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2X00
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BU of 2x00 by Molmil
CRYSTAL STRUCTURE OF A-ACHBP IN COMPLEX WITH GYMNODIMINE A
分子名称: GYMNODIMINE A, SOLUBLE ACETYLCHOLINE RECEPTOR
著者Bourne, Y, Radic, Z, Araoz, R, Talley, T.T, Benoit, E, Servent, D, Taylor, P, Molgo, J, Marchot, P.
登録日2009-12-04
公開日2010-03-02
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural Determinants in Phycotoxins and Achbp Conferring High Affinity Binding and Nicotinic Achr Antagonism.
Proc.Natl.Acad.Sci.USA, 107, 2010
2WZY
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BU of 2wzy by Molmil
Crystal structure of A-AChBP in complex with 13-desmethyl spirolide C
分子名称: 13-DESMETHYL SPIROLIDE C, SOLUBLE ACETYLCHOLINE RECEPTOR
著者Bourne, Y, Radic, Z, Araoz, R, Talley, T.T, Benoit, E, Servent, D, Taylor, P, Molgo, J, Marchot, P.
登録日2009-12-03
公開日2010-03-02
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Structural Determinants in Phycotoxins and Achbp Conferring High Affinity Binding and Nicotinic Achr Antagonism.
Proc.Natl.Acad.Sci.USA, 107, 2010
4XK9
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BU of 4xk9 by Molmil
Crystal structure of A-AChBP in complex with pinnatoxin G
分子名称: CHLORIDE ION, Pinnatoxin G, Soluble acetylcholine receptor
著者Bourne, Y, Sulzenbacher, G, Marchot, P.
登録日2015-01-10
公開日2015-06-03
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Marine Macrocyclic Imines, Pinnatoxins A and G: Structural Determinants and Functional Properties to Distinguish Neuronal alpha 7 from Muscle alpha 12 beta gamma delta nAChRs.
Structure, 23, 2015
4XHE
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BU of 4xhe by Molmil
Crystal Structure of A-AChBP in complex with pinnatoxin A
分子名称: CALCIUM ION, CHLORIDE ION, Pinnatoxin A, ...
著者Bourne, Y, Sulzenbacher, G, Marchot, P.
登録日2015-01-05
公開日2015-06-03
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Marine Macrocyclic Imines, Pinnatoxins A and G: Structural Determinants and Functional Properties to Distinguish Neuronal alpha 7 from Muscle alpha 12 beta gamma delta nAChRs.
Structure, 23, 2015
8QX2
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BU of 8qx2 by Molmil
Aplysia californica acetylcholine-binding protein in complex with racemic spiroimine (+)/(-)-4
分子名称: ISOPROPYL ALCOHOL, Soluble acetylcholine receptor, Spiroimine (+)-4 R
著者Sulzenbacher, G, Bourne, Y, Marchot, P.
登録日2023-10-20
公開日2024-04-03
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The Cyclic Imine Core Common to the Marine Macrocyclic Toxins Is Sufficient to Dictate Nicotinic Acetylcholine Receptor Antagonism.
Mar Drugs, 22, 2024
8QTL
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BU of 8qtl by Molmil
Aplysia californica acetylcholine-binding protein in complex with Spiroimine (-)-4 S
分子名称: CHLORIDE ION, ISOPROPYL ALCOHOL, Soluble acetylcholine receptor, ...
著者Sulzenbacher, G, Bourne, Y, Marchot, P.
登録日2023-10-12
公開日2024-04-03
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献The Cyclic Imine Core Common to the Marine Macrocyclic Toxins Is Sufficient to Dictate Nicotinic Acetylcholine Receptor Antagonism.
Mar Drugs, 22, 2024
8Q1M
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BU of 8q1m by Molmil
Aplysia californica acetylcholine-binding protein in complex with Spiroimine (+)-4 R
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, Soluble acetylcholine receptor, ...
著者Sulzenbacher, G, Bourne, Y, Marchot, P.
登録日2023-07-31
公開日2024-04-03
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The Cyclic Imine Core Common to the Marine Macrocyclic Toxins Is Sufficient to Dictate Nicotinic Acetylcholine Receptor Antagonism.
Mar Drugs, 22, 2024

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件を2024-07-24に公開中

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