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1LD6
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BU of 1ld6 by Molmil
STRUCTURE OF BPTI_8A MUTANT
分子名称: PANCREATIC TRYPSIN INHIBITOR
著者Cierpicki, T, Otlewski, J.
登録日2002-04-08
公開日2002-09-11
最終更新日2021-10-27
実験手法SOLUTION NMR
主引用文献NMR structures of two variants of bovine pancreatic trypsin inhibitor (BPTI) reveal unexpected influence of mutations on protein structure and stability.
J.Mol.Biol., 321, 2002
6IAD
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BU of 6iad by Molmil
Apo crystal structure of archaeal Methanocaldococcus infernus Elp3 (del1-54)
分子名称: Histone acetyltransferase, ELP3 family, SULFATE ION
著者Lin, T.Y, Glatt, S.
登録日2018-11-26
公開日2019-02-20
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献The Elongator subunit Elp3 is a non-canonical tRNA acetyltransferase.
Nat Commun, 10, 2019
6IA8
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BU of 6ia8 by Molmil
Apo crystal structure of archaeal Methanocaldococcus infernus Elp3 (del1-19)
分子名称: Histone acetyltransferase, ELP3 family, SULFATE ION
著者Lin, T.Y, Glatt, S.
登録日2018-11-26
公開日2019-02-20
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The Elongator subunit Elp3 is a non-canonical tRNA acetyltransferase.
Nat Commun, 10, 2019
6IAZ
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BU of 6iaz by Molmil
The archaeal Methanocaldococcus infernus Elp3 with N-terminus deletion (1-46)
分子名称: Histone acetyltransferase, ELP3 family, SULFATE ION
著者Lin, T.Y, Glatt, S.
登録日2018-11-28
公開日2019-02-20
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.901 Å)
主引用文献The Elongator subunit Elp3 is a non-canonical tRNA acetyltransferase.
Nat Commun, 10, 2019
7WBM
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BU of 7wbm by Molmil
Crystal structure of Legionella pneumophila effector protein Lpg0081
分子名称: Lpg0081, [(2R,3S,4R,5R)-5-(6-AMINOPURIN-9-YL)-3,4-DIHYDROXY-OXOLAN-2-YL]METHYL [HYDROXY-[[(2R,3S,4R,5S)-3,4,5-TRIHYDROXYOXOLAN-2-YL]METHOXY]PHOSPHORYL] HYDROGEN PHOSPHATE
著者Lee, J, Kim, H, Oh, B.H.
登録日2021-12-17
公開日2022-06-15
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Reversible modification of mitochondrial ADP/ATP translocases by paired Legionella effector proteins.
Proc.Natl.Acad.Sci.USA, 119, 2022
7WBK
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BU of 7wbk by Molmil
Crystal structure of Legionella pneumophila effector protein Lpg0081
分子名称: Lpg0081, SULFATE ION
著者Lee, J, Kim, H, Oh, B.H.
登録日2021-12-16
公開日2022-06-15
実験手法X-RAY DIFFRACTION (2.74 Å)
主引用文献Reversible modification of mitochondrial ADP/ATP translocases by paired Legionella effector proteins.
Proc.Natl.Acad.Sci.USA, 119, 2022
6IA6
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BU of 6ia6 by Molmil
Crystal structure of the bacterial Dehalococcoides mccartyi Elp3 with desulfo-CoA
分子名称: DESULFO-COENZYME A, ELP3 family, FE2/S2 (INORGANIC) CLUSTER, ...
著者Lin, T.Y, Glatt, S.
登録日2018-11-26
公開日2019-02-20
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The Elongator subunit Elp3 is a non-canonical tRNA acetyltransferase.
Nat Commun, 10, 2019
5B6F
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BU of 5b6f by Molmil
Crystal structure of the Fab fragment of an anti-Leukotriene C4 monoclonal antibody complexed with LTC4
分子名称: (5~{S},6~{R},7~{E},9~{E},11~{Z},14~{Z})-6-[(2~{R})-2-[[(4~{S})-4-azanyl-5-oxidanyl-5-oxidanylidene-pentanoyl]amino]-3-(2-hydroxy-2-oxoethylamino)-3-oxidanylidene-propyl]sulfanyl-5-oxidanyl-icosa-7,9,11,14-tetraenoic acid, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, SULFATE ION, ...
著者Sugahara, M, Ago, H, Saino, H, Miyano, M.
登録日2016-05-27
公開日2017-05-31
最終更新日2019-07-24
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structure of the Fab fragment of an anti-Leukotriene C4 monoclonal antibody complexed with LTC4
To Be Published
1BDC
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BU of 1bdc by Molmil
STAPHYLOCOCCUS AUREUS PROTEIN A, IMMUNOGLOBULIN-BINDING B DOMAIN, NMR, 10 STRUCTURES
分子名称: STAPHYLOCOCCUS AUREUS PROTEIN A
著者Gouda, H, Torigoe, H, Saito, A, Sato, M, Arata, Y, Shimada, I.
登録日1996-06-28
公開日1997-01-11
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Three-dimensional solution structure of the B domain of staphylococcal protein A: comparisons of the solution and crystal structures.
