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Crystal Structure of the first bromodomain of human BRDT in complex with the inhibitor JQ1
分子名称:	(6S)-6-(2-tert-butoxy-2-oxoethyl)-4-(4-chlorophenyl)-2,3,9-trimethyl-6,7-dihydrothieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-10-ium, Bromodomain testis-specific protein, POTASSIUM ION
著者	Filippakopoulos, P, Picaud, S, Qi, J, Felletar, I, Canning, P, Muniz, J, von Delft, F, Bountra, C, Arrowsmith, C.H, Edwards, A, Bradner, J, Knapp, S, Structural Genomics Consortium (SGC)
登録日	2012-06-15
公開日	2012-07-11
最終更新日	2023-09-13
実験手法	X-RAY DIFFRACTION (2.23 Å)
主引用文献	Small-Molecule Inhibition of BRDT for Male Contraception. Cell(Cambridge,Mass.), 150, 2012

Brd4 Bromodomain 2 in Complex with Acetylated Rel Peptide
分子名称:	2,3-DIHYDROXY-1,4-DITHIOBUTANE, Bromodomain-containing protein 4, Rel Peptide
著者	Zhang, H, Nair, S.K.
登録日	2013-05-22
公開日	2013-06-26
最終更新日	2024-10-09
実験手法	X-RAY DIFFRACTION (2 Å)
主引用文献	Brd4 maintains constitutively active NF-kappa B in cancer cells by binding to acetylated RelA. Oncogene, 33, 2014

Crystal Structure of Brd4 Bromodomain 1 in Complex with Acetylated Rel Peptide
分子名称:	Bromodomain-containing protein 4, Rel peptide
著者	Zhang, H, Nair, S.K.
登録日	2013-05-22
公開日	2013-06-26
最終更新日	2014-05-14
実験手法	X-RAY DIFFRACTION (1.5 Å)
主引用文献	Brd4 maintains constitutively active NF-kappa B in cancer cells by binding to acetylated RelA. Oncogene, 33, 2014