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7KH8
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BU of 7kh8 by Molmil
Human LMPTP in complex with inhibitor
分子名称: 3-[(2,6-dichlorophenyl)methyl]-8-(2-methylphenyl)-3H-purin-6-amine, Low molecular weight phosphotyrosine protein phosphatase, NITRATE ION
著者Stanford, S.M, Diaz, M.A, Ardecky, R.J, Zou, J, Roosild, T, Holmes, Z.J, Hedrick, M.P, Rodiles, S, Santelli, E, Chung, T.D.Y, Jackson, M.R, Bottini, N, Pinkerton, A.B.
登録日2020-10-20
公開日2021-05-19
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Discovery of Orally Bioavailable Purine-Based Inhibitors of the Low-Molecular-Weight Protein Tyrosine Phosphatase.
J.Med.Chem., 64, 2021
8FBZ
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BU of 8fbz by Molmil
Crystal Structure of apo human Glutathione Synthetase Y270E
分子名称: GLYCEROL, Glutathione synthetase, SULFATE ION
著者Stanford, S.M, Santelli, E, Sankaran, B, Murali, R, Bottini, N.
登録日2022-11-30
公開日2024-05-08
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献Targeting prostate tumor low-molecular weight tyrosine phosphatase for oxidation-sensitizing therapy.
Sci Adv, 10, 2024

221051

件を2024-06-12に公開中

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