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8Q3C
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BU of 8q3c by Molmil
Structure of Selenomonas ruminantium lactate dehydrogenase I85R mutant
分子名称: CHLORIDE ION, L-lactate dehydrogenase, NITRATE ION, ...
著者Bertrand, Q, Coquille, S, Iorio, A, Sterpone, F, Madern, D.
登録日2023-08-03
公開日2023-11-01
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Biochemical, structural and dynamical characterizations of the lactate dehydrogenase from Selenomonas ruminantium provide information about an intermediate evolutionary step prior to complete allosteric regulation acquisition in the super family of lactate and malate dehydrogenases.
J.Struct.Biol., 215, 2023
4N7Q
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BU of 4n7q by Molmil
Crystal structure of eukaryotic THIC from A. thaliana
分子名称: COBALT (II) ION, HEXANE-1,6-DIOL, Phosphomethylpyrimidine synthase, ...
著者Coquille, S.C, Roux, C, Mehta, A, Begley, T.P, Fitzpatrick, T.B, Thore, S.
登録日2013-10-16
公開日2013-11-13
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献High-resolution crystal structure of the eukaryotic HMP-P synthase (THIC) from Arabidopsis thaliana.
J.Struct.Biol., 184, 2013
4WN4
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BU of 4wn4 by Molmil
Crystal structure of designed cPPR-polyA protein
分子名称: Pentatricopeptide repeat protein
著者Coquille, S.C, Filipovska, A, Chia, T.S, Rajappa, L, Lingford, J.P, Razif, M.F.M, Thore, S, Rackham, O.
登録日2014-10-10
公開日2014-12-24
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.85 Å)
主引用文献An artificial PPR scaffold for programmable RNA recognition.
Nat Commun, 5, 2014
4WSL
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BU of 4wsl by Molmil
Crystal structure of designed cPPR-polyC protein
分子名称: Pentatricopeptide repeat protein
著者Coquille, S.C, Filipovska, A, Chia, T.S, Rajappa, L, Lingford, J.P, Razif, M.F.M, Thore, S, Rackham, O.
登録日2014-10-28
公開日2014-12-24
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.7 Å)
主引用文献An artificial PPR scaffold for programmable RNA recognition.
Nat Commun, 5, 2014
4H67
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BU of 4h67 by Molmil
Crystal structure of HMP synthase Thi5 from S. cerevisiae
分子名称: PYRIDOXAL-5'-PHOSPHATE, Pyrimidine precursor biosynthesis enzyme THI5, SULFATE ION
著者Coquille, S.C, Roux, C, Fitzpatrick, T, Thore, S.
登録日2012-09-19
公開日2012-10-17
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The Last Piece in the Vitamin B1 Biosynthesis Puzzle: STRUCTURAL AND FUNCTIONAL INSIGHT INTO YEAST 4-AMINO-5-HYDROXYMETHYL-2-METHYLPYRIMIDINE PHOSPHATE (HMP-P) SYNTHASE.
J.Biol.Chem., 287, 2012
4H65
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BU of 4h65 by Molmil
Crystal structure of SeMet derivative of HMP synthase Thi5 from S. cerevisiae
分子名称: Pyrimidine precursor biosynthesis enzyme THI5
著者Coquille, S.C, Roux, C, Fitzpatrick, T, Thore, S.
登録日2012-09-19
公開日2012-10-17
最終更新日2013-01-23
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The Last Piece in the Vitamin B1 Biosynthesis Puzzle: STRUCTURAL AND FUNCTIONAL INSIGHT INTO YEAST 4-AMINO-5-HYDROXYMETHYL-2-METHYLPYRIMIDINE PHOSPHATE (HMP-P) SYNTHASE.
J.Biol.Chem., 287, 2012
4H6D
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BU of 4h6d by Molmil
Crystal structure of PLP-soaked HMP synthase Thi5 from S. cerevisiae
分子名称: PYRIDOXAL-5'-PHOSPHATE, Pyrimidine precursor biosynthesis enzyme THI5
著者Coquille, S.C, Roux, C, Fitzpatrick, T, Thore, S.
登録日2012-09-19
公開日2012-10-17
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献The Last Piece in the Vitamin B1 Biosynthesis Puzzle: STRUCTURAL AND FUNCTIONAL INSIGHT INTO YEAST 4-AMINO-5-HYDROXYMETHYL-2-METHYLPYRIMIDINE PHOSPHATE (HMP-P) SYNTHASE.
J.Biol.Chem., 287, 2012
4PJS
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BU of 4pjs by Molmil
Crystal structure of designed (SeMet)-cPPR-NRE protein
分子名称: CALCIUM ION, Pentatricopeptide repeat protein
著者Coquille, S.C, Filipovska, A, Chia, T.S, Rajappa, L, Lingford, J.P, Razif, M.F.M, Thore, S, Rackham, O.
登録日2014-05-12
公開日2014-12-24
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献An artificial PPR scaffold for programmable RNA recognition.
Nat Commun, 5, 2014
4PJQ
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BU of 4pjq by Molmil
Crystal structure of designed cPPR-polyG protein
分子名称: Pentatricopeptide repeat protein
著者Coquille, S.C, Filipovska, A, Chia, T.S, Rajappa, L, Lingford, J.P, Razif, M.F.M, Thore, S, Rackham, O.
登録日2014-05-12
公開日2014-12-24
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.353 Å)
主引用文献An artificial PPR scaffold for programmable RNA recognition.
Nat Commun, 5, 2014
4PJR
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BU of 4pjr by Molmil
Crystal structure of designed cPPR-NRE protein
分子名称: MAGNESIUM ION, Pentatricopeptide repeat protein
著者Coquille, S.C, Filipovska, A, Chia, T.S, Rajappa, L, Lingford, J.P, Razif, M.F.M, Thore, S, Rackham, O.
登録日2014-05-12
公開日2014-12-24
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献An artificial PPR scaffold for programmable RNA recognition.
Nat Commun, 5, 2014
7NAY
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BU of 7nay by Molmil
Crystal structure of lactate dehydrogenase from Selenomonas ruminantium with NADH.
分子名称: 1,2-ETHANEDIOL, BORIC ACID, L-lactate dehydrogenase, ...
著者Bertrand, Q, Robin, A, Girard, E, Madern, D.
登録日2021-01-25
公開日2021-02-10
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献Biochemical, structural and dynamical characterizations of the lactate dehydrogenase from Selenomonas ruminantium provide information about an intermediate evolutionary step prior to complete allosteric regulation acquisition in the super family of lactate and malate dehydrogenases.
J.Struct.Biol., 215, 2023
8B75
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BU of 8b75 by Molmil
CRYSTAL STRUCTURE OF HUMAN SOLUBLE ADENYLYL CYCLASE IN COMPLEX WITH THE INHIBITOR TDI-011861
分子名称: Adenylate cyclase type 10, [(3~{R})-4-[2-[2-[[3-(2-azanyl-6-chloranyl-pyrimidin-4-yl)-1-[bis(fluoranyl)methyl]pyrazol-4-yl]methyl]phenoxy]ethyl]morpholin-3-yl]methanol
著者Steegborn, C, Kehr, M.
登録日2022-09-28
公開日2023-03-29
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献Design, Synthesis, and Pharmacological Evaluation of Second-Generation Soluble Adenylyl Cyclase (sAC, ADCY10) Inhibitors with Slow Dissociation Rates.
J.Med.Chem., 65, 2022

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件を2024-06-12に公開中

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