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4Y5L
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BU of 4y5l by Molmil
Endothiapepsin in its apo form
分子名称: ACETATE ION, DI(HYDROXYETHYL)ETHER, Endothiapepsin, ...
著者Schiebel, J, Heine, A, Klebe, G.
登録日2015-02-11
公開日2016-03-02
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (0.99 Å)
主引用文献Crystallographic Fragment Screening of an Entire Library
To Be Published
5ZE7
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BU of 5ze7 by Molmil
UDP Glucose alpha tetrahydrobiopterin glycosyltransferase from Synechococcus species PCC 7942 - apo form
分子名称: UDP-glucose:tetrahydrobiopterin glucosyltransferase
著者Killivalavan, A, Lee, K.H.
登録日2018-02-27
公開日2019-03-06
最終更新日2019-12-04
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献UDP Glucose alpha tetrahydrobiopterin glycosyltransferase from Synechococcus species PCC 7942 - apo form
To Be Published
5ZES
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BU of 5zes by Molmil
UDP Glucose alpha tetrahydrobiopterin glycosyltransferase from Synechococcus species PCC 7942 - UDP complex
分子名称: GLYCEROL, UDP-glucose:tetrahydrobiopterin glucosyltransferase, URIDINE-5'-DIPHOSPHATE
著者Killivalavan, A, Lee, K.H.
登録日2018-02-27
公開日2019-03-06
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献UDP Glucose alpha tetrahydrobiopterin glycosyltransferase from Synechococcus species PCC 7942 - UDP complex
To Be Published
6S1N
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BU of 6s1n by Molmil
Human polymerase delta holoenzyme Conformer 2
分子名称: DNA polymerase delta catalytic subunit, DNA polymerase delta subunit 2, DNA polymerase delta subunit 3, ...
著者Lancey, C, Hamdan, S.M, De Biasio, A.
登録日2019-06-19
公開日2019-12-25
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (4.86 Å)
主引用文献Structure of the processive human Pol delta holoenzyme.
Nat Commun, 11, 2020
6S2V
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BU of 6s2v by Molmil
Structure of the N-terminal catalytic region of T. thermophilus Rel
分子名称: (P)ppGpp synthetase I, SpoT/RelA, CHLORIDE ION, ...
著者Garcia-Pino, A.
登録日2019-06-22
公開日2020-07-08
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.96 Å)
主引用文献A nucleotide-switch mechanism mediates opposing catalytic activities of Rel enzymes.
Nat.Chem.Biol., 16, 2020
5ZEP
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BU of 5zep by Molmil
M. smegmatis hibernating state 70S ribosome structure
分子名称: 16S rRNA, 23S rRNA, 30S ribosomal protein S10, ...
著者Mishra, S, Ahmed, T, Tyagi, A, Shi, J, Bhushan, S.
登録日2018-02-27
公開日2018-09-26
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structures of Mycobacterium smegmatis 70S ribosomes in complex with HPF, tmRNA, and P-tRNA.
Sci Rep, 8, 2018
5ZKF
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BU of 5zkf by Molmil
Crystal Structure of N-terminal Domain of Plasmodium vivax p43 in space group P21
分子名称: Aminoacyl tRNA Synthetase Complex-Interacting Multifunctional Protein p43
著者Gupta, S, Sharma, M, Harlos, K, Manickam, Y, Sharma, A.
登録日2018-03-23
公開日2019-04-24
最終更新日2020-03-11
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Crystal structures of the two domains that constitute the Plasmodium vivax p43 protein.
Acta Crystallogr D Struct Biol, 76, 2020
8OOC
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BU of 8ooc by Molmil
CryoEM Structure INO80core Hexasome complex Rvb core refinement state1
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Chromatin-remodeling ATPase Ino80, ...
著者Zhang, M, Jungblut, A, Hoffmann, T, Eustermann, S.
登録日2023-04-05
公開日2023-08-02
実験手法ELECTRON MICROSCOPY (2.93 Å)
主引用文献Hexasome-INO80 complex reveals structural basis of noncanonical nucleosome remodeling.
Science, 381, 2023
5ZH2
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BU of 5zh2 by Molmil
CRYSTAL STRUCTURE OF PfKRS WITH INHIBITOR CLADO-5
分子名称: (3R)-6,8-dihydroxy-3-{[(2R,6R)-6-methyloxan-2-yl]methyl}-3,4-dihydro-1H-2-benzopyran-1-one, 3[N-MORPHOLINO]PROPANE SULFONIC ACID, CHLORIDE ION, ...
著者Babbar, P, Malhotra, N, Sharma, M, Harlos, K, Reddy, D.S, Manickam, Y, Sharma, A.
