8VJP
| Histidine-covalent stapled alpha-helical peptide (155H1) targeting hMcl-1 | 分子名称: | (4Z)-oct-4-en-1-ol, (S~1~R)-3-carbamoyl-4-methoxybenzene-1-sulfinic acid, Histidine-covalent stapled alpha-helical peptide, ... | 著者 | Muzzarelli, K.M, Assar, Z, Alboreggia, G, Pellecchia, M. | 登録日 | 2024-01-07 | 公開日 | 2024-05-15 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.13 Å) | 主引用文献 | Histidine-Covalent Stapled Alpha-Helical Peptides Targeting hMcl-1. J.Med.Chem., 67, 2024
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8GH7
| 142D6 bound to BIR3-XIAP | 分子名称: | 2-(2-(2-(2-(2-(2-ETHOXYETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHANOL, BIR3 inhibitor MAA-CHG-PRO-ZHW, E3 ubiquitin-protein ligase XIAP, ... | 著者 | Garza-Granados, A, McGuire, J, Baggio, C, Pellecchia, M, Pegan, S.D. | 登録日 | 2023-03-09 | 公開日 | 2023-07-05 | 最終更新日 | 2023-07-12 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Characterization of a Potent and Orally Bioavailable Lys-Covalent Inhibitor of Apoptosis Protein (IAP) Antagonist. J.Med.Chem., 66, 2023
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