5DQ2
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![BU of 5dq2 by Molmil](/molmil-images/mine/5dq2) | Endothiapepsin in complex with fragment 48 | 分子名称: | 1,2-ETHANEDIOL, Endothiapepsin, GLYCEROL, ... | 著者 | Radeva, N, Uehlein, M, Weiss, M, Heine, A, Klebe, G. | 登録日 | 2015-09-14 | 公開日 | 2016-09-28 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.514 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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5DR4
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![BU of 5dr4 by Molmil](/molmil-images/mine/5dr4) | Endothiapepsin in complex with fragment 231 | 分子名称: | 7-methyl-3,4-dihydro-2~{H}-pyrido[1,2-a]pyrimidin-3-ol, ACETATE ION, DIMETHYL SULFOXIDE, ... | 著者 | Schiebel, J, Heine, A, Klebe, G. | 登録日 | 2015-09-15 | 公開日 | 2016-09-28 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y35
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![BU of 4y35 by Molmil](/molmil-images/mine/4y35) | |
4Y37
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![BU of 4y37 by Molmil](/molmil-images/mine/4y37) | Endothiapepsin in complex with fragement 305 | 分子名称: | 4-chloro-2-methylthieno[2,3-d][1,2,3]diazaborinin-1(2H)-ol, ACETATE ION, Endothiapepsin, ... | 著者 | Krimmer, S.G, Heine, A, Klebe, G. | 登録日 | 2015-02-10 | 公開日 | 2016-02-17 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y3A
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![BU of 4y3a by Molmil](/molmil-images/mine/4y3a) | Endothiapepsin in complex with fragment 181 | 分子名称: | 1,2-ETHANEDIOL, 6-{[(3R,5S)-3,5-dimethylpiperidin-1-yl]methyl}-N,N-dimethyl-1,3,5-triazine-2,4-diamine, ACETATE ION, ... | 著者 | Ehrmann, F.R, Heine, A, Klebe, G. | 登録日 | 2015-02-10 | 公開日 | 2016-02-17 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.17 Å) | 主引用文献 | Crystallographic Fragment Sreening of an Entire Library To Be Published
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4Y3R
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![BU of 4y3r by Molmil](/molmil-images/mine/4y3r) | |
4Y3S
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![BU of 4y3s by Molmil](/molmil-images/mine/4y3s) | |
4Y47
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![BU of 4y47 by Molmil](/molmil-images/mine/4y47) | Endothiapepsin in complex with fragment 162 | 分子名称: | 4-oxo-N-[(1S)-1-(pyridin-3-yl)ethyl]-4-(thiophen-2-yl)butanamide, ACETATE ION, Endothiapepsin, ... | 著者 | Krimmer, S.G, Krug, M, Uehlein, M, Heine, A, Klebe, G. | 登録日 | 2015-02-10 | 公開日 | 2016-02-17 | 実験手法 | X-RAY DIFFRACTION (1.19 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y53
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![BU of 4y53 by Molmil](/molmil-images/mine/4y53) | Endothiapepsin in complex with fragment 54 | 分子名称: | 1,2-ETHANEDIOL, 3-(3,4-difluorophenyl)imidazo[2,1-c][1,2,4]triazine, Endothiapepsin, ... | 著者 | Radeva, N, Heine, A, Klebe, G. | 登録日 | 2015-02-11 | 公開日 | 2016-03-02 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.62 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y5C
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![BU of 4y5c by Molmil](/molmil-images/mine/4y5c) | |
4Y5M
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![BU of 4y5m by Molmil](/molmil-images/mine/4y5m) | Endothiapepsin in complex with fragment 328 | 分子名称: | 3-[(4E)-4-imino-5,6-dimethylfuro[2,3-d]pyrimidin-3(4H)-yl]-N,N-dimethylpropan-1-amine, DIMETHYL SULFOXIDE, Endothiapepsin, ... | 著者 | Fu, K, Heine, A, Klebe, G. | 登録日 | 2015-02-11 | 公開日 | 2016-03-02 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.28 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y3L
