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8T2H
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DYRK1A complex with DYR530
分子名称: (4P)-4-{(3M)-3-[3-fluoro-4-(4-methylpiperazin-1-yl)phenyl]-2-methyl-3H-imidazo[4,5-b]pyridin-5-yl}pyridin-2-amine, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, GLYCEROL, ...
著者Montfort, W.R, Basantes, L.E.
登録日2023-06-06
公開日2024-05-15
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Discovery of DYR684, a Potent, Selective, Metabolically Stable, DYRK1A/B PROTAC utilizing a Novel Cereblon Molecular Glue
To Be Published

221716

件を2024-06-26に公開中

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