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8GB1
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BU of 8gb1 by Molmil
Crystal structure of SAMHD1 dimer bound to deoxyguanosine linked inhibitor
分子名称: 5'-O-[(R)-(3-{[(1M)-3'-bromo[1,1'-biphenyl]-3-carbonyl]amino}propoxy)(hydroxy)phosphoryl]-2'-deoxyguanosine, Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, FE (III) ION
著者Egleston, M, Dong, L, Howlader, A.H, Bhat, S, Orris, B, Bianchet, M.A, Greenberg, M.M, Stivers, J.T.
登録日2023-02-24
公開日2023-06-07
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.46 Å)
主引用文献Deoxyguanosine-Linked Bifunctional Inhibitor of SAMHD1 dNTPase Activity and Nucleic Acid Binding.
Acs Chem.Biol., 18, 2023
8GB2
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BU of 8gb2 by Molmil
Crystal structure of Apo-SAMHD1
分子名称: Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, FE (III) ION
著者Egleston, M, Dong, L, Howlader, A.H, Bhat, S, Orris, B, Bianchet, M.A, Greenberg, M.M, Stivers, J.T.
登録日2023-02-24
公開日2023-06-07
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (3.07 Å)
主引用文献Deoxyguanosine-Linked Bifunctional Inhibitor of SAMHD1 dNTPase Activity and Nucleic Acid Binding.
Acs Chem.Biol., 18, 2023

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件を2024-07-10に公開中

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