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1V6I
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BU of 1v6i by Molmil
Peanut lectin-lactose complex in acidic pH
分子名称: CALCIUM ION, Galactose-binding lectin, MANGANESE (II) ION, ...
著者Kundhavai Natchiar, S, Arockia Jeyaprakash, A, Ramya, T.N.C, Thomas, C.J, Suguna, K, Surolia, A, Vijayan, M.
登録日2003-12-01
公開日2004-02-10
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural plasticity of peanut lectin: an X-ray analysis involving variation in pH, ligand binding and crystal structure.
Acta Crystallogr.,Sect.D, 60, 2004
5LQQ
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BU of 5lqq by Molmil
Structure of Autotaxin (ENPP2) with LM350
分子名称: 3-(6-chloranyl-2-methyl-1-phenyl-indol-3-yl)sulfanylbenzoic acid, CALCIUM ION, Ectonucleotide pyrophosphatase/phosphodiesterase family member 2, ...
著者Keune, W.J, Heidebrecht, T, Castelmur, E, Joosten, R.P, Perrakis, A.
登録日2016-08-17
公開日2016-12-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode.
J. Med. Chem., 60, 2017
6I9K
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BU of 6i9k by Molmil
Crystal structure of Jumping Spider Rhodopsin-1 bound to 9-cis retinal
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Kumopsin1, RETINAL
著者Varma, N, Mutt, E, Muehle, J, Panneels, V, Terakita, A, Deupi, X, Nogly, P, Schertler, F.X.G, Lesca, E.
登録日2018-11-23
公開日2019-07-03
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.145 Å)
主引用文献Crystal structure of jumping spider rhodopsin-1 as a light sensitive GPCR.
Proc.Natl.Acad.Sci.USA, 116, 2019
1RXG
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BU of 1rxg by Molmil
DEACETOXYCEPHALOSPORIN C SYNTHASE COMPLEXED WITH FE(II) AND 2-OXOGLUTARATE
分子名称: 2-OXOGLUTARIC ACID, DEACETOXYCEPHALOSPORIN C SYNTHASE, FE (III) ION, ...
著者Valegard, K, Terwisscha Van Scheltinga, A.C, Lloyd, M.D, Hara, T, Ramaswamy, S, Perrakis, A, Thompson, A, Lee, H.J, Baldwin, J.E, Shofield, C.J, Hajdu, J, Andersson, I.
登録日1998-06-05
公開日1999-06-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structure of a cephalosporin synthase.
Nature, 394, 1998
1RXF
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BU of 1rxf by Molmil
DEACETOXYCEPHALOSPORIN C SYNTHASE COMPLEXED WITH FE(II)
分子名称: DEACETOXYCEPHALOSPORIN C SYNTHASE, FE (III) ION
著者Valegard, K, Terwisscha Van Scheltinga, A.C, Lloyd, M.D, Hara, T, Ramaswamy, S, Perrakis, A, Thompson, A, Lee, H.J, Baldwin, J.E, Schofield, C.J, Hajdu, J, Andersson, I.
登録日1998-06-05
公開日1999-06-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structure of a cephalosporin synthase.
Nature, 394, 1998
6GVJ
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BU of 6gvj by Molmil
Human Mps1 kinase domain with ordered activation loop
分子名称: CHLORIDE ION, Dual specificity protein kinase TTK, GLYCEROL
著者Roorda, J.C, Hiruma, Y, Joosten, R.P, Perrakis, A.
登録日2018-06-21
公開日2019-01-09
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献A crystal structure of the human protein kinase Mps1 reveals an ordered conformation of the activation loop.
Proteins, 87, 2019
1RCQ
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BU of 1rcq by Molmil
The 1.45 A crystal structure of alanine racemase from a pathogenic bacterium, Pseudomonas aeruginosa, contains both internal and external aldimine forms
分子名称: D-LYSINE, PYRIDOXAL-5'-PHOSPHATE, catabolic alanine racemase DadX
著者Le Magueres, P, Im, H, Dvorak, A, Strych, U, Benedik, M, Krause, K.L.
登録日2003-11-04
公開日2004-06-01
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Crystal structure at 1.45 A resolution of alanine racemase from a pathogenic bacterium, Pseudomonas aeruginosa, contains both internal and external aldimine forms.
Biochemistry, 42, 2003
7Z3K
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BU of 7z3k by Molmil
Autotaxin in complex with orthosteric site-binder CpdA
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 7alpha-hydroxycholesterol, CALCIUM ION, ...
