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3LNM
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BU of 3lnm by Molmil
F233W mutant of the Kv2.1 paddle-Kv1.2 chimera channel
分子名称: (1R)-2-{[(S)-{[(2S)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-1-[(hexadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, F233W mutant of the Kv2.1 paddle-Kv1.2 chimera, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Tao, X, Lee, A, Limapichat, W, Dougherty, D.A, MacKinnon, R.
登録日2010-02-02
公開日2010-04-14
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献A gating charge transfer center in voltage sensors.
Science, 328, 2010
2YOE
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BU of 2yoe by Molmil
X-ray structure of a pentameric ligand gated ion channel from Erwinia chrysanthemi (ELIC) in complex with GABA and flurazepam
分子名称: CYS-LOOP LIGAND-GATED ION CHANNEL, Flurazepam, GAMMA-AMINO-BUTANOIC ACID
著者Spurny, R, Brams, M, Nury, H, Legrand, P, Ulens, C.
登録日2012-10-23
公開日2012-10-31
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.9 Å)
主引用文献Pentameric Ligand-Gated Ion Channel Elic is Activated by Gaba and Modulated by Benzodiazepines.
Proc.Natl.Acad.Sci.USA, 109, 2012
7S7V
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BU of 7s7v by Molmil
Crystal structure of iNicSnFR3a Fluorescent Nicotine Sensor
分子名称: iNicSnFR 3.0 Fluorescent Nicotine Sensor
著者Fan, C, Shivange, A.V, Looger, L.L, Lester, H.A, Rees, D.C.
登録日2021-09-17
公開日2021-10-13
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Correction: Fluorescence activation mechanism and imaging of drug permeation with new sensors for smoking-cessation ligands.
Elife, 11, 2022
7S7T
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BU of 7s7t by Molmil
iNicSnFR3a Nicotine Sensor comprising Periplasmic Binding sequence plus Fluorescent Sequence with varenicline bound
分子名称: IODIDE ION, VARENICLINE, iNicSnFR 3.0 Fluorescent Nicotine Sensor
著者Fan, C, Shivange, A.V, Looger, L.L, Lester, H.A, Rees, D.C.
登録日2021-09-17
公開日2021-10-13
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Correction: Fluorescence activation mechanism and imaging of drug permeation with new sensors for smoking-cessation ligands.
Elife, 11, 2022
7S7U
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BU of 7s7u by Molmil
Crystal structure of iNicSnFR3a Fluorescent Nicotine Sensor with nicotine bound
分子名称: iNicSnFR 3.0 Fluorescent Nicotine Sensor
著者Fan, C, Shivange, A.V, Looger, L.L, Lester, H.A, Rees, D.C.
登録日2021-09-17
公開日2021-10-13
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Correction: Fluorescence activation mechanism and imaging of drug permeation with new sensors for smoking-cessation ligands.
Elife, 11, 2022
4A98
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BU of 4a98 by Molmil
X-ray structure of a pentameric ligand gated ion channel from Erwinia chrysanthemi (ELIC) in complex with bromoflurazepam
分子名称: 7-BROMO-1-[2-(DIETHYLAMINO)ETHYL]-5-(2-FLUOROPHENYL)-1,3-DIHYDRO-2H-1,4-BENZODIAZEPIN-2-ONE, CYS-LOOP LIGAND-GATED ION CHANNEL
著者Spurny, R, Brams, M, Nury, H, Legrand, P, Ulens, C.
登録日2011-11-24
公開日2012-10-17
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.61 Å)
主引用文献Pentameric Ligand-Gated Ion Channel Elic is Activated by Gaba and Modulated by Benzodiazepines.
Proc.Natl.Acad.Sci.USA, 109, 2012
4A97
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BU of 4a97 by Molmil
X-ray structure of a pentameric ligand gated ion channel from Erwinia chrysanthemi (ELIC) in complex with zopiclone
分子名称: (5R)-6-(5-chloropyridin-2-yl)-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyrazin-5-yl 4-methylpiperazine-1-carboxylate, CYS-LOOP LIGAND-GATED ION CHANNEL
著者Spurny, R, Brams, M, Ulens, C.
登録日2011-11-24
公開日2012-10-17
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.343 Å)
主引用文献Pentameric Ligand-Gated Ion Channel Elic is Activated by Gaba and Modulated by Benzodiazepines.
Proc.Natl.Acad.Sci.USA, 109, 2012
6EFR
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BU of 6efr by Molmil
Crystal Structure of iNicSnFR 1.0
分子名称: iNicSnFR 1.0, a genetically encoded nicotine biosensor,Green fluorescent protein
著者Shivange, A.V, Borden, P.M.
登録日2018-08-17
公開日2019-01-23
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Nicotinic Drugs in the Endoplasmic Reticulum: Beginning the Inside-out Pathway of Addiction and Therapy
J.Gen.Physiol., 2019

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件を2024-07-24に公開中

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