Biochemistry, 31, 1992
2ZM4
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BU of 2zm4 by Molmil
Crystal structure of imidazo quinoxaline 1 bound to the kinase domain of human LCK, activated form (auto-phosphorylated on TYR394)
分子名称: DIMETHYL SULFOXIDE, N-(2-chloro-6-methylphenyl)-8-[(3S)-3-methylpiperazin-1-yl]imidazo[1,5-a]quinoxalin-4-amine, Proto-oncogene tyrosine-protein kinase LCK, ...
著者Tsuji, E.
登録日2008-04-11
公開日2008-10-14
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The importance of CH/pi hydrogen bonds in rational drug design: An ab initio fragment molecular orbital study to leukocyte-specific protein tyrosine (LCK) kinase
Bioorg.Med.Chem., 16, 2008
2ZYB
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BU of 2zyb by Molmil
Crystal structure of phenylimidazo pyrazin 2 bound to the kinase domain of human LCK, (auto-phosphorylated on TYR394)
分子名称: N-(2,6-dimethylphenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine, Proto-oncogene tyrosine-protein kinase LCK, SULFATE ION
著者Tsuji, E.
登録日2009-01-19
公開日2009-02-03
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献The importance of CH/pi hydrogen bonds in rational drug design: An ab initio fragment molecular orbital study to leukocyte-specific protein tyrosine (LCK) kinase
Bioorg.Med.Chem., 16, 2008
2ZM1
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BU of 2zm1 by Molmil
Crystal structure of imidazo pyrazin 1 bound to the kinase domain of human LCK, (auto-phosphorylated on TYR394)
分子名称: DIMETHYL SULFOXIDE, N-(2-chlorophenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine, Proto-oncogene tyrosine-protein kinase LCK, ...
著者Tsuji, E.
登録日2008-04-10
公開日2008-10-14
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The importance of CH/pi hydrogen bonds in rational drug design: An ab initio fragment molecular orbital study to leukocyte-specific protein tyrosine (LCK) kinase
Bioorg.Med.Chem., 16, 2008
1BDD
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BU of 1bdd by Molmil
STAPHYLOCOCCUS AUREUS PROTEIN A, IMMUNOGLOBULIN-BINDING B DOMAIN, NMR, MINIMIZED AVERAGE STRUCTURE
分子名称: STAPHYLOCOCCUS AUREUS PROTEIN A
著者Gouda, H, Torigoe, H, Saito, A, Sato, M, Arata, Y, Shimada, I.
登録日1996-06-28
公開日1997-01-11
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Three-dimensional solution structure of the B domain of staphylococcal protein A: comparisons of the solution and crystal structures.
Biochemistry, 31, 1992
1CQZ
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BU of 1cqz by Molmil
CRYSTAL STRUCTURE OF MURINE SOLUBLE EPOXIDE HYDROLASE.
分子名称: EPOXIDE HYDROLASE
著者Argiriadi, M.A, Morisseau, C, Hammock, B.D, Christianson, D.W.
登録日1999-08-12
公開日1999-11-19
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Detoxification of environmental mutagens and carcinogens: structure, mechanism, and evolution of liver epoxide hydrolase.
Proc.Natl.Acad.Sci.USA, 96, 1999
3A7D
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BU of 3a7d by Molmil
Crystal Structures of rat Catechol-O-Methyltransferase complexed with new bi-substrate type inhibitor
分子名称: 5'-deoxy-5'-[4-({[(2,3-dihydroxy-5-nitrophenyl)carbonyl]amino}methyl)-1H-1,2,3-triazol-1-yl]adenosine, Catechol O-methyltransferase, MAGNESIUM ION, ...
著者Tsuji, E.
登録日2009-09-26
公開日2010-09-15
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Hit to Lead: Comprehensive Strategy of de novo Scaffold Generation by FBDD. Part 2: Ligand Fishing using Mass Spectrometry by Detection of Ligand-Protein Non-Covalent Complex after Matrix Click Chemistry
To be Published
3A7E
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BU of 3a7e by Molmil
Crystal structure of human COMT complexed with SAM and 3,5-dinitrocatechol
分子名称: 3,5-DINITROCATECHOL, Catechol O-methyltransferase, MAGNESIUM ION, ...
著者Tsuji, E.
登録日2009-09-26
公開日2010-09-15
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Hit to Lead: Comprehensive Strategy of de novo Scaffold Generation by FBDD. Part 1: In silico Fragments Linking and Verification of Spatial Proximity using Inter Ligand NOE Approachs
To be Published
1JWD
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BU of 1jwd by Molmil
Ca2+-induced Structural Changes in Calcyclin: High-resolution Solution Structure of Ca2+-bound Calcyclin.
分子名称: Calcyclin
著者Maler, L, Sastry, M, Chazin, W.J.
登録日2001-09-04
公開日2002-03-27
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献A structural basis for S100 protein specificity derived from comparative analysis of apo and Ca(2+)-calcyclin
J.Mol.Biol., 317, 2002
2DCP
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BU of 2dcp by Molmil
Fully automated NMR structure determination of the ENTH-VHS domain AT3G16270 from Arabidopsis thaliana
分子名称: hypothetical protein (RAFL09-17-B18)
著者Lopez-Mendez, B, Guntert, P.
登録日2006-01-12
公開日2006-10-17
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Automated Protein Structure Determination from NMR Spectra
J.Am.Chem.Soc., 128, 2006

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件を2024-07-17に公開中

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