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3S86
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BU of 3s86 by Molmil
Crystal Structure of TM0159 with bound IMP
分子名称: INOSINIC ACID, Nucleoside-triphosphatase, SULFATE ION
著者Sommerhalter, M, Smith, C, Awwad, K, Desai, A.
登録日2011-05-27
公開日2012-06-06
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural and functional characterization of a noncanonical nucleoside triphosphate pyrophosphatase from Thermotoga maritima.
Acta Crystallogr.,Sect.D, 69, 2013
4WH4
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BU of 4wh4 by Molmil
Protein GB1 Quadruple Mutant I6H/N8H/K28H/Q32H
分子名称: GLYCEROL, Immunoglobulin G-binding protein G, SULFATE ION
著者Cunningham, T.C, Horne, W.S, Saxena, S.
登録日2014-09-19
公開日2015-08-05
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The double-histidine Cu2+-binding motif: a highly rigid, site-specific spin probe for electron spin resonance distance measurements.
Angew.Chem.Int.Ed.Engl., 54, 2015
5EW9
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BU of 5ew9 by Molmil
Crystal Structure of Aurora A Kinase Domain Bound to MK-5108
分子名称: 4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acid, Aurora kinase A
著者Shiau, A.K, Motamedi, A.
登録日2015-11-20
公開日2016-01-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.181 Å)
主引用文献A Cell Biologist's Field Guide to Aurora Kinase Inhibitors.
Front Oncol, 5, 2015
4YUR
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BU of 4yur by Molmil
Crystal Structure of Plk4 Kinase Domain Bound to Centrinone
分子名称: 2-({2-fluoro-4-[(2-fluoro-3-nitrobenzyl)sulfonyl]phenyl}sulfanyl)-5-methoxy-N-(3-methyl-1H-pyrazol-5-yl)-6-(morpholin-4-yl)pyrimidin-4-amine, Serine/threonine-protein kinase PLK4
著者Shiau, A.K, Motamedi, A.
登録日2015-03-19
公開日2015-06-17
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Cell biology. Reversible centriole depletion with an inhibitor of Polo-like kinase 4.
Science, 348, 2015
3KJS
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BU of 3kjs by Molmil
Crystal Structure of T. cruzi DHFR-TS with 3 high affinity DHFR inhibitors: DQ1 inhibitor complex
分子名称: 1,2-ETHANEDIOL, Dihydrofolate reductase-thymidylate synthase, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Schormann, N, Senkovich, O, Chattopadhyay, D.
登録日2009-11-03
公開日2010-06-09
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Synthesis and characterization of potent inhibitors of Trypanosoma cruzi dihydrofolate reductase.
Bioorg.Med.Chem., 18, 2010

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件を2024-10-16に公開中

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