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human beta-II tryptase in complex with 4-(3-Aminomethyl-phenyl)- piperidin-1-yl-(5-phenethyl- pyridin-3-yl)-methanone
分子名称:	1-[3-(1-{[5-(2-PHENYLETHYL)PYRIDIN-3-YL]CARBONYL}PIPERIDIN-4-YL)PHENYL]METHANAMINE, HUMAN BETA2 TRYPTASE
著者	Maignan, S, Guilloteau, J.-P, Dupuy, A, Levell, J, Astles, P, Eastwood, P, Cairns, J, Houille, O, Aldous, S, Merriman, G, Whiteley, B, Pribish, J, Czekaj, M, Liang, G, Davidson, J, Harrison, T, Morley, A, Watson, S, Fenton, G, Mccarthy, C, Romano, J, Mathew, R, Engers, D, Gardyan, M, Sides, K, Kwong, J, Tsay, J, Rebello, S, Shen, L, Wang, J, Luo, Y, Giardino, O, Lim, H.-K, Smith, K, Pauls, H.
登録日	2005-03-09
公開日	2005-03-22
最終更新日	2023-12-13
実験手法	X-RAY DIFFRACTION (2.2 Å)
主引用文献	Structure Based Design of 4-(3-Aminomethylphenyl) Piperidinyl-1-Amides: Novel, Potent, Selective, and Orally Bioavailable Inhibitors of Bii Tryptase Bioorg.Med.Chem., 13, 2005

beta-tryptase inhibitor
分子名称:	1-{3-[1-({5-[(2-fluorophenyl)ethynyl]furan-2-yl}carbonyl)piperidin-4-yl]phenyl}methanamine, TRYPTASE ALPHA/BETA-1
著者	Mathieu, M, Maignan, S.
登録日	2011-11-04
公開日	2012-01-25
最終更新日	2024-05-01
実験手法	X-RAY DIFFRACTION (2.05 Å)
主引用文献	Structure-Based Library Design and the Discovery of a Potent and Selective Mast Cell Beta-Tryptase Inhibitor as an Oral Therapeutic Agent. Bioorg.Med.Chem.Lett., 22, 2012

Crystal structure of benzophenone synthase from Garcinia mangostana L. pericarps reveals basis for substrate specificity and catalysis
分子名称:	2,4,6-trihydroxybenzophenone synthase, GLYCEROL, IMIDAZOLE, ...
著者	Songsiriritthigul, C, Nualkaew, N, Chen, C.-J.
登録日	2020-06-12
公開日	2020-12-09
最終更新日	2023-11-29
実験手法	X-RAY DIFFRACTION (2.301 Å)
主引用文献	Crystal structure of benzophenone synthase from Garcinia mangostana L. pericarps reveals basis for substrate specificity and catalysis. Acta Crystallogr.,Sect.F, 76, 2020