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8VJP
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BU of 8vjp by Molmil
Histidine-covalent stapled alpha-helical peptide (155H1) targeting hMcl-1
分子名称: (4Z)-oct-4-en-1-ol, (S~1~R)-3-carbamoyl-4-methoxybenzene-1-sulfinic acid, Histidine-covalent stapled alpha-helical peptide, ...
著者Muzzarelli, K.M, Assar, Z, Alboreggia, G, Pellecchia, M.
登録日2024-01-07
公開日2024-05-15
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.13 Å)
主引用文献Histidine-Covalent Stapled Alpha-Helical Peptides Targeting hMcl-1.
J.Med.Chem., 67, 2024
8GH7
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BU of 8gh7 by Molmil
142D6 bound to BIR3-XIAP
分子名称: 2-(2-(2-(2-(2-(2-ETHOXYETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHANOL, BIR3 inhibitor MAA-CHG-PRO-ZHW, E3 ubiquitin-protein ligase XIAP, ...
著者Garza-Granados, A, McGuire, J, Baggio, C, Pellecchia, M, Pegan, S.D.
登録日2023-03-09
公開日2023-07-05
最終更新日2023-07-12
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Characterization of a Potent and Orally Bioavailable Lys-Covalent Inhibitor of Apoptosis Protein (IAP) Antagonist.
J.Med.Chem., 66, 2023

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件を2024-10-16に公開中

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