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4PM0
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BU of 4pm0 by Molmil
PDE7A catalytic domain in complex with 2-(Cyclopentylamino)thieno[3,2-d]pyrimidin-4(3H)-one derivative
分子名称: 2-(cyclopentylamino)-3-ethyl-7-ethynylthieno[3,2-d]pyrimidin-4(3H)-one, High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A, MAGNESIUM ION, ...
著者Kawai, K, Endo, Y, Asano, T, Amano, S, Sawada, K, Ueo, N, Takahashi, N, Sonoda, Y, Kamei, N, Nagata, N.
登録日2014-05-20
公開日2014-12-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Discovery of 2-(Cyclopentylamino)thieno[3,2-d]pyrimidin-4(3H)-one Derivatives as a New Series of Potent Phosphodiesterase 7 Inhibitors.
J.Med.Chem., 57, 2014
2D05
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BU of 2d05 by Molmil
Chitosanase From Bacillus circulans mutant K218P
分子名称: Chitosanase, SULFATE ION
著者Fukamizo, T, Amano, S, Yamaguchi, K, Yoshikawa, T, Katsumi, T, Saito, J, Suzuki, M, Miki, K, Nagata, Y, Ando, A.
登録日2005-07-25
公開日2005-12-06
最終更新日2021-11-10
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Bacillus circulans MH-K1 Chitosanase: Amino Acid Residues Responsible for Substrate Binding
J.Biochem.(Tokyo), 138, 2005
4Y2B
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BU of 4y2b by Molmil
Co-crystal structure of 3-ethyl-2-(isopropylamino)-7-(pyridin-3-yl)thieno[3,2-d]pyrimidin-4(3H)-one bound to PDE7A
分子名称: 3-ethyl-2-(propan-2-ylamino)-7-(pyridin-3-yl)thieno[3,2-d]pyrimidin-4(3H)-one, High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A, MAGNESIUM ION, ...
著者Endo, Y, Kawai, K, Asano, T, Amano, S, Asanuma, Y, Sawada, K, Onodera, Y, Ueo, N, Takahashi, N, Sonoda, Y, Kamei, N, Irie, T.
登録日2015-02-09
公開日2015-04-08
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献2-(Isopropylamino)thieno[3,2-d]pyrimidin-4(3H)-one derivatives as selective phosphodiesterase 7 inhibitors with potent in vivo efficacy
Bioorg.Med.Chem.Lett., 25, 2015
3IJM
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BU of 3ijm by Molmil
The structure of a restriction endonuclease-like fold superfamily protein from Spirosoma linguale.
分子名称: GLYCEROL, SODIUM ION, SULFATE ION, ...
著者Cuff, M.E, Tesar, C, Samano, S, Bearden, J, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2009-08-04
公開日2009-09-22
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The structure of a restriction endonuclease-like fold superfamily protein from Spirosoma linguale.
TO BE PUBLISHED
2VDA
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BU of 2vda by Molmil
Solution structure of the SecA-signal peptide complex
分子名称: MALTOPORIN, TRANSLOCASE SUBUNIT SECA
著者Gelis, I, Bonvin, A.M.J.J, Keramisanou, D, Koukaki, M, Gouridis, G, Karamanou, S, Economou, A, Kalodimos, C.G.
登録日2007-10-01
公開日2007-11-27
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural Basis for Signal-Sequence Recognition by the Translocase Motor Seca as Determined by NMR
Cell(Cambridge,Mass.), 131, 2007
2FSH
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BU of 2fsh by Molmil
Complex SecA:AMP-PNP from Escherichia coli
分子名称: PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, Preprotein translocase secA subunit
著者Papanikolau, Y, Petratos, K, Economou, A.
登録日2006-01-23
公開日2007-01-16
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of dimeric SecA, the Escherichia coli preprotein translocase motor.
J.Mol.Biol., 366, 2007
2FSG
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BU of 2fsg by Molmil
Complex SecA:ATP from Escherichia coli
分子名称: ADENOSINE-5'-TRIPHOSPHATE, Preprotein translocase secA subunit
著者Papanikolau, Y, Petratos, K, Economou, A.
登録日2006-01-23
公開日2007-01-16
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of dimeric SecA, the Escherichia coli preprotein translocase motor.
J.Mol.Biol., 366, 2007
7OSL
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BU of 7osl by Molmil
Cryo-EM structure of nonameric EPEC SctV-C
分子名称: Translocator EscV
著者Fahrenkamp, D, Wald, J, Yuan, B, Marlovits, T.C.
登録日2021-06-09
公開日2021-09-29
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Structural Dynamics of the Functional Nonameric Type III Translocase Export Gate.
J.Mol.Biol., 433, 2021
2FSF
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BU of 2fsf by Molmil
Escherichia coli SecA, the preprotein translocase dimeric ATPase
分子名称: Preprotein translocase secA subunit
著者Papanikolau, Y, Petratos, K, Economou, A.
登録日2006-01-23
公開日2007-01-16
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of dimeric SecA, the Escherichia coli preprotein translocase motor.
J.Mol.Biol., 366, 2007
2FSI
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BU of 2fsi by Molmil
Complex SecA:ADP from Escherichia coli
分子名称: ADENOSINE-5'-DIPHOSPHATE, Preprotein translocase secA subunit
著者Papanikolau, Y, Petratos, K, Economou, A.
登録日2006-01-23
公開日2007-01-16
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献Structure of dimeric SecA, the Escherichia coli preprotein translocase motor.
J.Mol.Biol., 366, 2007

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