登録日2018-03-11
公開日2018-06-27
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.66 Å)
主引用文献Specific Stereoisomeric Conformations Determine the Drug Potency of Cladosporin Scaffold against Malarial Parasite
J. Med. Chem., 61, 2018
4YCT
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BU of 4yct by Molmil
Endothiapepsin in complex with fragment 216
分子名称: 1,2-ETHANEDIOL, 4-(trifluoromethyl)benzenecarboximidamide, ACETATE ION, ...
著者Stieler, M, Heine, A, Klebe, G.
登録日2015-02-20
公開日2016-03-02
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.13 Å)
主引用文献Crystallographic Fragment Screening of an Entire Library
To Be Published
6D3W
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BU of 6d3w by Molmil
Chromosomal trehalose-6-phosphate phosphatase from P. aeruginosa
分子名称: 1,2-ETHANEDIOL, ACETIC ACID, CALCIUM ION, ...
著者Hofmann, A, Cross, M, Park, S.-Y.
登録日2018-04-17
公開日2018-05-09
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Trehalose 6-phosphate phosphatases of Pseudomonas aeruginosa.
FASEB J., 32, 2018
8OO6
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BU of 8oo6 by Molmil
Pol I bound to extended and displaced DNA section - closed conformation
分子名称: DNA polymerase I, Displaced primer, Extending Primer, ...
著者Botto, M, Borsellini, A, Lamers, M.H.
登録日2023-04-04
公開日2023-08-09
最終更新日2023-11-01
実験手法ELECTRON MICROSCOPY (4.3 Å)
主引用文献A four-point molecular handover during Okazaki maturation.
Nat.Struct.Mol.Biol., 30, 2023
4YD3
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BU of 4yd3 by Molmil
Endothiapepsin in complex with fragment 224
分子名称: 2-(1H-indol-3-yl)-N-[(1-methyl-1H-pyrrol-2-yl)methyl]ethanamine, ACETATE ION, DI(HYDROXYETHYL)ETHER, ...
著者Stieler, M, Heine, A, Klebe, G.
登録日2015-02-20
公開日2016-03-02
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.248 Å)
主引用文献Crystallographic Fragment Screening of an Entire Library
To Be Published
5ZKE
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BU of 5zke by Molmil
Crystal Structure of N-terminal Domain of Plasmodium vivax p43 in space group P212121
分子名称: Aminoacyl tRNA Synthetase Complex-Interacting Multifunctional Protein p43
著者Gupta, S, Sharma, M, Harlos, K, Manickam, Y, Sharma, A.
登録日2018-03-23
公開日2019-04-24
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.492 Å)
主引用文献Crystal structures of the two domains that constitute the Plasmodium vivax p43 protein.
Acta Crystallogr D Struct Biol, 76, 2020
5ZJQ
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BU of 5zjq by Molmil
Structure of AbdB/Exd complex bound to a 'Red14' DNA sequence
分子名称: DNA (5'-D(*GP*CP*AP*TP*GP*AP*TP*TP*TP*AP*TP*GP*AP*C)-3'), DNA (5'-D(*GP*TP*CP*AP*TP*AP*AP*AP*TP*CP*AP*TP*GP*C)-3'), Homeobox protein abdominal-B, ...
著者Baburajendran, N, Zeiske, T, Kaczynska, A, Mann, R, Honig, B, Shapiro, L, Palmer, A.G.
登録日2018-03-22
公開日2018-08-29
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.443 Å)
主引用文献Intrinsic DNA Shape Accounts for Affinity Differences between Hox-Cofactor Binding Sites.
Cell Rep, 24, 2018
5ZK4
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BU of 5zk4 by Molmil
The structure of DSZS acyltransferase with carrier protein
分子名称: DisA protein, DisD protein, N-[2-(acetylamino)ethyl]-N~3~-[(2R)-2-hydroxy-3,3-dimethyl-4-(phosphonooxy)butanoyl]-beta-alaninamide, ...
著者Miyanaga, A, Ouchi, R, Kudo, F, Eguchi, T.
登録日2018-03-23
公開日2018-06-13
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Structural basis of protein-protein interactions between a trans-acting acyltransferase and acyl carrier protein in polyketide disorazole biosynthesis
J. Am. Chem. Soc., 140, 2018
1SU9
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BU of 1su9 by Molmil
Reduced structure of the soluble domain of ResA
分子名称: Thiol-disulfide oxidoreductase resA
著者Crow, A, Acheson, R.M, Le Brun, N.E, Oubrie, A.
登録日2004-03-26
公開日2004-05-11
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structural Basis of Redox-coupled Protein Substrate Selection by the Cytochrome c Biosynthesis Protein ResA.
J.Biol.Chem., 279, 2004
8ORC
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BU of 8orc by Molmil
Mus Musculus Acetylcholinesterase in complex with AL237
分子名称: 1-[2-(dimethylamino)ethyl]-3-(2-methoxyphenyl)thiourea, 2,5,8,11,14,17,20,23-OCTAOXAPENTACOSAN-25-OL, 2-(2-METHOXYETHOXY)ETHANOL, ...
