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2RK8
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BU of 2rk8 by Molmil
The Structure of rat cytosolic PEPCK in complex with phosphonoformate
分子名称: DI(HYDROXYETHYL)ETHER, FORMIC ACID, MANGANESE (II) ION, ...
著者Sullivan, S.M, Stiffin, R.M, Carlson, G.M, Holyoak, T.
登録日2007-10-16
公開日2008-01-29
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Differential Inhibition of Cytosolic PEPCK by Substrate Analogues. Kinetic and Structural Characterization of Inhibitor Recognition.
Biochemistry, 47, 2008
2RKA
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BU of 2rka by Molmil
The Structure of rat cytosolic PEPCK in complex with phosphoglycolate
分子名称: 2-PHOSPHOGLYCOLIC ACID, MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, ...
著者Sullivan, S.M, Stiffin, R.M, Carlson, G.M, Holyoak, T.
登録日2007-10-16
公開日2008-01-29
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Differential Inhibition of Cytosolic PEPCK by Substrate Analogues. Kinetic and Structural Characterization of Inhibitor Recognition.
Biochemistry, 47, 2008
2RKE
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BU of 2rke by Molmil
The Structure of rat cytosolic PEPCK in complex with sulfoacetate.
分子名称: MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, cytosolic [GTP], ...
著者Sullivan, S.M, Stiffin, R.M, Carlson, G.M, Holyoak, T.
登録日2007-10-16
公開日2008-01-29
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Differential Inhibition of Cytosolic PEPCK by Substrate Analogues. Kinetic and Structural Characterization of Inhibitor Recognition.
Biochemistry, 47, 2008
2RK7
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BU of 2rk7 by Molmil
The Structure of rat cytosolic PEPCK in complex with oxalate
分子名称: MANGANESE (II) ION, OXALATE ION, Phosphoenolpyruvate carboxykinase, ...
著者Sullivan, S.M, Stiffin, R.M, Carlson, G.M, Holyoak, T.
登録日2007-10-16
公開日2008-01-29
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Differential Inhibition of Cytosolic PEPCK by Substrate Analogues. Kinetic and Structural Characterization of Inhibitor Recognition.
Biochemistry, 47, 2008
4YWD
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BU of 4ywd by Molmil
Structure of rat cytosolic pepck in complex with 2,3-Pyridine dicarboxylic acid
分子名称: MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, cytosolic [GTP], ...
著者Balan, M.D, Johnson, T.A, Mcleod, M.J, Lotosky, W.R, Holyoak, T.
登録日2015-03-20
公開日2015-09-23
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Inhibition and Allosteric Regulation of Monomeric Phosphoenolpyruvate Carboxykinase by 3-Mercaptopicolinic Acid.
Biochemistry, 54, 2015
4YW8
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BU of 4yw8 by Molmil
Structure of rat cytosolic pepck in complex with 3-mercaptopicolinic acid
分子名称: 1,2-ETHANEDIOL, 3-sulfanylpyridine-2-carboxylic acid, MANGANESE (II) ION, ...
著者Balan, M.D, Johnson, T.A, Mcleod, M.J, Lotosky, W.R, Holyoak, T.
登録日2015-03-20
公開日2015-09-23
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Inhibition and Allosteric Regulation of Monomeric Phosphoenolpyruvate Carboxykinase by 3-Mercaptopicolinic Acid.
Biochemistry, 54, 2015
4YW9
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BU of 4yw9 by Molmil
Structure of rat cytosolic pepck in complex with 3-mercaptopicolinic acid and GTP
分子名称: 3-sulfanylpyridine-2-carboxylic acid, GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, ...
著者Balan, M.D, Johnson, T.A, Mcleod, M.J, Lotosky, W.R, Holyoak, T.
登録日2015-03-20
公開日2015-09-23
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Inhibition and Allosteric Regulation of Monomeric Phosphoenolpyruvate Carboxykinase by 3-Mercaptopicolinic Acid.
Biochemistry, 54, 2015
4YWB
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BU of 4ywb by Molmil
Structure of rat cytosolic pepck in complex with 3-mercaptopicolinic acid and oxalic acid
分子名称: 3-sulfanylpyridine-2-carboxylic acid, CHLORIDE ION, MANGANESE (II) ION, ...
