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3QN7
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BU of 3qn7 by Molmil
Potent and selective bicyclic peptide inhibitor (UK18) of human urokinase-type plasminogen activator(uPA)
分子名称: 1,3,5-tris(bromomethyl)benzene, Bicyclic peptide inhibitor, Urokinase-type plasminogen activator
著者Angelini, A, Cendron, L, Touati, J, Winter, G, Zanotti, G, Heinis, C.
登録日2011-02-08
公開日2012-02-15
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Bicyclic peptide inhibitor reveals large contact interface with a protease target
Acs Chem.Biol., 7, 2012
6ZH9
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BU of 6zh9 by Molmil
Ternary complex CR3022 H11-H4 and RBD (SARS-CoV-2)
分子名称: CR3022 Light chain, CR3022 heavy, Nanobody H11-H4, ...
著者Naismith, J.H, Mikolajek, H, Le Bas, A.
登録日2020-06-21
公開日2020-09-02
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3.31 Å)
主引用文献Neutralizing nanobodies bind SARS-CoV-2 spike RBD and block interaction with ACE2.
Nat.Struct.Mol.Biol., 27, 2020
2QIL
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BU of 2qil by Molmil
TOXIC SHOCK SYNDROME TOXIN-1 AT 2.07 A RESOLUTION
分子名称: TOXIC SHOCK SYNDROME TOXIN-1
著者Acharya, K.R, Papageorgiou, A.C.
登録日1997-03-27
公開日1997-08-12
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献The refined crystal structure of toxic shock syndrome toxin-1 at 2.07 A resolution.
J.Mol.Biol., 260, 1996
1BOY
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BU of 1boy by Molmil
EXTRACELLULAR REGION OF HUMAN TISSUE FACTOR
分子名称: HUMAN TISSUE FACTOR
著者Boys, C.W.G, Tuddenham, E.G.D, Harlos, K.
登録日1996-01-11
公開日1996-06-10
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structure of the extracellular region of human tissue factor.
Nature, 370, 1994
1D0N
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BU of 1d0n by Molmil
THE CRYSTAL STRUCTURE OF CALCIUM-FREE EQUINE PLASMA GELSOLIN.
分子名称: HORSE PLASMA GELSOLIN
著者Burtnick, L.D, Robinson, R, Li, C.
登録日1999-09-13
公開日1999-09-15
最終更新日2019-08-14
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The crystal structure of plasma gelsolin: implications for actin severing, capping, and nucleation.
Cell(Cambridge,Mass.), 90, 1997
1QIL
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BU of 1qil by Molmil
INACTIVE MUTANT TOXIC SHOCK SYNDROME TOXIN-1 AT 2.5 A
分子名称: TOXIC SHOCK SYNDROME TOXIN-1
著者Acharya, K.R, Papageorgiou, A.C.
登録日1997-03-27
公開日1997-08-12
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of a biologically inactive mutant of toxic shock syndrome toxin-1 at 2.5 A resolution.
Protein Sci., 5, 1996
1STE
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BU of 1ste by Molmil
STAPHYLOCOCCAL ENTEROTOXIN C2 FROM STAPHYLOCOCCUS AUREUS
分子名称: STAPHYLOCOCCAL ENTEROTOXIN C2, ZINC ION
著者Acharya, K.R, Papageorgiou, A.C.
登録日1995-08-21
公開日1996-12-23
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of the superantigen enterotoxin C2 from Staphylococcus aureus reveals a zinc-binding site.
Structure, 3, 1995
1UNS
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BU of 1uns by Molmil
IDENTIFICATION OF A SECONDARY ZINC-BINDING SITE IN STAPHYLOCOCCAL ENTEROTOXIN C2: IMPLICATIONS FOR SUPERANTIGEN RECOGNITION
分子名称: ENTEROTOXIN TYPE C-2, ZINC ION
著者Papageorgiou, A.C, Baker, M.D, McLeod, J.D, Goda, S, Sansom, D.M, Tranter, H.S, Acharya, K.R.
登録日2003-09-15
公開日2003-11-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Identification of a Secondary Zinc-Binding Site in Staphylococcal Enterotoxin C2: Implications for Superantigen Recognition
J.Biol.Chem., 279, 2004
1QRZ
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BU of 1qrz by Molmil
CATALYTIC DOMAIN OF PLASMINOGEN
分子名称: PLASMINOGEN
著者Peisach, E, Wang, J, de los Santos, T, Reich, E, Ringe, D.
登録日1999-06-16
公開日1999-10-14
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of the proenzyme domain of plasminogen.
Biochemistry, 38, 1999
1UOT
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BU of 1uot by Molmil
HUMAN CD55 DOMAINS 3 & 4
分子名称: COMPLEMENT DECAY-ACCELERATING FACTOR
著者Williams, P, Chaudhry, Y, Goodfellow, I.G, Billington, J, Spiller, B, Evans, D.J, Lea, S.M.
