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2VBQ
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BU of 2vbq by Molmil
Structure of AAC(6')-Iy in complex with bisubstrate analog CoA-S- monomethyl-acetylneamine.
分子名称: (3R,9Z)-17-[(2R,3S,4R,5R,6R)-5-amino-6-{[(1R,2R,3S,4R,6S)-4,6-diamino-2,3-dihydroxycyclohexyl]oxy}-3,4-dihydroxytetrahydro-2H-pyran-2-yl]-3-hydroxy-2,2-dimethyl-4,8,15-trioxo-12-thia-5,9,16-triazaheptadec-9-en-1-yl [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-hydroxy-3-(phosphonooxy)tetrahydrofuran-2-yl]methyl dihydrogen diphosphate, AMINOGLYCOSIDE 6'-N-ACETYLTRANSFERASE, GLYCEROL, ...
著者Vetting, M.W, Magalhaes, M.L, Freiburger, L, Gao, F, Auclair, K, Blanchard, J.S.
登録日2007-09-14
公開日2008-01-08
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Kinetic and Structural Analysis of Bisubstrate Inhibition of the Salmonella Enterica Aminoglycoside 6'-N-Acetyltransferase.
Biochemistry, 47, 2008
6T90
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BU of 6t90 by Molmil
OCT4-SOX2-bound nucleosome - SHL-6
分子名称: DNA (146-MER), Green fluorescent protein,POU domain, class 5, ...
著者Michael, A.K, Kempf, G, Cavadini, S, Bunker, R.D, Thoma, N.H.
登録日2019-10-25
公開日2020-05-06
最終更新日2020-07-08
実験手法ELECTRON MICROSCOPY (3.05 Å)
主引用文献Mechanisms of OCT4-SOX2 motif readout on nucleosomes.
Science, 368, 2020
6T93
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BU of 6t93 by Molmil
Nucleosome with OCT4-SOX2 motif at SHL-6
分子名称: DNA (153-MER), Histone H2A type 1-B/E, Histone H2B type 1-J, ...
著者Michael, A.K, Kempf, G, Cavadini, S, Bunker, R.D, Thoma, N.H.
登録日2019-10-25
公開日2020-05-06
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (3.49 Å)
主引用文献Mechanisms of OCT4-SOX2 motif readout on nucleosomes.
Science, 368, 2020
6YOV
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BU of 6yov by Molmil
OCT4-SOX2-bound nucleosome - SHL+6
分子名称: DNA (142-MER), Green fluorescent protein,POU domain, class 5, ...
著者Michael, A.K, Kempf, G, Cavadini, S, Bunker, R.D, Thoma, N.H.
登録日2020-04-15
公開日2020-05-06
最終更新日2020-07-08
実験手法ELECTRON MICROSCOPY (3.42 Å)
主引用文献Mechanisms of OCT4-SOX2 motif readout on nucleosomes.
Science, 368, 2020
8AXW
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BU of 8axw by Molmil
The structure of mouse AsterC (GramD1c) with Ezetimibe
分子名称: (3~{R},4~{S})-1-(4-fluorophenyl)-3-[(3~{S})-3-(4-fluorophenyl)-3-oxidanyl-propyl]-4-(4-hydroxyphenyl)azetidin-2-one, CHLORIDE ION, ETHANOL, ...
著者Fairall, L, Xiao, X, Burger, L, Tontonoz, P, Schwabe, J.W.R.
登録日2022-09-01
公開日2023-09-13
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Aster-dependent nonvesicular transport facilitates dietary cholesterol uptake.
Science, 382, 2023
6YIZ
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BU of 6yiz by Molmil
Crystal structure of PqsR (MvfR) ligand-binding domain in complex with triazolo-pyridine inverse agonist A
分子名称: 7-oxidanylidene-8-[2-(4-sulfonaphthalen-1-yl)hydrazinyl]-8~{H}-naphthalene-1,3-disulfonic acid, MAGNESIUM ION, Transcriptional regulator MvfR, ...
著者Schmelz, S, Blankenfeldt, W.
登録日2020-04-01
公開日2021-04-14
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.163 Å)
主引用文献A New PqsR Inverse Agonist Potentiates Tobramycin Efficacy to Eradicate Pseudomonas aeruginosa Biofilms.
Adv Sci, 8, 2021
5NJJ
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BU of 5njj by Molmil
PTB domain of human Numb isoform-1
分子名称: ALA-TYR-ILE-GLY-PRO-PTR-LEU, Protein numb homolog, SULFATE ION
著者Mapelli, M, Di Fiore, P.P.
登録日2017-03-29
公開日2017-12-13
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献A Numb-Mdm2 fuzzy complex reveals an isoform-specific involvement of Numb in breast cancer.
J. Cell Biol., 217, 2018
5NJK
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BU of 5njk by Molmil
PTB domain of human Numb isoform-1
分子名称: ALA-TYR-ILE-GLY-PRO-PTR-LEU, Protein numb homolog, SULFATE ION
著者Mapelli, M, Di Fiore, P.P.
登録日2017-03-29
公開日2017-12-13
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.13 Å)
主引用文献A Numb-Mdm2 fuzzy complex reveals an isoform-specific involvement of Numb in breast cancer.
J. Cell Biol., 217, 2018

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件を2024-09-11に公開中

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