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5DR8
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BU of 5dr8 by Molmil
Endothiapepsin in complex with fragment 330
分子名称: 2-chlorobenzohydrazide, ACETATE ION, Endothiapepsin, ...
著者Heine, A, Knoerlein, A, Schiebel, J, Klebe, G.
登録日2015-09-15
公開日2016-09-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.47 Å)
主引用文献Crystallographic Fragment Screening of an Entire Library
To Be Published
5EG4
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BU of 5eg4 by Molmil
BOVINE TRYPSIN IN COMPLEX WITH CYCLIC INHIBITOR
分子名称: (13S,16R)-N-(4-carbamimidoylbenzyl)-16-((N-cyclohexylsulfamoyl)amino)-3,9,15-trioxo-2,10,14-triaza-6(1,4)-piperazina-1, 11(1,4)-dibenzenacycloheptadecaphane-13-carboxamide, ACETATE ION, ...
著者Knoerlein, A, Wagner, S, Heine, A, Steinmetzer, T, Klebe, G.
登録日2015-10-26
公開日2016-07-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.32 Å)
主引用文献Optimization of Cyclic Plasmin Inhibitors: From Benzamidines to Benzylamines.
J.Med.Chem., 59, 2016

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件を2024-07-10に公開中

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