登録日2003-09-23
公開日2003-09-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Mapping Cd55 Function. The Structure of Two Pathogen-Binding Domains at 1.7 A
J.Biol.Chem., 278, 2003
2AMV
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BU of 2amv by Molmil
THE STRUCTURE OF GLYCOGEN PHOSPHORYLASE B WITH AN ALKYL-DIHYDROPYRIDINE-DICARBOXYLIC ACID
分子名称: 2,3-DICARBOXY-4-(2-CHLORO-PHENYL)-1-ETHYL-5-ISOPROPOXYCARBONYL-6-METHYL-PYRIDINIUM, GLYCEROL, PROTEIN (GLYCOGEN PHOSPHORYLASE), ...
著者Zographos, S.E, Oikonomakos, N.G, Johnson, L.N.
登録日1998-10-13
公開日1998-10-21
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The structure of glycogen phosphorylase b with an alkyldihydropyridine-dicarboxylic acid compound, a novel and potent inhibitor.
Structure, 5, 1997
8A2F
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BU of 8a2f by Molmil
Crystal Structure of Ljunganvirus 1 2A protein
分子名称: 2A protein
著者von Castelmur, E, Zhu, L, Wang, X, Fry, E, Ren, J, Perrakis, A, Stuart, D.I.
登録日2022-06-03
公開日2023-06-14
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献Structural plasticity of 2A proteins in the Parechovirus family
To Be Published
8A2E
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BU of 8a2e by Molmil
Crystal Structure of Human Parechovirus 3 2A protein
分子名称: 2A protein, GLYCEROL, SULFATE ION
著者von Castelmur, E, Zhu, L, wang, X, Fry, E, Ren, J, Perrakis, A, Stuart, D.I.
登録日2022-06-03
公開日2023-06-14
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献Structural plasticity of 2A proteins in the Parechovirus family.
To Be Published
8A2G
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BU of 8a2g by Molmil
Crystal structure of Sebokelevirus 2A2 protein
分子名称: 1,2-ETHANEDIOL, 2A2 protein, TETRAETHYLENE GLYCOL
著者Zhu, L, Von Castelmur, E, Whang, X, Ren, J, Fry, E, Perrakis, A, Stuart, D.I.
登録日2022-06-03
公開日2023-06-14
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Structural plasticity of 2A proteins in the Parechovirus family
to be published
1NOJ
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BU of 1noj by Molmil
COMPLEX OF GLYCOGEN PHOSPHORYLASE WITH A TRANSITION STATE ANALOGUE NOJIRIMYCIN TETRAZOLE AND PHOSPHATE IN THE T STATE
分子名称: GLYCOGEN PHOSPHORYLASE, NOJIRIMYCINE TETRAZOLE, PHOSPHATE ION, ...
著者Johnson, L.N, Mitchell, E.P.
登録日1996-03-12
公開日1996-07-11
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Ternary complex crystal structures of glycogen phosphorylase with the transition state analogue nojirimycin tetrazole and phosphate in the T and R states.
Biochemistry, 35, 1996
1NOK
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BU of 1nok by Molmil
COMPLEX OF GLYCOGEN PHOSPHORYLASE WITH A TRANSITION STATE ANALOGUE NOJIRIMYCIN TETRAZOLE AND PHOSPHATE IN THE T STATE
分子名称: GLYCOGEN PHOSPHORYLASE, NOJIRIMYCINE TETRAZOLE, PYRIDOXAL-5'-PHOSPHATE
著者Johnson, L.N, Mitchell, E.P.
登録日1996-03-12
公開日1996-07-11
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Ternary complex crystal structures of glycogen phosphorylase with the transition state analogue nojirimycin tetrazole and phosphate in the T and R states.
Biochemistry, 35, 1996
1PYG
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BU of 1pyg by Molmil
STRUCTURAL BASIS FOR THE ACTIVATION OF GLYCOGEN PHOSPHORYLASE B BY ADENOSINE MONOPHOSPHATE
分子名称: ADENOSINE MONOPHOSPHATE, GLYCOGEN PHOSPHORYLASE B, PYRIDOXAL-5'-DIPHOSPHATE
著者Sprang, S.
登録日1992-07-07
公開日1994-01-31
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.87 Å)
主引用文献Structural basis for the activation of glycogen phosphorylase b by adenosine monophosphate.
Science, 254, 1991
1PKM
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BU of 1pkm by Molmil
THE REFINED THREE-DIMENSIONAL STRUCTURE OF CAT MUSCLE (M1) PYRUVATE KINASE, AT A RESOLUTION OF 2.6 ANGSTROMS
分子名称: M1 PYRUVATE KINASE
著者Allen, S.C, Muirhead, H.
登録日1995-07-13
公開日1995-10-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Refined three-dimensional structure of cat-muscle (M1) pyruvate kinase at a resolution of 2.6 A.
