2VF2
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![BU of 2vf2 by Molmil](/molmil-images/mine/2vf2) | X-ray crystal structure of HsaD from Mycobacterium tuberculosis | 分子名称: | 2-HYDROXY-6-OXO-6-PHENYLHEXA-2,4-DIENOATE HYDROLASE BPHD, GLYCEROL, SULFATE ION | 著者 | Lack, N, Lowe, E.D, Liu, J, Eltis, L.D, Noble, M.E.M, Sim, E, Westwood, I.M. | 登録日 | 2007-10-29 | 公開日 | 2007-11-06 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Structure of Hsad, a Steroid-Degrading Hydrolase, from Mycobacterium Tuberculosis. Acta Crystallogr.,Sect.F, 64, 2008
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5JZS
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![BU of 5jzs by Molmil](/molmil-images/mine/5jzs) | HsaD bound to 3,5-dichloro-4-hydroxybenzoic acid | 分子名称: | 2-hydroxy-6-oxo-6-phenylhexa-2,4-dienoate hydrolase BphD, 3,5-dichloro-4-hydroxybenzoic acid | 著者 | Ryan, A, Polycarpou, E, Lack, N, Evangelopoulos, D, Sieg, C, Halman, A, Bhakta, S, Sinclair, A, Eleftheriadou, O, McHugh, T.D, Keany, S, Lowe, E.D, Ballet, R, Abuhammad, A, Ciulli, A, Sim, E. | 登録日 | 2016-05-17 | 公開日 | 2017-04-05 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.27 Å) | 主引用文献 | Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach. Br. J. Pharmacol., 174, 2017
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2XW7
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![BU of 2xw7 by Molmil](/molmil-images/mine/2xw7) | Structure of Mycobacterium smegmatis putative reductase MS0308 | 分子名称: | DIHYDROFOLATE REDUCTASE, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, SODIUM ION, ... | 著者 | Evangelopoulos, D, Gupta, A, Lack, N, Cronin, N, Daviter, T, Sim, E, Keep, N.H, Bhakta, S. | 登録日 | 2010-11-01 | 公開日 | 2010-12-01 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Characterization of an Oxidoreductase from the Arylamine N-Acetyltransferase Operon in Mycobacterium Smegmatis. FEBS J., 278, 2011
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5WJA
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![BU of 5wja by Molmil](/molmil-images/mine/5wja) | Crystal structure of H107A peptidylglycine alpha-hydroxylating monooxygenase (PHM) in complex with citrate | 分子名称: | CITRATE ANION, COPPER (II) ION, GLYCEROL, ... | 著者 | Maheshwari, S, Rudzka, K, Gabelli, S.B, Amzel, L.M. | 登録日 | 2017-07-21 | 公開日 | 2018-07-18 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Effects of copper occupancy on the conformational landscape of peptidylglycine alpha-hydroxylating monooxygenase. Commun Biol, 1, 2018
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5WKW
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![BU of 5wkw by Molmil](/molmil-images/mine/5wkw) | Crystal structure of apo wild type peptidylglycine alpha-hydroxylating monooxygenase (PHM) | 分子名称: | DI(HYDROXYETHYL)ETHER, GLYCEROL, Peptidyl-glycine alpha-amidating monooxygenase | 著者 | Maheshwari, S, Rudzka, K, Gabelli, S.B, Amzel, L.M. | 登録日 | 2017-07-25 | 公開日 | 2018-07-18 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Effects of copper occupancy on the conformational landscape of peptidylglycine alpha-hydroxylating monooxygenase. Commun Biol, 1, 2018
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5WM0
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![BU of 5wm0 by Molmil](/molmil-images/mine/5wm0) | |
6ALA
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![BU of 6ala by Molmil](/molmil-images/mine/6ala) | Crystal structure of H108A peptidylglycine alpha-hydroxylating monooxygenase (PHM) in complex with citrate | 分子名称: | CITRATE ANION, COPPER (II) ION, GLYCEROL, ... | 著者 | Maheshwari, S, Rudzka, K, Gabelli, S.B, Amzel, L.M. | 登録日 | 2017-08-07 | 公開日 | 2018-07-18 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.59 Å) | 主引用文献 | Effects of copper occupancy on the conformational landscape of peptidylglycine alpha-hydroxylating monooxygenase. Commun Biol, 1, 2018
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6ALV
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![BU of 6alv by Molmil](/molmil-images/mine/6alv) | Crystal structure of H107A-peptidylglycine alpha-hydroxylating monooxygenase (PHM) mutant (no CuH bound) | 分子名称: | AZIDE ION, COPPER (II) ION, GLYCEROL, ... | 著者 | Maheshwari, S, Rudzka, K, Gabelli, S.B, Amzel, L.M. | 登録日 | 2017-08-08 | 公開日 | 2018-07-18 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Effects of copper occupancy on the conformational landscape of peptidylglycine alpha-hydroxylating monooxygenase. Commun Biol, 1, 2018
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6AN3
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![BU of 6an3 by Molmil](/molmil-images/mine/6an3) | Crystal structure of H172A-peptidylglycine alpha-hydroxylating monooxygenase (PHM) mutant soaked with peptide (no CuH bound, no peptide bound) | 分子名称: | COPPER (II) ION, DI(HYDROXYETHYL)ETHER, Peptidyl-glycine alpha-amidating monooxygenase | 著者 | Maheshwari, S, Rudzka, K, Gabelli, S.B, Amzel, L.M. | 登録日 | 2017-08-11 | 公開日 | 2018-07-18 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Effects of copper occupancy on the conformational landscape of peptidylglycine alpha-hydroxylating monooxygenase. Commun Biol, 1, 2018
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6AY0
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![BU of 6ay0 by Molmil](/molmil-images/mine/6ay0) | Crystal structure of H108A peptidylglycine alpha-hydroxylating monooxygenase (PHM) soaked with peptide | 分子名称: | COPPER (II) ION, Peptidyl-glycine alpha-amidating monooxygenase | 著者 | Maheshwari, S, Rudzka, K, Gabelli, S.B, Amzel, L.M. | 登録日 | 2017-09-07 | 公開日 | 2018-07-18 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Effects of copper occupancy on the conformational landscape of peptidylglycine alpha-hydroxylating monooxygenase. Commun Biol, 1, 2018
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6AMP
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![BU of 6amp by Molmil](/molmil-images/mine/6amp) | Crystal structure of H172A PHM (CuH absent, CuM present) | 分子名称: | COPPER (II) ION, Peptidyl-glycine alpha-amidating monooxygenase | 著者 | Maheshwari, S, Rudzka, K, Gabelli, S.B, Amzel, L.M. | 登録日 | 2017-08-10 | 公開日 | 2018-07-18 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.48 Å) | 主引用文献 | Effects of copper occupancy on the conformational landscape of peptidylglycine alpha-hydroxylating monooxygenase. Commun Biol, 1, 2018
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6AO6
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![BU of 6ao6 by Molmil](/molmil-images/mine/6ao6) | Crystal structure of H108A peptidylglycine alpha-hydroxylating monooxygenase (PHM) | 分子名称: | COPPER (II) ION, GLYCEROL, NICKEL (II) ION, ... | 著者 | Maheshwari, S, Rudzka, K, Gabelli, S.B, Amzel, L.M. | 登録日 | 2017-08-15 | 公開日 | 2018-07-18 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.98 Å) | 主引用文献 | Effects of copper occupancy on the conformational landscape of peptidylglycine alpha-hydroxylating monooxygenase. Commun Biol, 1, 2018
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5SYD
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![BU of 5syd by Molmil](/molmil-images/mine/5syd) | |