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1OCE
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BU of 1oce by Molmil
ACETYLCHOLINESTERASE (E.C. 3.1.1.7) COMPLEXED WITH MF268
分子名称: ACETYLCHOLINESTERASE, CIS-2,6-DIMETHYLMORPHOLINOOCTYLCARBAMYLESEROLINE
著者Bartolucci, C, Perola, E, Cellai, L, Brufani, M, Lamba, D.
登録日1998-06-12
公開日1999-05-18
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献"Back door" opening implied by the crystal structure of a carbamoylated acetylcholinesterase.
Biochemistry, 38, 1999
398D
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BU of 398d by Molmil
3'-DNA-RNA-5' JUNCTION FORMED DURING INITIATION OF MINUS-STRAND SYNTHESIS OF HIV REPLICATION
分子名称: DNA/RNA (5'-R(*GP*CP*CP*AP)-D(*CP*TP*GP*C)-3'), RNA (5'-R(*GP*CP*AP*GP*UP*GP*GP*C)-3')
著者Mueller, U, Meier, G, Mochi-Onori, A, Cellai, L, Heumann, H.
登録日1998-05-04
公開日1998-10-06
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Crystal structure of an eight-base pair duplex containing the 3'-DNA-RNA-5' junction formed during initiation of minus-strand synthesis of HIV replication.
Biochemistry, 37, 1998
1BYX
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BU of 1byx by Molmil
CHIMERIC HYBRID DUPLEX R(GCAGUGGC).R(GCCA)D(CTGC) COMPRISING THE TRNA-DNA JUNCTION FORMED DURING INITIATION OF HIV-1 REVERSE TRANSCRIPTION
分子名称: DNA/RNA (5'-R(*GP*CP*CP*A)-D(P*CP*TP*GP*C)-3'), RNA (5'-R(*GP*CP*AP*GP*UP*GP*GP*C)-3')
著者Szyperski, T, Goette, M, Billeter, M, Perola, E, Cellai, L.
登録日1998-10-20
公開日1999-10-20
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献NMR structure of the chimeric hybrid duplex r(gcaguggc).r(gcca)d(CTGC) comprising the tRNA-DNA junction formed during initiation of HIV-1 reverse transcription.
J.Biomol.NMR, 13, 1999
2BAG
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BU of 2bag by Molmil
3D Structure of Torpedo californica acetylcholinesterase complexed with Ganstigmine
分子名称: 1S,3AS,8AS-TRIMETHYL-1-OXIDO-1,2,3,3A,8,8A-HEXAHYDROPYRROLO[2,3-B]INDOL-5-YL 2-ETHYLPHENYLCARBAMATE, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Lamba, D, Bartolucci, C, Siotto, M, Racchi, M, Villetti, G, Delcanale, M.
登録日2005-10-14
公開日2006-08-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural Determinants of Torpedo californica Acetylcholinesterase Inhibition by the Novel and Orally Active Carbamate Based Anti-Alzheimer Drug Ganstigmine (CHF-2819)
J.Med.Chem., 49, 2006

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