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4MTZ
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BU of 4mtz by Molmil
Structure of XIAP-BIR1 in complex with NF023
分子名称: 8-({3-[({3-[(4,6,8-trisulfonaphthalen-1-yl)carbamoyl]phenyl}carbamoyl)amino]benzoyl}amino)naphthalene-1,3,5-trisulfonic acid, E3 ubiquitin-protein ligase XIAP, SULFATE ION, ...
著者Cossu, F, Milani, M, Grassi, S, Mastrangelo, E, Bolognesi, M.
登録日2013-09-20
公開日2014-09-24
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Protein-protein interactions in nfkb pathway: novel tools to promote apoptosis in cancer therapy
To be Published
4OXC
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BU of 4oxc by Molmil
Crystal structure of XIAP BIR1 domain
分子名称: E3 ubiquitin-protein ligase XIAP, ZINC ION
著者Milani, M, Cossu, F, Mastrangelo, E.
登録日2014-02-05
公開日2015-02-11
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献NF023 binding to XIAP-BIR1: Searching drugs for regulation of the NF-kappa B pathway.
Proteins, 83, 2015
4EC4
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BU of 4ec4 by Molmil
XIAP-BIR3 in complex with a potent divalent Smac mimetic
分子名称: (3S,6S,7S,9aS,3'S,6'S,7'S,9a'S)-N,N'-(benzene-1,4-diylbis{butane-4,1-diyl-1H-1,2,3-triazole-1,4-diyl[(S)-phenylmethanediyl]})bis[7-(hydroxymethyl)-6-{[(2S)-2-(methylamino)butanoyl]amino}-5-oxooctahydro-1H-pyrrolo[1,2-a]azepine-3-carboxamide], 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, Baculoviral IAP repeat-containing protein 4, ...
著者Mastrangelo, E, Cossu, F, Bolognesi, M, Milani, M.
登録日2012-03-26
公開日2012-12-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structural insight into inhibitor of apoptosis proteins recognition by a potent divalent smac-mimetic.
Plos One, 7, 2012
4EB9
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BU of 4eb9 by Molmil
cIAP1-BIR3 in complex with a divalent Smac mimetic
分子名称: (3S,6S,7S,9aS,3'S,6'S,7'S,9a'S)-N,N'-(benzene-1,4-diylbis{butane-4,1-diyl-1H-1,2,3-triazole-1,4-diyl[(S)-phenylmethanediyl]})bis[7-(hydroxymethyl)-6-{[(2S)-2-(methylamino)butanoyl]amino}-5-oxooctahydro-1H-pyrrolo[1,2-a]azepine-3-carboxamide], Baculoviral IAP repeat-containing protein 2, ZINC ION
著者Cossu, F, Mastrangelo, E, Bolognesi, M, Milani, M.
登録日2012-03-23
公開日2012-12-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural insight into inhibitor of apoptosis proteins recognition by a potent divalent smac-mimetic.
Plos One, 7, 2012

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件を2024-06-26に公開中

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