著者Ekstrom, F.E, Linusson, A.
登録日2023-04-13
公開日2024-04-24
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Enzyme Dynamics Determine Potency and Selectivity of Inhibitors Targeting Disease-Transmitting Mosquitoes
To Be Published
4CI5
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BU of 4ci5 by Molmil
Structural basis for GL479 a dual Peroxisome Proliferator-Activated Receptor gamma agonist
分子名称: 2-methyl-2-[4-[2-[4-[(E)-phenyldiazenyl]phenoxy]ethyl]phenoxy]propanoic acid, PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA
著者Santos, J.C, Bernardes, A, Polikarpov, I.
登録日2013-12-05
公開日2014-12-24
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Different binding and recognition modes of GL479, a dual agonist of Peroxisome Proliferator-Activated Receptor alpha / gamma.
J. Struct. Biol., 191, 2015
5ZQ6
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BU of 5zq6 by Molmil
SidE-Ubi-ADPr
分子名称: ADENOSINE-5'-DIPHOSPHATE, SidE, Ubiquitin
著者Wang, Y, Gao, A, Gao, P.
登録日2018-04-17
公開日2018-05-23
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.009 Å)
主引用文献Structural Insights into Non-canonical Ubiquitination Catalyzed by SidE.
Cell, 173, 2018
4Y44
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BU of 4y44 by Molmil
Endothiapepsin in complex with fragment 164
分子名称: 4,6-dimethyl-2-{[3-(morpholin-4-yl)propyl]amino}pyridine-3-carbonitrile, ACETATE ION, Endothiapepsin, ...
著者Krimmer, S.G, Heine, A, Klebe, G.
登録日2015-02-10
公開日2016-02-17
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.24 Å)
主引用文献Crystallographic Fragment Screening of an Entire Library
To Be Published
8OTP
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BU of 8otp by Molmil
Crystal structure of human carbonic anhydrase II with 1-cyclopropyl-6-fluoro-4-oxo-7-(4-(4-sulfamoylbenzoyl)piperazin-1-yl)-1,4-dihydroquinoline-3-carboxylic acid
分子名称: 1-cyclopropyl-6-fluoranyl-4-oxidanylidene-7-[4-(4-sulfamoylphenyl)carbonylpiperazin-1-yl]quinoline-3-carboxylic acid, Carbonic anhydrase 2, GLYCEROL, ...
著者Angeli, A, Ferraroni, M.
登録日2023-04-21
公開日2024-05-01
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Crystal structure of human carbonic anhydrase II with 1-cyclopropyl-6-fluoro-4-oxo-7-(4-(4-sulfamoylbenzoyl)piperazin-1-yl)-1,4-dihydroquinoline-3-carboxylic acid
To Be Published
4Y50
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BU of 4y50 by Molmil
Endothiapepsin in complex with fragment 81
分子名称: 1,2-ETHANEDIOL, 3-(dimethylamino)benzohydrazide, ACETATE ION, ...
著者Schiebel, J, Heine, A, Klebe, G.
登録日2015-02-11
公開日2016-03-02
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.32 Å)
主引用文献Crystallographic Fragment Screening of an Entire Library
To Be Published
8OUI
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BU of 8oui by Molmil
Complex of ASCT2 with Suppressyn
分子名称: ALANINE, Neutral amino acid transporter B(0), Suppressyn
著者Khare, S, Kumar, A, Reyes, N.
登録日2023-04-23
公開日2024-05-01
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.39 Å)
主引用文献Receptor-recognition and antiviral mechanisms of retrovirus-derived human proteins.
Nat.Struct.Mol.Biol., 2024
8OUB
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BU of 8oub by Molmil
The crystal structure of human carbonic anhydrase II with 1-cyclopropyl-6-fluoro-4-oxo-7-(4-((4-sulfamoylbenzyl)carbamoyl)piperazin-1-yl)-1,4-dihydroquinoline-3-carboxylic acid
分子名称: 1-cyclopropyl-6-fluoranyl-4-oxidanylidene-7-[4-[(4-sulfamoylphenyl)methylcarbamoyl]piperazin-1-yl]quinoline-3-carboxylic acid, Carbonic anhydrase 2, ZINC ION
著者Angeli, A, Ferraroni, M.
登録日2023-04-22
公開日2024-05-01
実験手法X-RAY DIFFRACTION (1.178 Å)
主引用文献The crystal structure of human carbonic anhydrase II with 1-cyclopropyl-6-fluoro-4-oxo-7-(4-((4-sulfamoylbenzyl)carbamoyl)piperazin-1-yl)-1,4-dihydroquinoline-3-carboxylic acid
To Be Published

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件を2024-07-17に公開中

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