著者Salgado-Polo, F, Ford, P, Heckmann, B, Perrakis, A.
登録日2022-03-02
公開日2023-01-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Autotaxin facilitates selective LPA receptor signaling.
Cell Chem Biol, 30, 2023
7Z3L
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BU of 7z3l by Molmil
Autotaxin in complex with hybrid compound ziritaxestat (GLPG1690)
分子名称: 2-[[2-ethyl-8-methyl-6-[4-[2-(3-oxidanylazetidin-1-yl)-2-oxidanylidene-ethyl]piperazin-1-yl]imidazo[1,2-a]pyridin-3-yl]-methyl-amino]-4-(4-fluorophenyl)-1,3-thiazole-5-carbonitrile, 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Salgado-Polo, F, Ford, P, Heckmann, B, Perrakis, A.
登録日2022-03-02
公開日2023-01-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Autotaxin facilitates selective LPA receptor signaling.
Cell Chem Biol, 30, 2023
7ZOM
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BU of 7zom by Molmil
Crystal structure of N-terminal catalytic domain of human PLAAT3
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, Phospholipase A and acyltransferase 3
著者von Castelmur, E, Perrakis, A.
登録日2022-04-26
公開日2023-04-26
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.601 Å)
主引用文献Crystal structure of N-terminal catalytic domain of human PLAAT3
To Be Published
7ZU3
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BU of 7zu3 by Molmil
Crystal Structure of Human Parechovirus 1 2A protein lacking the C-terminal oligomerisation helix
分子名称: Protein 2A
著者von Castelmur, E, Perrakis, A.
登録日2022-05-11
公開日2023-05-24
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献Human Parechovirus 1 2A protein
To Be Published
7ZUO
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BU of 7zuo by Molmil
Crystal Structure of Ljungan virus 4 2A2 protein, P212121 form
分子名称: 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, DI(HYDROXYETHYL)ETHER, ...
著者von Castelmur, E, Perrakis, A.
登録日2022-05-12
公開日2023-05-24
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献Structural Plasticity of Parechovirus H/NC-motif 2A proteins
To Be Published
7ZUA
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BU of 7zua by Molmil
Crystal Structure of Ljungan virus 4 2A2 protein I222 crystal form
分子名称: ACETATE ION, Protein 2A
著者von Castelmur, E, Perrakis, A.
登録日2022-05-11
公開日2023-05-24
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献Structural plasticity of Parechovirus family H-box 2A proteins
To Be Published
7ZV1
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BU of 7zv1 by Molmil
Crystal Structure of Aichivirus A 2A protein L64M, L109M mutant
分子名称: Protein 2A
著者von Castelmur, E, Perrakis, A.
登録日2022-05-13
公開日2023-05-31
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献Structural and functional repurposing of picornavirus H/NC-motif 2A proteins
To Be Published
7ZTW
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BU of 7ztw by Molmil
Crystal Structure of Human Parechovirus 1 2A protein
分子名称: ACETATE ION, Protein 2A, SODIUM ION
著者von Castelmur, E, Perrakis, A.
登録日2022-05-11
公開日2023-05-24
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Human Parechovirus 1 2A protein
To Be Published
7ZU4
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BU of 7zu4 by Molmil
Crystal Structure of Human Parechovirus 1 2A protein lacking the C-terminal oligomerisation helix
分子名称: 1,2-ETHANEDIOL, GLYCEROL, Protein 2A, ...
著者von Castelmur, E, Perrakis, A.
登録日2022-05-11
公開日2023-05-24
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Human Parechovirus 1 2A protein
To Be Published
7ZV6
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BU of 7zv6 by Molmil
Crystal Structure of Aichivirus A 2A protein
分子名称: Protein 2A
著者von Castelmur, E, Perrakis, A.
登録日2022-05-13
公開日2023-05-24
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.83 Å)
主引用文献Structural and functional repurposing of picornavirus H/NC-motif 2A proteins
To Be Published
5FWL
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BU of 5fwl by Molmil
Atomic cryoEM structure of Hsp90-Cdc37-Cdk4 complex
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CYCLIN-DEPENDENT KINASE 4, HEAT SHOCK PROTEIN HSP 90 BETA, ...
著者Verba, K.A, Wang, R.Y.R, Arakawa, A, Liu, Y, Yokoyama, S, Agard, D.A.
