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2WTW
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BU of 2wtw by Molmil
Aurora-A Inhibitor Structure (2nd crystal form)
分子名称: 4-{[9-CHLORO-7-(2,6-DIFLUOROPHENYL)-5H-PYRIMIDO[5,4-D][2]BENZAZEPIN-2-YL]AMINO}BENZOIC ACID, SERINE/THREONINE-PROTEIN KINASE 6 AURORA/IPL1-RELATED KINASE 1, BREAST TUMOR-AMPLIFIED KINASE, ...
著者Kosmopoulou, M, Bayliss, R.
登録日2009-09-24
公開日2010-01-26
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.302 Å)
主引用文献Crystal Structure of an Aurora-A Mutant that Mimics Aurora-B Bound to Mln8054: Insights Into Selectivity and Drug Design.
Biochem.J., 427, 2010
2WTV
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BU of 2wtv by Molmil
Aurora-A Inhibitor Structure
分子名称: 1,2-ETHANEDIOL, 4-{[9-CHLORO-7-(2,6-DIFLUOROPHENYL)-5H-PYRIMIDO[5,4-D][2]BENZAZEPIN-2-YL]AMINO}BENZOIC ACID, ACETATE ION, ...
著者Kosmopoulou, M, Bayliss, R.
登録日2009-09-22
公開日2010-01-26
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal Structure of an Aurora-A Mutant that Mimics Aurora-B Bound to Mln8054: Insights Into Selectivity and Drug Design.
Biochem.J., 427, 2010
2XOC
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BU of 2xoc by Molmil
C-terminal cysteine-rich domain of human CHFR bound to mADPr
分子名称: ADENINE, ADENOSINE-5'-DIPHOSPHATE, E3 UBIQUITIN-PROTEIN LIGASE CHFR, ...
著者Oberoi, J, Bayliss, R.
登録日2010-08-11
公開日2010-09-29
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献Structural Basis of Poly(Adp-Ribose) Recognition by the Multizinc Binding Domain of Checkpoint with Forkhead-Associated and Ring Domains (Chfr).
J.Biol.Chem., 285, 2010
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件を2024-10-16に公開中

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