Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
9MSI
DownloadVisualize
BU of 9msi by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 T18N
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-28
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
6WW8
DownloadVisualize
BU of 6ww8 by Molmil
BRD4 Bromodomain 1 in complex with triple CDK4/6-PI3K-BET inhibitor
分子名称: 7-cyclopentyl-N,N-dimethyl-2-({4-[5-(morpholin-4-yl)-7-oxo-7H-thieno[3,2-b]pyran-3-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide, Bromodomain-containing protein 4
著者Vann, K.R, Kutateladze, T.G.
登録日2020-05-08
公開日2020-08-26
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.302 Å)
主引用文献A triple action CDK4/6-PI3K-BET inhibitor with augmented cancer cell cytotoxicity.
Cell Discov, 6, 2020
6VBA
DownloadVisualize
BU of 6vba by Molmil
Structure of human Uracil DNA Glycosylase (UDG) bound to Aurintricarboxylic acid (ATA)
分子名称: 3,3'-[(3-carboxy-4-oxocyclohexa-2,5-dien-1-ylidene)methylene]bis(6-hydroxybenzoic acid), Uracil-DNA glycosylase
著者Moiani, D, Arvai, A.S, Tainer, J.A.
登録日2019-12-18
公開日2021-03-03
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献An effective human uracil-DNA glycosylase inhibitor targets the open pre-catalytic active site conformation.
Prog.Biophys.Mol.Biol., 163, 2021
3FAA
DownloadVisualize
BU of 3faa by Molmil
Crystal structure of TGFbRI complexed with a 2-aminoimidazole inhibitor
分子名称: N-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1H-imidazol-2-yl]acetamide, PHOSPHATE ION, TGF-beta receptor type-1
著者Boriack-Sjodin, P.A, Fitch, C.
登録日2008-11-16
公開日2009-01-27
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (3.35 Å)
主引用文献2-Aminoimidazoles inhibitors of TGF-beta receptor 1.
Bioorg.Med.Chem.Lett., 19, 2009
7TAB
DownloadVisualize
BU of 7tab by Molmil
G-925 bound to the SMARCA4 (BRG1) Bromodomain
分子名称: 2-(6-amino-5-phenylpyridazin-3-yl)phenol, Isoform 4 of Transcription activator BRG1
著者Tang, Y, Poy, F, Taylor, A.M, Cochran, A.G, Bellon, S.F.
登録日2021-12-20
公開日2022-08-17
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.16 Å)
主引用文献GNE-064: A Potent, Selective, and Orally Bioavailable Chemical Probe for the Bromodomains of SMARCA2 and SMARCA4 and the Fifth Bromodomain of PBRM1.
J.Med.Chem., 65, 2022
7TD9
DownloadVisualize
BU of 7td9 by Molmil
G-059 bound to the SMARCA4 (BRG1) Bromodomain
分子名称: 4-phenyl-5H-pyridazino[4,3-b]indol-3-amine, Isoform 4 of Transcription activator BRG1
著者Tang, Y, Poy, F, Taylor, A.M, Cochran, A.G, Bellon, S.F.
登録日2021-12-30
公開日2022-08-17
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献GNE-064: A Potent, Selective, and Orally Bioavailable Chemical Probe for the Bromodomains of SMARCA2 and SMARCA4 and the Fifth Bromodomain of PBRM1.
J.Med.Chem., 65, 2022
6IBO
DownloadVisualize
BU of 6ibo by Molmil
Catalytic deficiency of O-GlcNAc transferase leads to X-linked intellectual disability
分子名称: (2S,3R,4R,5S,6R)-3-(acetylamino)-4,5-dihydroxy-6-(hydroxymethyl)tetrahydro-2H-thiopyran-2-yl [(2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl]methyl dihydrogen diphosphate, ALA-VAL-SER-ARG-ALA, PHOSPHATE ION, ...
著者Gundogdu, M, van Aalten, D.M.F.
登録日2018-11-30
公開日2019-07-24
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Catalytic deficiency of O-GlcNAc transferase leads to X-linked intellectual disability.
Proc.Natl.Acad.Sci.USA, 116, 2019
5V84
DownloadVisualize
BU of 5v84 by Molmil
CECR2 in complex with Cpd6 (6-allyl-N,2-dimethyl-7-oxo-N-(1-(1-phenylethyl)piperidin-4-yl)-6,7-dihydro-1H-pyrrolo[2,3-c]pyridine-4-carboxamide)
分子名称: Cat eye syndrome critical region protein 2, N,2-dimethyl-7-oxo-N-{1-[(1S)-1-phenylethyl]piperidin-4-yl}-6-(prop-2-en-1-yl)-6,7-dihydro-1H-pyrrolo[2,3-c]pyridine-4- carboxamide, SULFATE ION
著者Murray, J.M, Kiefer, J.R, Jayaran, H, Bellon, S, Boy, F.
登録日2017-03-21