著者Balan, M.D, Johnson, T.A, Lotosky, W.R, Mcleod, M.J, Holyoak, T.
登録日2015-03-20
公開日2015-09-23
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Inhibition and Allosteric Regulation of Monomeric Phosphoenolpyruvate Carboxykinase by 3-Mercaptopicolinic Acid.
Biochemistry, 54, 2015
3DT2
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BU of 3dt2 by Molmil
The structure of rat cytosolic PEPCK in complex with oxalate and GTP
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, OXALATE ION, ...
著者Sullivan, S.M, Holyoak, T.
登録日2008-07-14
公開日2008-08-26
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Enzymes with lid-gated active sites must operate by an induced fit mechanism instead of conformational selection.
Proc.Natl.Acad.Sci.Usa, 105, 2008
3DT7
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BU of 3dt7 by Molmil
The structure of rat cytosolic PEPCK in complex with beta-sulfopyruvate and GTP
分子名称: 2-ETHOXYETHANOL, GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, ...
著者Sullivan, S.M, Holyoak, T.
登録日2008-07-14
公開日2008-08-26
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Enzymes with lid-gated active sites must operate by an induced fit mechanism instead of conformational selection.
Proc.Natl.Acad.Sci.Usa, 105, 2008
3DT4
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BU of 3dt4 by Molmil
The structure of rat cytosolic PEPCK in complex with oxalate and GTP
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, OXALATE ION, ...
著者Sullivan, S.M, Holyoak, T.
登録日2008-07-14
公開日2008-08-26
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Enzymes with lid-gated active sites must operate by an induced fit mechanism instead of conformational selection.
Proc.Natl.Acad.Sci.Usa, 105, 2008
3DTB
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BU of 3dtb by Molmil
The structure of rat cytosolic PEPCK in complex with phosphoglycolate and GDP
分子名称: 2-PHOSPHOGLYCOLIC ACID, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, BICARBONATE ION, ...
著者Sullivan, S.M, Holyoak, T.
登録日2008-07-14
公開日2008-08-26
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Enzymes with lid-gated active sites must operate by an induced fit mechanism instead of conformational selection.
Proc.Natl.Acad.Sci.Usa, 105, 2008
3MOF
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BU of 3mof by Molmil
The structure of rat cytosolic PEPCK mutant A467G in complex with oxalate and GTP
分子名称: 1,2-ETHANEDIOL, GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, ...
著者Johnson, T.A, Holyoak, T.
登録日2010-04-22
公開日2010-06-02
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Increasing the conformational entropy of the Omega-loop lid domain in phosphoenolpyruvate carboxykinase impairs catalysis and decreases catalytic fidelity .
Biochemistry, 49, 2010
3MOE
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BU of 3moe by Molmil
The structure of rat cytosolic PEPCK mutant A467G in complex with Beta-Sulfopyruvate and GTP
分子名称: 1,2-ETHANEDIOL, GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, ...
著者Johnson, T.A, Holyoak, T.
登録日2010-04-22
公開日2010-06-02
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Increasing the conformational entropy of the Omega-loop lid domain in phosphoenolpyruvate carboxykinase impairs catalysis and decreases catalytic fidelity .
Biochemistry, 49, 2010
3MOH
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BU of 3moh by Molmil
The structure of rat cytosolic PEPCK mutant A467G in complex with phosphoglycolate and GDP
分子名称: 1,2-ETHANEDIOL, 2-PHOSPHOGLYCOLIC ACID, GUANOSINE-5'-DIPHOSPHATE, ...
著者Johnson, T.A, Holyoak, T.
登録日2010-04-22
公開日2010-06-02
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Increasing the conformational entropy of the Omega-loop lid domain in phosphoenolpyruvate carboxykinase impairs catalysis and decreases catalytic fidelity .
Biochemistry, 49, 2010
3N25
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BU of 3n25 by Molmil
The structure of muscle pyruvate kinase in complex with proline, pyruvate, and Mn2+
分子名称: 1,2-ETHANEDIOL, GLYCEROL, MANGANESE (II) ION, ...
著者Fenton, A.W, Johnson, T.A, Holyoak, T.
登録日2010-05-17
公開日2010-07-28
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献The pyruvate kinase model system, a cautionary tale for the use of osmolyte perturbations to support conformational equilibria in allostery.
