録日2021-04-06
公開日2021-09-01
最終更新日2021-09-15
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Discovery of C13-Aminobenzoyl Cycloheximide Derivatives that Potently Inhibit Translation Elongation.
J.Am.Chem.Soc., 143, 2021
4CRL
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BU of 4crl by Molmil
Crystal structure of human CDK8-Cyclin C in complex with cortistatin A
分子名称: CORTISTATIN A, CYCLIN-C, CYCLIN-DEPENDENT KINASE 8, ...
著者Myers, A.G, Shair, M.D.
登録日2014-02-27
公開日2015-09-23
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Mediator Kinase Inhibition Further Activates Super-Enhancer- Associated Genes in Aml
Nature, 526, 2015
8TQD
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BU of 8tqd by Molmil
NF-Kappa-B1 Bound with a Covalent Inhibitor
分子名称: 1-(2-bromo-4-chlorophenyl)-N-{(3S)-1-[(E)-iminomethyl]pyrrolidin-3-yl}methanesulfonamide, Nuclear factor NF-kappa-B p105 subunit
著者Hilbert, B.J.
登録日2023-08-07
公開日2024-04-24
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献DrugMap: A quantitative pan-cancer analysis of cysteine ligandability.
Cell, 187, 2024
8Q1H
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BU of 8q1h by Molmil
LSD1 Y391K-CoREST bound to Histone H3 N-terminal tail
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, Histone H3.3C, Lysine-specific histone demethylase 1A, ...
著者Barone, M, Mattevi, A.
登録日2023-07-31
公開日2024-05-15
最終更新日2024-07-17
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Uncoupling histone modification crosstalk by engineering lysine demethylase LSD1.
Nat.Chem.Biol., 2024
8Q1J
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BU of 8q1j by Molmil
LSD1 Y391K-CoREST bound to Acetylated K14 of Histone H3
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, Histone H3.3C, Lysine-specific histone demethylase 1A, ...
著者Barone, M, Mattevi, A.
登録日2023-07-31
公開日2024-05-15
最終更新日2024-07-17
実験手法X-RAY DIFFRACTION (2.87 Å)
主引用文献Uncoupling histone modification crosstalk by engineering lysine demethylase LSD1.
Nat.Chem.Biol., 2024
8Q1G
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BU of 8q1g by Molmil
LSD1-CoREST bound to Acetylated K14 of Histone H3
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, Histone H3.3C, Lysine-specific histone demethylase 1A, ...
著者Barone, M, Mattevi, A.
登録日2023-07-31
公開日2024-05-15
最終更新日2024-07-17
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Uncoupling histone modification crosstalk by engineering lysine demethylase LSD1.
Nat.Chem.Biol., 2024

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件を2024-08-14に公開中

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