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5YAW
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BU of 5yaw by Molmil
Fragment-based Drug Discovery of inhibitors to block PDEdelta-RAS protein-protein interaction
分子名称: 3-[(4-methoxyphenyl)methylsulfanyl]-5-(2-methylpropyl)-4-(phenylmethyl)-1,2,4-triazole, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta
著者Bing, X, Yanlian, L, Danyan, C.
登録日2017-09-01
公開日2018-09-05
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.027 Å)
主引用文献Fragment-based Drug Discovery of inhibitors to block PDEdelta-RAS protein-protein interaction
To Be Published
5YAV
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BU of 5yav by Molmil
Fragment-based Drug Discovery of inhibitors to block PDEdelta-RAS protein-protein interaction
分子名称: 1-phenyl-5-propan-2-ylsulfanyl-1,2,3,4-tetrazole, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta
著者Bing, X, Yanlian, L, Danyan, C.
登録日2017-09-01
公開日2018-09-05
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.989 Å)
主引用文献Fragment-based Drug Discovery of inhibitors to block PDEdelta-RAS protein-protein interaction
To Be Published
5YOU
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BU of 5you by Molmil
Crystal structure of BRD4-BD1 bound with hjp64
分子名称: (3~{R})-4-cyclopropyl-~{N},1,3-trimethyl-~{N}-(4-methylphenyl)-2-oxidanylidene-3~{H}-quinoxaline-6-carboxamide, Bromodomain-containing protein 4
著者Bing, X, Jianping, H, Yanlian, L, Danyan, C.
登録日2017-10-31
公開日2018-11-07
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.503 Å)
主引用文献Crystal structure of BRD4-BD1 bound with hjp64
To Be Published
6INS
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BU of 6ins by Molmil
X-RAY ANALYSIS OF THE SINGLE CHAIN B29-A1 PEPTIDE-LINKED INSULIN MOLECULE. A COMPLETELY INACTIVE ANALOGUE
分子名称: INSULIN, ZINC ION
著者Derewenda, U, Derewenda, Z, Dodson, E.J, Dodson, G.G, Bing, X, Markussen, J.
登録日1992-11-25
公開日1994-01-31
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献X-ray analysis of the single chain B29-A1 peptide-linked insulin molecule. A completely inactive analogue.
J.Mol.Biol., 220, 1991
8YM7
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BU of 8ym7 by Molmil
Crystal structure of Lysine Specific Demethylase 1 (LSD1) with JH-45
分子名称: 4-[5-(4-azanylpiperidin-1-yl)-8-(4-methylphenyl)pyrido[3,4-b]pyrazin-7-yl]-2-fluoranyl-benzenecarbonitrile, FLAVIN-ADENINE DINUCLEOTIDE, Lysine-specific histone demethylase 1A, ...
著者Zhiyan, D, Danyan, C, Hong, J, Tongchao, L, Bing, X.
登録日2024-03-08
公開日2024-05-22
実験手法X-RAY DIFFRACTION (2.83 Å)
主引用文献Discovery of Novel LSD1 Inhibitors for the Treatment of Autosomal Dominant Polycystic Kidney Disease
To Be Published
5XHY
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BU of 5xhy by Molmil
BRD4 bound with compound Bdi1
分子名称: Bromodomain-containing protein 4, ~{N}-(4-cyclopropyl-1,3,3-trimethyl-2-oxidanylidene-quinoxalin-6-yl)-4-methyl-benzenesulfonamide
著者Xiong, B, Cao, D, Li, Y.
登録日2017-04-25
公開日2018-05-02
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.976 Å)
主引用文献BRD4 bound with compound Bdi1
To Be Published

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件を2024-07-10に公開中

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