公開日2017-06-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献GNE-886: A Potent and Selective Inhibitor of the Cat Eye Syndrome Chromosome Region Candidate 2 Bromodomain (CECR2).
ACS Med Chem Lett, 8, 2017
1B7I
DownloadVisualize
BU of 1b7i by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 K61R
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-30
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
1B7K
DownloadVisualize
BU of 1b7k by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 R47H
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
6AME
DownloadVisualize
BU of 6ame by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 M21A
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
8MSI
DownloadVisualize
BU of 8msi by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 N14SQ44T
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
1MSJ
DownloadVisualize
BU of 1msj by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 T15V
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
7AME
DownloadVisualize
BU of 7ame by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 T15A
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
1MSI
DownloadVisualize
BU of 1msi by Molmil
STRUCTURE OF ANTIFREEZE GLYCOPROTEIN QAE(HPLC 12)
分子名称: TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12
著者Jia, Z, Deluca, C.I, Chao, H, Davies, P.L.
登録日1996-10-08
公開日1997-12-24
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Structural basis for the binding of a globular antifreeze protein to ice.
Nature, 384, 1996
8AME
DownloadVisualize
BU of 8ame by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 N14SA16H
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
1B7J
DownloadVisualize
BU of 1b7j by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 V20A
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-30
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
1EKL
DownloadVisualize
BU of 1ekl by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 E35K
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-21
公開日1999-04-29
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
7UI7
DownloadVisualize
BU of 7ui7 by Molmil
CryoEM structure of LARGE1 from C2 reconstruction
分子名称: MANGANESE (II) ION, Xylosyl- and glucuronyltransferase LARGE1
著者Schnicker, N.J, Joseph, S, Campbell, K.P.
登録日2022-03-28
公開日2023-03-08
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献CryoEM structure of LARGE1 from C2 reconstruction
To Be Published
3AME
DownloadVisualize
BU of 3ame by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 Q9TQ44T
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
1JAB
DownloadVisualize
BU of 1jab by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 T18S
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
2SPG
DownloadVisualize
BU of 2spg by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 T15S
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-21
公開日1999-04-28
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
2AME
DownloadVisualize
BU of 2ame by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 N14Q
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-18
公開日1999-04-30
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
2JIA
DownloadVisualize
BU of 2jia by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 K61I
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999
4AME
DownloadVisualize
BU of 4ame by Molmil
TYPE III ANTIFREEZE PROTEIN ISOFORM HPLC 12 T18A
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Graether, S.P, Deluca, C.I, Baardsnes, J, Hill, G.A, Davies, P.L, Jia, Z.
登録日1999-01-24
公開日1999-04-29
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Quantitative and qualitative analysis of type III antifreeze protein structure and function.
J.Biol.Chem., 274, 1999

224931

件を2024-09-11に公開中

PDB statisticsPDBj update infoContact PDBjnumon