登録日2016-02-18
公開日2016-07-06
最終更新日2019-10-23
実験手法ELECTRON MICROSCOPY (9 Å)
主引用文献Atomic Structure of Hsp90-Cdc37-Cdk4 Reveals that Hsp90 Traps and Stabilizes an Unfolded Kinase.
Science, 352, 2016
8A2F
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BU of 8a2f by Molmil
Crystal Structure of Ljunganvirus 1 2A protein
分子名称: 2A protein
著者von Castelmur, E, Zhu, L, Wang, X, Fry, E, Ren, J, Perrakis, A, Stuart, D.I.
登録日2022-06-03
公開日2023-06-14
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献Structural plasticity of 2A proteins in the Parechovirus family
To Be Published
8A2E
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BU of 8a2e by Molmil
Crystal Structure of Human Parechovirus 3 2A protein
分子名称: 2A protein, GLYCEROL, SULFATE ION
著者von Castelmur, E, Zhu, L, wang, X, Fry, E, Ren, J, Perrakis, A, Stuart, D.I.
登録日2022-06-03
公開日2023-06-14
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献Structural plasticity of 2A proteins in the Parechovirus family.
To Be Published
8A2G
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BU of 8a2g by Molmil
Crystal structure of Sebokelevirus 2A2 protein
分子名称: 1,2-ETHANEDIOL, 2A2 protein, TETRAETHYLENE GLYCOL
著者Zhu, L, Von Castelmur, E, Whang, X, Ren, J, Fry, E, Perrakis, A, Stuart, D.I.
登録日2022-06-03
公開日2023-06-14
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Structural plasticity of 2A proteins in the Parechovirus family
to be published
5HJ0
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BU of 5hj0 by Molmil
Crystal Structure of Mis18 'Yippee-like' Domain
分子名称: Kinetochore protein mis18, ZINC ION
著者Medina-Pritchard, B, Subramanian, L, Allshire, R, Arockia Jeyaprakash, A.
登録日2016-01-12
公開日2016-03-09
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.64 Å)
主引用文献Centromere localization and function of Mis18 requires Yippee-like domain-mediated oligomerization.
Embo Rep., 17, 2016
5FWK
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BU of 5fwk by Molmil
Atomic cryoEM structure of Hsp90-Cdc37-Cdk4 complex
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CYCLIN-DEPENDENT KINASE 4, HEAT SHOCK PROTEIN HSP 90 BETA, ...
著者Verba, K.A, Wang, R.Y.R, Arakawa, A, Liu, Y, Yokoyama, S, Agard, D.A.
登録日2016-02-17
公開日2016-07-06
最終更新日2019-08-21
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Atomic Structure of Hsp90-Cdc37-Cdk4 Reveals that Hsp90 Traps and Stabilizes an Unfolded Kinase.
Science, 352, 2016
5FWP
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BU of 5fwp by Molmil
Atomic cryoEM structure of Hsp90-Cdc37-Cdk4 complex
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CYCLIN-DEPENDENT KINASE 4, HEAT SHOCK PROTEIN HSP 90 BETA, ...
著者Verba, K.A, Wang, R.Y.R, Arakawa, A, Liu, Y, Yokoyama, S, Agard, D.A.
登録日2016-02-18
公開日2016-10-26
最終更新日2019-12-18
実験手法ELECTRON MICROSCOPY (7.2 Å)
主引用文献Atomic Structure of Hsp90:Cdc37:Cdk4 Reveals that Hsp90 Traps and Stabilizes an Unfolded Kinase.
Science, 352, 2016
5FWM
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BU of 5fwm by Molmil
Atomic cryoEM structure of Hsp90-Cdc37-Cdk4 complex
分子名称: ADENOSINE-5'-TRIPHOSPHATE, CYCLIN-DEPENDENT KINASE 4, HEAT SHOCK PROTEIN HSP 90 BETA, ...
著者Verba, K.A, Wang, R.Y.R, Arakawa, A, Liu, Y, Yokoyama, S, Agard, D.A.
登録日2016-02-18
公開日2016-07-06
最終更新日2019-10-23
実験手法ELECTRON MICROSCOPY (8 Å)
主引用文献Atomic Structure of Hsp90-Cdc37-Cdk4 Reveals that Hsp90 Traps and Stabilizes an Unfolded Kinase.
Science, 352, 2016

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