Acta Crystallogr.,Sect.D, 52, 1996
2GPN
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BU of 2gpn by Molmil
100 K STRUCTURE OF GLYCOGEN PHOSPHORYLASE AT 2.0 ANGSTROMS RESOLUTION
分子名称: GLYCOGEN PHOSPHORYLASE B
著者Gregoriou, M, Noble, M.E.M, Watson, K.A, Garman, E.F, Krulle, T.M, De La Fuente, C, Fleet, G.W.J, Oikonomakos, N.G, Johnson, L.N.
登録日1998-03-26
公開日1998-07-01
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献The structure of a glycogen phosphorylase glucopyranose spirohydantoin complex at 1.8 A resolution and 100 K: the role of the water structure and its contribution to binding.
Protein Sci., 7, 1998
2Y0S
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BU of 2y0s by Molmil
Crystal structure of Sulfolobus shibatae RNA polymerase in P21 space group
分子名称: DNA-DIRECTED RNA POLYMERASE, DNA-DIRECTED RNA POLYMERASE SUBUNIT A'', DNA-DIRECTED RNA POLYMERASE SUBUNIT D, ...
著者Wojtas, M, Peralta, B, Ondiviela, M, Mogni, M, Bell, S.D, Abrescia, N.G.A.
登録日2010-12-07
公開日2011-02-16
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Archaeal RNA polymerase: the influence of the protruding stalk in crystal packing and preliminary biophysical analysis of the Rpo13 subunit.
Biochem. Soc. Trans., 39, 2011
6Z2M
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BU of 6z2m by Molmil
H11-D4, SARS-CoV-2 RBD, CR3022 ternary complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CR3022 antibody, Spike glycoprotein, ...
著者Naismith, J.H, Ren, J, Zhou, D, Zhao, Y, Stuart, D.I.
登録日2020-05-17
公開日2020-06-03
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.71 Å)
主引用文献Structural characterisation of a nanobody derived from a naive library that neutralises SARS-CoV-2
To Be Published
6YZ7
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BU of 6yz7 by Molmil
H11-D4, SARS-CoV-2 RBD, CR3022 ternary complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Antibody Cr3022, Antibody light chain, ...
著者Naismith, J.H, Ren, J, Zhou, D, Zhao, Y, Stuart, D.I.
登録日2020-05-06
公開日2020-06-03
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structural characterisation of a nanobody derived from a naive library that neutralises SARS-CoV-2
To Be Published, 2020
1A6S
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BU of 1a6s by Molmil
M-DOMAIN FROM GAG POLYPROTEIN OF ROUS SARCOMA VIRUS, NMR, 20 STRUCTURES
分子名称: GAG POLYPROTEIN
著者Mcdonnell, J.M, Fushman, D, Cahill, S.M, Zhou, W, Wolven, A, Wilson, C.B, Nelle, T.D, Resh, M.D, Wills, J, Cowburn, D.
登録日1998-03-02
公開日1998-10-14
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure and dynamics of the bioactive retroviral M domain from Rous sarcoma virus
J.Mol.Biol., 279, 1998
1A8I
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BU of 1a8i by Molmil
SPIROHYDANTOIN INHIBITOR OF GLYCOGEN PHOSPHORYLASE
分子名称: BETA-D-GLUCOPYRANOSE SPIROHYDANTOIN, GLYCOGEN PHOSPHORYLASE B
著者Gregoriou, M, Noble, M.E.M, Watson, K.A, Garman, E.F, Krulle, T.M, De La Fuente, C, Fleet, G.W.J, Oikonomakos, N.G, Johnson, L.N.
登録日1998-03-25
公開日1998-07-01
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (1.78 Å)
主引用文献The structure of a glycogen phosphorylase glucopyranose spirohydantoin complex at 1.8 A resolution and 100 K: the role of the water structure and its contribution to binding.
Protein Sci., 7, 1998
1AXR
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COOPERATIVITY BETWEEN HYDROGEN-BONDING AND CHARGE-DIPOLE INTERACTIONS IN THE INHIBITION OF BETA-GLYCOSIDASES BY AZOLOPYRIDINES: EVIDENCE FROM A STUDY WITH GLYCOGEN PHOSPHORYLASE B
分子名称: 4,5,6-TRIHYDROXY-7-HYDROXYMETHYL-4,5,6,7-TETRAHYDRO-1H-[1,2,3]TRIAZOLO[1,5-A]PYRIDIN-8-YLIUM, GLYCOGEN PHOSPHORYLASE, PHOSPHATE ION, ...
著者Oikonomakos, N.G, Heightman, T.D.
登録日1997-10-20
公開日1998-01-28
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Cooperative interactions of the catalytic nucleophile and the catalytic acid in the inhibition of beta-glycosidases. Calculations and their validation by comparative kinetic and structural studies of the inhibition of glycogen phosphorylase b.
HELV.CHIM.ACTA, 81, 1998

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