3KI0
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ki0 by Molmil](/molmil-images/mine/3ki0) | Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-D | 分子名称: | 3-(morpholin-4-ylmethyl)-1,5-dihydro-6H-[1,2]diazepino[4,5,6-cd]indol-6-one, CHLORIDE ION, Cholix toxin | 著者 | Jorgensen, R, Edwards, P.R, Merrill, A.R. | 登録日 | 2009-10-31 | 公開日 | 2010-10-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.29 Å) | 主引用文献 | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
|
|
3KI7
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ki7 by Molmil](/molmil-images/mine/3ki7) | Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-I | 分子名称: | 2-{2-[4-(pyrrolidin-1-ylmethyl)phenyl]ethyl}-5,6-dihydroimidazo[4,5,1-jk][1,4]benzodiazepin-7(4H)-one, Cholix toxin | 著者 | Jorgensen, R, Edwards, P.R, Merrill, A.R. | 登録日 | 2009-10-31 | 公開日 | 2010-10-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.32 Å) | 主引用文献 | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
|
|
3KI2
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ki2 by Molmil](/molmil-images/mine/3ki2) | |
3KI4
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ki4 by Molmil](/molmil-images/mine/3ki4) | Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-P | 分子名称: | (11bR)-3-oxo-1,2,3,11b-tetrahydrochromeno[4,3,2-de]isoquinoline-10-sulfonic acid, Cholix toxin, GLYCEROL | 著者 | Jorgensen, R, Edwards, P.R, Merrill, A.R. | 登録日 | 2009-10-31 | 公開日 | 2010-10-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
|
|
3KI3
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ki3 by Molmil](/molmil-images/mine/3ki3) | Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-H | 分子名称: | 2-[(dimethylamino)methyl]-5,6-dihydroimidazo[4,5,1-jk][1,4]benzodiazepin-7(4H)-one, Cholix toxin | 著者 | Jorgensen, R, Edwards, P.R, Merrill, A.R. | 登録日 | 2009-10-31 | 公開日 | 2010-10-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.27 Å) | 主引用文献 | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
|
|
3KI1
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ki1 by Molmil](/molmil-images/mine/3ki1) | Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-F | 分子名称: | 2-{4-[3-(dimethylamino)propoxy]phenyl}-5,6-dihydroimidazo[4,5,1-jk][1,4]benzodiazepin-7(4H)-one, Cholix toxin | 著者 | Jorgensen, R, Edwards, P.R, Merrill, A.R. | 登録日 | 2009-10-31 | 公開日 | 2010-10-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.43 Å) | 主引用文献 | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
|
|
3KI6
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ki6 by Molmil](/molmil-images/mine/3ki6) | Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-L | 分子名称: | 8-fluoro-2-(3-piperidin-1-ylpropanoyl)-1,3,4,5-tetrahydrobenzo[c][1,6]naphthyridin-6(2H)-one, Cholix toxin | 著者 | Jorgensen, R, Edwards, P.R, Merrill, A.R. | 登録日 | 2009-10-31 | 公開日 | 2010-10-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published
|
|
3KI5
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ki5 by Molmil](/molmil-images/mine/3ki5) | |
3NY6
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ny6 by Molmil](/molmil-images/mine/3ny6) | Catalytic fragment of cholix toxin from vibrio cholerae in complex with inhibitor V30 | 分子名称: | 2-[(5,6-dimethyl-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(2-hydroxyethyl)acetamide, Cholix toxin, GLYCEROL, ... | 著者 | Merrill, A.R, Jorgensen, R. | 登録日 | 2010-07-14 | 公開日 | 2010-12-29 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.68 Å) | 主引用文献 | Newly discovered and characterized antivirulence compounds inhibit bacterial mono-ADP-ribosyltransferase toxins. Antimicrob.Agents Chemother., 55, 2011
|
|