5V11
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![BU of 5v11 by Molmil](/molmil-images/mine/5v11) | |
3KPY
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![BU of 3kpy by Molmil](/molmil-images/mine/3kpy) | Crystal Structure of hPNMT in Complex AdoHcy and 6-Chlorooxindole | 分子名称: | 6-chloro-1,3-dihydro-2H-indol-2-one, Phenylethanolamine N-methyltransferase, S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Drinkwater, N, Martin, J.L. | 登録日 | 2009-11-17 | 公開日 | 2010-09-29 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Fragment-based screening by X-ray crystallography, MS and isothermal titration calorimetry to identify PNMT (phenylethanolamine N-methyltransferase) inhibitors. Biochem.J., 431, 2010
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3KQV
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![BU of 3kqv by Molmil](/molmil-images/mine/3kqv) | Crystal Structure of hPNMT in Complex AdoHcy and Formanilide | 分子名称: | FORMANILIDE, Phenylethanolamine N-methyltransferase, S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Drinkwater, N, Martin, J.L. | 登録日 | 2009-11-17 | 公開日 | 2010-09-29 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Fragment-based screening by X-ray crystallography, MS and isothermal titration calorimetry to identify PNMT (phenylethanolamine N-methyltransferase) inhibitors. Biochem.J., 431, 2010
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3KPW
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![BU of 3kpw by Molmil](/molmil-images/mine/3kpw) | |
3KQP
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![BU of 3kqp by Molmil](/molmil-images/mine/3kqp) | |
3KQT
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3KPU
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![BU of 3kpu by Molmil](/molmil-images/mine/3kpu) | Crystal Structure of hPNMT in Complex AdoHcy and 4-quinolinol | 分子名称: | Phenylethanolamine N-methyltransferase, S-ADENOSYL-L-HOMOCYSTEINE, quinolin-4-ol | 著者 | Drinkwater, N, Martin, J.L. | 登録日 | 2009-11-17 | 公開日 | 2010-09-29 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Fragment-based screening by X-ray crystallography, MS and isothermal titration calorimetry to identify PNMT (phenylethanolamine N-methyltransferase) inhibitors. Biochem.J., 431, 2010
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3KR0
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![BU of 3kr0 by Molmil](/molmil-images/mine/3kr0) | |
3KR2
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![BU of 3kr2 by Molmil](/molmil-images/mine/3kr2) | |
3KQM
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![BU of 3kqm by Molmil](/molmil-images/mine/3kqm) | |
3KQS
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![BU of 3kqs by Molmil](/molmil-images/mine/3kqs) | |
3KPJ
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![BU of 3kpj by Molmil](/molmil-images/mine/3kpj) | |
3KQW
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![BU of 3kqw by Molmil](/molmil-images/mine/3kqw) | |
3KPV
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![BU of 3kpv by Molmil](/molmil-images/mine/3kpv) | Crystal Structure of hPNMT in Complex AdoHcy and Adenine | 分子名称: | ADENINE, Phenylethanolamine N-methyltransferase, S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Drinkwater, N, Martin, J.L. | 登録日 | 2009-11-17 | 公開日 | 2010-09-29 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Fragment-based screening by X-ray crystallography, MS and isothermal titration calorimetry to identify PNMT (phenylethanolamine N-methyltransferase) inhibitors. Biochem.J., 431, 2010
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3KQQ
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![BU of 3kqq by Molmil](/molmil-images/mine/3kqq) | |
3KQY
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![BU of 3kqy by Molmil](/molmil-images/mine/3kqy) | |
3KQO
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![BU of 3kqo by Molmil](/molmil-images/mine/3kqo) | |
3KR1
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![BU of 3kr1 by Molmil](/molmil-images/mine/3kr1) | |
3LH9
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![BU of 3lh9 by Molmil](/molmil-images/mine/3lh9) | |
3LH8
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![BU of 3lh8 by Molmil](/molmil-images/mine/3lh8) | |
3LHA
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![BU of 3lha by Molmil](/molmil-images/mine/3lha) | |
2XA7
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![BU of 2xa7 by Molmil](/molmil-images/mine/2xa7) | AP2 clathrin adaptor core in active complex with cargo peptides | 分子名称: | ADAPTOR-RELATED PROTEIN COMPLEX 2, ALPHA 2 SUBUNIT, AP-2 COMPLEX SUBUNIT BETA, ... | 著者 | Jackson, L.P, Kelly, B.T, McCoy, A.J, Evans, P.R, Owen, D.J. | 登録日 | 2010-03-29 | 公開日 | 2010-07-21 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | A Large Scale Conformational Change Couples Membrane Recruitment to Cargo Binding in the Ap2 Clathrin Adaptor Complex Cell(Cambridge,Mass.), 141, 2010
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3QBC
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![BU of 3qbc by Molmil](/molmil-images/mine/3qbc) | |
4DM3
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![BU of 4dm3 by Molmil](/molmil-images/mine/4dm3) | Crystal structure of human PNMT in complex adohcy, resorcinol and imidazole | 分子名称: | IMIDAZOLE, Phenylethanolamine N-methyltransferase, RESORCINOL, ... | 著者 | Nair, P.C, Malde, A.K, Mark, A.E. | 登録日 | 2012-02-06 | 公開日 | 2012-04-25 | 最終更新日 | 2018-01-24 | 実験手法 | X-RAY DIFFRACTION (2.4001 Å) | 主引用文献 | Missing fragments: detecting cooperative binding in fragment-based drug design. ACS Med Chem Lett, 3, 2012
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