8CKH
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8QCC
| E.coli IspE in complex with a ligand (1) | 分子名称: | 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Hamid, R. | 登録日 | 2023-08-25 | 公開日 | 2024-09-11 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | E.coli IspE in complex with a ligand (1) To Be Published
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8QCN
| E.coli IspE in complex with a ligand (2) | 分子名称: | 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, ADENOSINE-5'-DIPHOSPHATE, ~{N}-[3-(4-azanyl-2-oxidanylidene-1~{H}-pyrimidin-5-yl)prop-2-ynyl]cyclopropanesulfonamide | 著者 | Hamid, R. | 登録日 | 2023-08-27 | 公開日 | 2024-09-11 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | E.coli IspE in complex with a ligand (2) To Be Published
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8QC7
| New monoclinic EcIspE | 分子名称: | 4-DIPHOSPHOCYTIDYL-2-C-METHYL-D-ERYTHRITOL, 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, ADENOSINE-5'-DIPHOSPHATE, ... | 著者 | Hamid, R. | 登録日 | 2023-08-25 | 公開日 | 2024-09-11 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | New monoclinic EcIspE To Be Published
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8QCO
| E.coli IspE in complex with a ligand (3) | 分子名称: | 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, ADENOSINE-5'-DIPHOSPHATE, ~{N}-[3-(4-azanyl-2-oxidanylidene-1~{H}-pyrimidin-5-yl)prop-2-ynyl]cyclopentanesulfonamide | 著者 | Hamid, R. | 登録日 | 2023-08-28 | 公開日 | 2024-09-11 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | E.coli IspE in complex with a ligand (3) To Be Published
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8A29
| Apo 1-deoxy-D-xylulose 5-phosphate synthase from Pseudomonas aeruginosa | 分子名称: | 1-deoxy-D-xylulose-5-phosphate synthase, CALCIUM ION, CHLORIDE ION, ... | 著者 | Hamid, R, Adam, S, Lacour, A, Monjas, L, Hirsch, A. | 登録日 | 2022-06-02 | 公開日 | 2023-06-14 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | 1-deoxy-D-xylulose-5-phosphate synthase from Pseudomonas aeruginosa and Klebsiella pneumoniae reveals conformational changes upon cofactor binding. J.Biol.Chem., 299, 2023
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8A4D
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8A45
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8A5K
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8BZX
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3SFK
| Crystal structure of Plasmodium falciparum dihydroorotate dehydrogenase bound with Inhibitor DSM267 | 分子名称: | 2-(1,1-difluoroethyl)-5-methyl-N-[4-(trifluoromethyl)phenyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine, Dihydroorotate dehydrogenase (quinone), mitochondrial, ... | 著者 | Deng, X, Phillips, M. | 登録日 | 2011-06-13 | 公開日 | 2011-07-06 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Structure-Guided Lead Optimization of Triazolopyrimidine-Ring Substituents Identifies Potent Plasmodium falciparum Dihydroorotate Dehydrogenase Inhibitors with Clinical Candidate Potential. J.Med.Chem., 54, 2011
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