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![BU of 4y3l by Molmil](/molmil-images/mine/4y3l) | Endothiapepsin in complex with fragment 205 | 分子名称: | ACETATE ION, DIMETHYL SULFOXIDE, Endothiapepsin, ... | 著者 | Ehrmann, F.R, Huschmann, F.U, Heine, A, Klebe, G. | 登録日 | 2015-02-10 | 公開日 | 2016-02-17 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.16 Å) | 主引用文献 | Crystallographic Fragment Sreening of an Entire Library To Be Published
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4Y4B
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![BU of 4y4b by Molmil](/molmil-images/mine/4y4b) | Endothiapepsin in complex with fragment 323 | 分子名称: | 6,6,8-trimethyl-5,6-dihydro[1,3]dioxolo[4,5-g]quinoline, ACETATE ION, Endothiapepsin, ... | 著者 | Fu, K, Heine, A, Klebe, G. | 登録日 | 2015-02-10 | 公開日 | 2016-02-17 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.108 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y3E
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![BU of 4y3e by Molmil](/molmil-images/mine/4y3e) | Endothiapepsin in complex with fragment 5 | 分子名称: | 1H-isoindol-3-amine, ACETATE ION, DIMETHYL SULFOXIDE, ... | 著者 | Radeva, N, Uehlein, M, Weiss, M.S, Heine, A, Klebe, G. | 登録日 | 2015-02-10 | 公開日 | 2016-02-17 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y3Q
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![BU of 4y3q by Molmil](/molmil-images/mine/4y3q) | |
4Y3D
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![BU of 4y3d by Molmil](/molmil-images/mine/4y3d) | |
4Y4U
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![BU of 4y4u by Molmil](/molmil-images/mine/4y4u) | Endothiapepsin in complex with fragment 14 | 分子名称: | 1-(4-bromo-2-chlorophenyl)-3-methylthiourea, DI(HYDROXYETHYL)ETHER, Endothiapepsin, ... | 著者 | Radeva, N, Uehlein, M, Weiss, M.S, Heine, A, Klebe, G. | 登録日 | 2015-02-11 | 公開日 | 2016-03-02 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.754 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y4Z
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![BU of 4y4z by Molmil](/molmil-images/mine/4y4z) | Endothiapepsin in complex with fragment 73 | 分子名称: | (1Z)-N,N-diethylethanimidamide, 1,2-ETHANEDIOL, ACETATE ION, ... | 著者 | Schiebel, J, Heine, A, Klebe, G. | 登録日 | 2015-02-11 | 公開日 | 2016-03-02 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.48 Å) | 主引用文献 | Crystallographic Fragment Screening of an Entire Library To Be Published
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4Y58
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![BU of 4y58 by Molmil](/molmil-images/mine/4y58) | |
4Y5K
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![BU of 4y5k by Molmil](/molmil-images/mine/4y5k) | |
4YD5
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![BU of 4yd5 by Molmil](/molmil-images/mine/4yd5) | |
4YD7
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![BU of 4yd7 by Molmil](/molmil-images/mine/4yd7) | |
4Y5A
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![BU of 4y5a by Molmil](/molmil-images/mine/4y5a) | Endothiapepsin in complex with fragment 206 | 分子名称: | 1,2-ETHANEDIOL, 1-[5-(trifluoromethyl)furan-2-yl]methanamine, ACETATE ION, ... | 著者 | Ehrmann, F.R, Huschmann, F.U, Heine, A, Klebe, G. | 登録日 | 2015-02-11 | 公開日 | 2016-03-02 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Crystallographic Fragment Sreening of an Entire Library To Be Published
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4Y5L
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![BU of 4y5l by Molmil](/molmil-images/mine/4y5l) | |
4YCT
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![BU of 4yct by Molmil](/molmil-images/mine/4yct) | |