Protein Sci., 19, 2010
7L3V
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BU of 7l3v by Molmil
PEPCK MMQX structure 120ms post-mixing with oxaloacetic acid
分子名称: CARBON DIOXIDE, GUANOSINE-5'-DIPHOSPHATE, MANGANESE (II) ION, ...
著者Clinger, J.A, Moreau, D.W, McLeod, M.J, Holyoak, T, Thorne, R.E.
登録日2020-12-18
公開日2021-10-13
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献Millisecond mix-and-quench crystallography (MMQX) enables time-resolved studies of PEPCK with remote data collection.
Iucrj, 8, 2021
7L36
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BU of 7l36 by Molmil
PEPCK steady-state structure with Mn and GTP
分子名称: CHLORIDE ION, GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, ...
著者Clinger, J.A, Moreau, D.W, McLeod, M.J, Holyoak, T, Thorne, R.E.
登録日2020-12-17
公開日2021-10-13
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献Millisecond mix-and-quench crystallography (MMQX) enables time-resolved studies of PEPCK with remote data collection.
Iucrj, 8, 2021
7L3M
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BU of 7l3m by Molmil
PEPCK MMQX structure 40ms post-mixing with oxaloacetic acid
分子名称: CARBON DIOXIDE, GUANOSINE-5'-DIPHOSPHATE, MANGANESE (II) ION, ...
著者Clinger, J.A, Moreau, D.W, McLeod, M.J, Holyoak, T, Thorne, R.E.
登録日2020-12-18
公開日2021-10-13
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献Millisecond mix-and-quench crystallography (MMQX) enables time-resolved studies of PEPCK with remote data collection.
Iucrj, 8, 2021
4GMZ
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BU of 4gmz by Molmil
Structure of rat cytosolic PEPCK Ld_2g in complex with Beta-Sulfopyruvate and GTP
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, ...
著者Johnson, T.A, Holyoak, T.
登録日2012-08-16
公開日2013-07-03
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献The {Omega}-loop lid domain of phosphoenolpyruvate carboxykinase is essential for catalytic function.
Biochemistry, 51, 2012
4GMM
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BU of 4gmm by Molmil
Structure of rat cytosolic PEPCK Ld_1g in complex with Beta-Sulfopyruvate and GTP
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, ...
著者Johnson, T.A, Holyoak, T.
登録日2012-08-16
公開日2013-07-03
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.736 Å)
主引用文献The {Omega}-loop lid domain of phosphoenolpyruvate carboxykinase is essential for catalytic function.
Biochemistry, 51, 2012
4GMW
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BU of 4gmw by Molmil
Structure of rat cytosolic PEPCK Ld_1g in complex with PEP and GDP
分子名称: GUANOSINE-5'-DIPHOSPHATE, MANGANESE (II) ION, PHOSPHOENOLPYRUVATE, ...
著者Johnson, T.A, Holyoak, T.
登録日2012-08-16
公開日2013-07-03
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献The {Omega}-loop lid domain of phosphoenolpyruvate carboxykinase is essential for catalytic function.
Biochemistry, 51, 2012
4GMU
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BU of 4gmu by Molmil
Structure of rat cytosolic PEPCK Ld_1g in complex with oxalate and GTP
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, OXALATE ION, ...
著者Johnson, T.A, Holyoak, T.
登録日2012-08-16
公開日2013-07-03
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献The {Omega}-loop lid domain of phosphoenolpyruvate carboxykinase is essential for catalytic function.
Biochemistry, 51, 2012
4GNQ
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BU of 4gnq by Molmil
Structure of rat cytosolic PEPCK Ld_3g in complex with oxalate and GTP
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, OXALATE ION, ...
著者Johnson, T.A, Holyoak, T.
登録日2012-08-17
公開日2013-07-03
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献The {Omega}-loop lid domain of phosphoenolpyruvate carboxykinase is essential for catalytic function.
Biochemistry, 51, 2012
4GNM
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BU of 4gnm by Molmil
Structure of rat cytosolic PEPCK Ld_2g in complex with oxalate and GTP
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, OXALATE ION, ...
著者Johnson, T.A, Holyoak, T.
登録日2012-08-17
公開日2013-07-03
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The {Omega}-loop lid domain of phosphoenolpyruvate carboxykinase is essential for catalytic function.
Biochemistry, 51, 2012

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